BDBM50522007 CHEMBL4446542

SMILES COc1cc(OC)cc(c1)C(=O)Nc1nc(C2CCC2)c(s1)N1CCN(C)CC1

InChI Key InChIKey=MEUYKBTYBNRUHB-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50522007   

TargetTransient receptor potential cation channel subfamily V member 4(Human)
Astellas Pharma

Curated by ChEMBL

LigandBDBM50522007(CHEMBL4446542)Copy SMILESCopy InChI

Affinity DataIC50:  84nMAssay Description:Inhibition of human TRPV4 expressed in HEK293 cells assessed as reduction in Ca2+ influx incubated for 30 mins by Fluo4-AM dye basedMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI