BDBM357921 US10214536, Compound 288

SMILES CC(C)c1ccc2oc3nc(N)c(C(=O)Nc4nnn[nH]4)cc3c(=O)c2c1

InChI Key InChIKey=JDIHMNISRGRMDY-UHFFFAOYSA-N

Data  1 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 357921   

TargetSerine/threonine-protein kinase TBK1(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 357921BDBM357921(US10214536, Compound 288)
Affinity DataIC50: 180nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent
PDB3D3D Structure (crystal)