BDBM50504782 CHEMBL4567799

SMILES CN1CC(Cn2c3CCNC(=O)c3c3ccccc23)CC1=O

InChI Key InChIKey=UERBETVZEWZRSL-UHFFFAOYSA-N

Data  1 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50504782   

TargetBromodomain-containing protein 4(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50504782(CHEMBL4567799)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of GST-tagged BRD4 BD1 (49 to 170 residues) (unknown origin) using streptavidin-D2 biotinylated tetra-acetylated histone H4 peptide as sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed