BDBM50150755 CHEMBL3775270
SMILES CCCCn1c2ncn(CC)c2c(=O)[nH]c1=O
InChI Key InChIKey=MJFNWOLXWYRXQS-UHFFFAOYSA-N
Data 7 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50150755
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of GST-tagged human BRD4 bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of GST-tagged human BRDT bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of GST-tagged human BRD3 bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of human BRD3 bromodomain2 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of GST-tagged human BRD4 bromodomain2 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of GST-tagged human BRD2 bromodomain2 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 1.88E+4nMAssay Description:Inhibition of GST-tagged human BRD2 bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair