BDBM791693 (R)-2-(2-(((4-((8-chloro-1,7-naphthyridin-2-yl)amino)cyclohexyl)methyl)amino)pyrimidin-5-yl)-N-(oxetan-3-yl)propanamide::US12544374, Compound C54

SMILES C[C@@H](C(=O)NC1COC1)c1cnc(NCC2CCC(Nc3ccc4ccnc(Cl)c4n3)CC2)nc1

InChI Key InChIKey=ONGLVKUUEUYJSJ-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 791693   

LigandChemical structure of BindingDB Monomer ID 791693BDBM791693((R)-2-(2-(((4-((8-chloro-1,7-naphthyridin-2-yl)ami...)
Affinity DataIC50: 75nMAssay Description:This cell based assay measures the ability of compounds to inhibit the constitutive cAMP activity of GPR6 receptor expressed in CHO-K1 cells. CHO cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/22/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 791693BDBM791693((R)-2-(2-(((4-((8-chloro-1,7-naphthyridin-2-yl)ami...)
Affinity DataIC50: 115nMAssay Description:The ELISA portion of the assay is performed in a black Maxisorp 96-well plate that is coated overnight at 4° C. with 100 uL/well of the cell lysa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/22/2026
Entry Details
US Patent