BDBM412510 5-fluoro-N-(5-(5-((3-fluoropyridin-2- yl)oxy)-2-methylphenyl)pyrazin-2- yl)-4-methylnicotinamide::US10399967, Compound 143

SMILES Cc1ccc(Oc2ncccc2F)cc1-c1cnc(NC(=O)c2cncc(F)c2C)cn1

InChI Key InChIKey=GVRPMKMPHLFNQQ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 412510   

TargetInterleukin-2(Human)
Prcl Research

US Patent
LigandChemical structure of BindingDB Monomer ID 412510BDBM412510(US10399967, Compound 143 | 5-fluoro-N-(5-(5-((3-fl...)
Affinity DataIC50: 35nMAssay Description:Human peripheral blood mononuclear cells (PBMCs) are prepared from heparinized human blood by separation over a Ficoll density gradient.PBMCs are sti...More data for this Ligand-Target Pair
Ligand InfoSimilars
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Date in BDB:
7/27/2020
Entry Details
US Patent