BDBM50299866 CHEMBL578153::N-(1-(3-(5-Methyl-1H-imidazol-1-yl)propylamino)-2-nitrovinyl)-4-(trifluoromethyl)benzenamine::US8772508, 6
SMILES Cc1cncn1CCCN=C(C[N+]([O-])=O)Nc1ccc(cc1)C(F)(F)F
InChI Key InChIKey=GPQHOIQTHKOAGY-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50299866
Affinity DataKi: 34nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
Affinity DataKi: 34nM IC50: 430nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair