BDBM50145054 (E)-1-(6-Hydroxy-4,7-dimethoxy-benzofuran-5-yl)-3-(3-methoxy-phenyl)-propenone::1-(6-hydroxy-4,7-dimethoxybenzofuran-5-yl)-3-(3-methoxyphenyl)prop-2-en-1-one::CHEMBL76543

SMILES COc1cccc(\C=C\C(=O)c2c(O)c(OC)c3occc3c2OC)c1

InChI Key InChIKey=NZQFVFZKSNUANG-BQYQJAHWSA-N

Data  1 Kd  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50145054   

TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Institute Of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50145054((E)-1-(6-Hydroxy-4,7-dimethoxy-benzofuran-5-yl)-3-...)
Affinity DataKd:  800nMAssay Description:Dissociation constant for the blockage of voltage-gated potassium channel subunit Kv1.3 in human lymphocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Institute Of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50145054((E)-1-(6-Hydroxy-4,7-dimethoxy-benzofuran-5-yl)-3-...)
Affinity DataEC50:  900nMAssay Description:Inhibition in Kv1.3 expressed in human Jurkat cells by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Institute Of Medical Research Biotechnology Centre

Curated by ChEMBL
LigandPNGBDBM50145054((E)-1-(6-Hydroxy-4,7-dimethoxy-benzofuran-5-yl)-3-...)
Affinity DataEC50:  800nMAssay Description:Inhibition in Kv1.3 expressed in human L929 by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed