BDBM263263 2,5-dimethyl-1-[4-(2-oxo-2h-pyridin-1-ylmethyl)-benzyl]-1h-pyrrole-3-carboxylicacid (1-amino-isoquinolin-6-ylmethyl)-amide::US9533987, example 44
SMILES Cc1cc(C(=O)NCc2ccc3c(N)nccc3c2)c(C)n1Cc1ccc(Cn2ccccc2=O)cc1
InChI Key InChIKey=GBMUDCZNXCHCOS-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 263263
Affinity DataIC50: 7.09E+3nMAssay Description:Human serine protease enzymes plasmin, thrombin, trypsin, Factor Xa and Factor XIIa were assayed for enzymatic activity using an appropriate fluoroge...More data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMAssay Description:Plasma kallikrein inhibitory activity in vitro was determined using standard published methods (see e.g. Johansen et al., Int. J. Tiss. Reac. 1986, 8...More data for this Ligand-Target Pair