BDBM50551477 CHEMBL4741051

SMILES CN1CC(CC1=O)c1ccc(cc1)S(=O)(=O)N1CCCCC1

InChI Key InChIKey=FJZVEOQSYSYUQK-UHFFFAOYSA-N

Data  1 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50551477   

TargetBromodomain-containing protein 4(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50551477(CHEMBL4741051)
Affinity DataIC50:  1.44E+5nMAssay Description:Inhibition of GST-tagged BRD4-BD1 (49 to 170 residues) (unknown origin) using Histone H4 peptide as substrate incubated for 1.5 hrs by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed