BDBM270908 3-(benzenesulfonyl)-6-(cyclohex-1-en-1-yl)-1H-pyrrolo[3,2-b]pyridin-2-amine::US10059713, Example 25
SMILES Nc1[nH]c2cc(cnc2c1S(=O)(=O)c1ccccc1)C1=CCCCC1
InChI Key InChIKey=PARBIUXQJSUUPC-UHFFFAOYSA-N
Data 1 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 270908
Affinity DataEC50: 46nMAssay Description:GPR43 agonist/PAM activity was determined by measuring changes in intracellular calcium levels using a Ca2+ sensitive fluorescent dye. The changes in...More data for this Ligand-Target Pair