BDBM426493 US10543183, Compound SB742881::US10669296, Compound SB742881::US10945978, Compound 25

SMILES CC(CCOc1cccc(CC(O)=O)c1)N(CC(c1ccccc1)c1ccccc1)Cc1cccc(c1Cl)C(F)(F)F

InChI Key InChIKey=ZLJZDYOBXVOTSA-UHFFFAOYSA-N

Data  6 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 426493   

TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
The Rockefeller University

US Patent
LigandPNGBDBM426493(US10543183, Compound SB742881 | US10669296, Compou...)
Affinity DataEC50:  74nMAssay Description:As used herein, reference to the activity of an LXR agonist at LXRα and LXRβ refer to the activity as measured using the ligand sensing ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
The Rockefeller University

US Patent
LigandPNGBDBM426493(US10543183, Compound SB742881 | US10669296, Compou...)
Affinity DataEC50:  25nMAssay Description:As used herein, reference to the activity of an LXR agonist at LXRα and LXRβ refer to the activity as measured using the ligand sensing ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
The Rockefeller University

US Patent
LigandPNGBDBM426493(US10543183, Compound SB742881 | US10669296, Compou...)
Affinity DataEC50:  25nMAssay Description:As used herein, reference to the activity of an LXR agonist at LXRα and LXRβ refer to the activity as measured using the ligand sensing ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
The Rockefeller University

US Patent
LigandPNGBDBM426493(US10543183, Compound SB742881 | US10669296, Compou...)
Affinity DataEC50:  25nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
The Rockefeller University

US Patent
LigandPNGBDBM426493(US10543183, Compound SB742881 | US10669296, Compou...)
Affinity DataEC50:  74nMAssay Description:As used herein, reference to the activity of an LXR agonist at LXRα and LXRβ refer to the activity as measured using the ligand sensing ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
The Rockefeller University

US Patent
LigandPNGBDBM426493(US10543183, Compound SB742881 | US10669296, Compou...)
Affinity DataEC50:  74nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails US Patent