BDBM197128 US9216182, 1.74
SMILES CC(C)N1CCN(CC1)C(=O)OC1CCN(CC1)c1ccn2cc(C)nc2c1
InChI Key InChIKey=XAQBWJISZRMNHF-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 197128
Affinity DataKi: 0.400nMAssay Description:The potency of compounds of the invention as H3 receptor antagonists can be assessed by measuring the blockade of (R)-alpha-methylhistamine-mediated ...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMpH: 7.5Assay Description:The affinity of compounds of the invention to the H3 receptor can be assessed by measuring displacement of binding of the radioligand [3H]-N-α-Methy...More data for this Ligand-Target Pair