BDBM50260102 CHEMBL4059589

SMILES CN1[C@H](c2cc(ccc2C1=O)-c1c(C)noc1C)c1ccccc1

InChI Key InChIKey=CHAKVDDAHQGTLR-IBGZPJMESA-N

Data  1 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50260102   

TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50260102(CHEMBL4059589)
Affinity DataIC50:  14nMAssay Description:Inhibition of GST-tagged BRD4 (unknown origin) using biotinylated acetyl-histone H4 peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair