BDBM154577 K03859 (2)

SMILES CN1CCN(Cc2ccc(NC(=O)c3cccc4cc(Oc5cc(NC(C)=O)ncn5)ccc34)cc2C(F)(F)F)CC1

InChI Key InChIKey=MZZJNOOADWVFPD-UHFFFAOYSA-N

Data  8 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 154577   

TargetCyclin-dependent kinase 2(Human)
University of Oxford

LigandPNGBDBM154577(K03859 (2))
Affinity DataIC50: >1.00E+4nMT: 303.15°CAssay Description:For IC50 measurements, a 384-well microtiter plate contained 8-point serial dilutions of inhibitors and 16-point serial dilutions of staurosporine as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2 [F80T](Human)
University of Oxford

LigandPNGBDBM154577(K03859 (2))
Affinity DataIC50:  7.10E+3nMT: 303.15°CAssay Description:For IC50 measurements, a 384-well microtiter plate contained 8-point serial dilutions of inhibitors and 16-point serial dilutions of staurosporine as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2 [F80M](Human)
University of Oxford

LigandPNGBDBM154577(K03859 (2))
Affinity DataIC50: >1.00E+4nMT: 303.15°CAssay Description:For IC50 measurements, a 384-well microtiter plate contained 8-point serial dilutions of inhibitors and 16-point serial dilutions of staurosporine as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2 [C118L,A144C](Human)
University of Oxford

LigandPNGBDBM154577(K03859 (2))
Affinity DataIC50: >1.00E+4nMT: 303.15°CAssay Description:For IC50 measurements, a 384-well microtiter plate contained 8-point serial dilutions of inhibitors and 16-point serial dilutions of staurosporine as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2 [C118I](Human)
University of Oxford

LigandPNGBDBM154577(K03859 (2))
Affinity DataIC50: >1.00E+4nMT: 303.15°CAssay Description:For IC50 measurements, a 384-well microtiter plate contained 8-point serial dilutions of inhibitors and 16-point serial dilutions of staurosporine as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2 [A144C](Human)
University of Oxford

LigandPNGBDBM154577(K03859 (2))
Affinity DataIC50: >1.00E+4nMT: 303.15°CAssay Description:For IC50 measurements, a 384-well microtiter plate contained 8-point serial dilutions of inhibitors and 16-point serial dilutions of staurosporine as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2 [A144G](Human)
University of Oxford

LigandPNGBDBM154577(K03859 (2))
Affinity DataIC50: >1.00E+4nMT: 303.15°CAssay Description:For IC50 measurements, a 384-well microtiter plate contained 8-point serial dilutions of inhibitors and 16-point serial dilutions of staurosporine as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2 [C118L](Human)
University of Oxford

LigandPNGBDBM154577(K03859 (2))
Affinity DataIC50: >1.00E+4nMT: 303.15°CAssay Description:For IC50 measurements, a 384-well microtiter plate contained 8-point serial dilutions of inhibitors and 16-point serial dilutions of staurosporine as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed