BDBM50241256 CHEMBL233000::N-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)benzamide
SMILES O=C(Nc1sc2CCCCc2c1C#N)c1ccccc1
InChI Key InChIKey=OKFHWMLGUMHKFC-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50241256
TargetRAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataKd: >4.00E+4nMAssay Description:Binding affinity to human AKT3More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of JNK3More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human AKT3More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant full length JNK1alpha1More data for this Ligand-Target Pair
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of human truncated JNK3More data for this Ligand-Target Pair
Affinity DataIC50: >1.58E+4nMAssay Description:Inhibition of mitogen-activated protein kinase p38alphaMore data for this Ligand-Target Pair
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb
Curated by ChEMBL
Bristol-Myers Squibb
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair