BDBM50130268 CHEMBL329383::N-(2,5-Dibromo-3-fluoro-phenyl)-4-methoxy-3-piperazin-1-yl-benzenesulfonamide::N-(2,5-dibromo-3-fluorophenyl)-4-methoxy-3-(piperazin-1-yl)benzenesulfonamide::SB-357134
SMILES COc1ccc(cc1N1CCNCC1)S(=O)(=O)Nc1cc(Br)cc(F)c1Br
InChI Key InChIKey=BLWHAZZXRHTFJE-UHFFFAOYSA-N
Data 23 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 23 hits for monomerid = 50130268
Affinity DataKi: 2.60nMAssay Description:Antagonist activity at human recombinant 5HT6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity towards human 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity against 5 Hydroxy tryptamine 6 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity towards [3H]LSD-labeled human 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-LSD from human cloned 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity against human 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: <3.98E+3nMAssay Description:Compound was evaluated for binding affinity against human cloned 5-hydroxytryptamine 1D receptor in CHO cells using [3H]5-HT as the radioligandMore data for this Ligand-Target Pair
Affinity DataKi: <3.98E+3nMAssay Description:Compound was evaluated for binding affinity against human cloned 5-HT2B receptor in HEK 293 cells using [3H]5-HT as the radioligandMore data for this Ligand-Target Pair
Affinity DataKi: <3.98E+3nMAssay Description:Compound was evaluated for binding affinity against human cloned 5-hydroxytryptamine 1B receptor in CHO cells using [3H]5-HT as the radioligandMore data for this Ligand-Target Pair
Affinity DataKi: <5.01E+3nMAssay Description:Compound was evaluated for binding affinity against human cloned 5-hydroxytryptamine 2C receptor in HEK 293 cells using [3H]mesulergine as the radiol...More data for this Ligand-Target Pair
Affinity DataKi: <5.01E+3nMAssay Description:Compound was evaluated for binding affinity against Dopamine receptor D3 in CHO cells using [125I]iodosulpiride as the radioligandMore data for this Ligand-Target Pair
Affinity DataKi: <5.01E+3nMAssay Description:Compound was evaluated for the binding affinity against human cloned 5-hydroxytryptamine 4 receptor in HeLa cells using [3H]-LSD as the radioligandMore data for this Ligand-Target Pair
Affinity DataKi: <5.01E+3nMAssay Description:Compound was evaluated for binding affinity against Dopamine receptor D2 in CHO cells using [125I]iodosulpiride as the radioligandMore data for this Ligand-Target Pair
Affinity DataKi: <6.31E+3nMAssay Description:Compound was evaluated for binding affinity against human cloned 5-hydroxytryptamine 1A receptor in HEK 293 cells using [3H]8-OH-DPAT as the radiolig...More data for this Ligand-Target Pair
Affinity DataKi: <7.94E+3nMAssay Description:Compound was evaluated for binding affinity against human cloned 5-hydroxytryptamine 2A receptor in HEK 293 cells using [3H]ketanserin as the radioli...More data for this Ligand-Target Pair
Affinity DataKi: <7.94E+3nMAssay Description:Compound was evaluated for binding affinity against Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-hydroxytryptamine 7 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+4nMAssay Description:Compound was evaluated for binding affinity against human cloned 5-hydroxytryptamine 1F receptor in CHO cells using [3H]-5-HT as the radioligandMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+4nMAssay Description:Compound was evaluated for binding affinity against human cloned 5-hydroxytryptamine 1E receptor in CHO cells using [3H]5-HT as the radioligandMore data for this Ligand-Target Pair