BDBM50484648 CHEMBL1940046

SMILES COc1ccc(cc1OC)S(=O)(=O)N(Cc1ccc2OC(C)(C)Cc2c1)c1ccccc1

InChI Key InChIKey=SRYXTPSNXWOGLW-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50484648   

TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50484648(CHEMBL1940046)
Affinity DataIC50:  306nMAssay Description:Inhibition of HIF1 in human LN229 cells after 1 hr preincubation under hypoxic condition measured after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed