BDBM481764 3-(4-chlorophenethyl)-5-((5- methyl-4-oxopyrido[3,4- d]pyrimidin-3(4H)- yl)methyl)-1,3,4-oxadiazol- 2(3H)-one::US10913742, Example 6
SMILES Cc1cncc2ncn(Cc3nn(CCc4ccc(Cl)cc4)c(=O)o3)c(=O)c12
InChI Key InChIKey=KMNAEBCIGPEECD-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 481764
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 13nMAssay Description:The IC50 (effective concentration) of compounds on the human and rat TRPA1 channels were determined using a FLIPR Tetra instrument. CHO cells express...More data for this Ligand-Target Pair