BDBM356607 N-(2-Fluorobenzyl)-3-[3-(3-{[(methylamino)carbonyl]amino}phenyl)imidazo[1,2-b]pyridazin-7-yl]benzamide::US10213427, Example 96::US10813930, Ex. No. 96

SMILES CNC(=O)Nc1cccc(c1)-c1cnc2cc(cnn12)-c1cccc(c1)C(=O)NCc1ccccc1F

InChI Key InChIKey=NAIAJRBRVXKICR-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 356607   

TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 356607BDBM356607(N-(2-Fluorobenzyl)-3-[3-(3-{[(methylamino)carbonyl...)
Affinity DataIC50: 25nMAssay Description:FGFR3 Enzymatic Assay The inhibitor potency of compounds of the invention was measured in an enzyme assay that measures peptide phosphorylation using...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2021
Entry Details
US Patent

TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 356607BDBM356607(N-(2-Fluorobenzyl)-3-[3-(3-{[(methylamino)carbonyl...)
Affinity DataIC50: 25nMAssay Description:The inhibitor potency of compounds of the invention was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent