BDBM50139402 (4-{2-[2-(2-Methyl-piperidin-1-yl)-ethyl]-benzofuran-5-yl}-phenyl)-morpholin-4-yl-methanone::CHEMBL161130

SMILES CC1CCCCN1CCc1cc2cc(ccc2o1)-c1ccc(cc1)C(=O)N1CCOCC1

InChI Key InChIKey=AWAROEZGWJEDHM-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50139402   

TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50139402((4-{2-[2-(2-Methyl-piperidin-1-yl)-ethyl]-benzofur...)
Affinity DataKi:  3nMAssay Description:Binding potency was determined by displacement of [3H]-N-alpha-methyl histamine from cloned human histamine H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50139402((4-{2-[2-(2-Methyl-piperidin-1-yl)-ethyl]-benzofur...)
Affinity DataKi:  3nMAssay Description:Binding potency was determined by displacement of [3H]N-alpha-methyl histamine from cloned human histamine H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50139402((4-{2-[2-(2-Methyl-piperidin-1-yl)-ethyl]-benzofur...)
Affinity DataKi:  13nMAssay Description:Binding potency was determined by displacement of [3H]N-alpha-methyl histamine from histamine H3 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50139402((4-{2-[2-(2-Methyl-piperidin-1-yl)-ethyl]-benzofur...)
Affinity DataKi:  14nMAssay Description:Binding potency was determined by displacement of [3H]-N-alpha-methyl histamine from histamine H3 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed