Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with Target = 'Bromodomain testis-specific protein [21-137]'
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205431BDBM205431((6S+2S)-PEG1 (7))
Affinity DataKi:  0.290nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205453BDBM205453(MTI (35))
Affinity DataKi:  0.560nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205431BDBM205431((6S+2S)-PEG1 (7))
Affinity DataIC50: 0.574nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205433BDBM205433((6S+2S)-PEG3 (9))
Affinity DataIC50: 0.878nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205434BDBM205434((6S+2S)-PEG4 (10))
Affinity DataIC50: 1.09nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205435BDBM205435((6S+2S)-PEG7 (11))
Affinity DataIC50: 1.59nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205432BDBM205432((6S+2S)-PEG2 (8))
Affinity DataIC50: 1.84nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205430BDBM205430((6S+2S)-PEG0 (6))
Affinity DataIC50: 2.36nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205439BDBM205439(6S+IBET-PEG3 (20))
Affinity DataIC50: 5.78nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205441BDBM205441(6S+IBET-PEG7 (22))
Affinity DataIC50: 6.10nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205440BDBM205440(6S+IBET-PEG4 (21))
Affinity DataIC50: 6.20nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205438BDBM205438(6S+IBET-PEG2 (19))
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205437BDBM205437(6S+IBET-PEG1 (18))
Affinity DataIC50: 12.1nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205442BDBM205442(2S+IBET-PEG7 (28))
Affinity DataIC50: 13.2nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205452BDBM205452(IBETx2-PEG7 (34))
Affinity DataIC50: 13.6nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205447BDBM205447(2S+IBET-PEG4 (27))
Affinity DataIC50: 21.7nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205454BDBM205454(2S+IBET-PEG2 (25))
Affinity DataIC50: 23.2nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205446BDBM205446(2S+IBET-PEG3 (26))
Affinity DataIC50: 31.7nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205444BDBM205444(2S+IBET-PEG1 (24))
Affinity DataIC50: 40.3nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205429BDBM205429( (R)-JQ1 (3) | US9320741, (R)-JQ1 | US10407441, Co...)
Affinity DataKd:  47nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205451BDBM205451(IBETx2-PEG4 (33))
Affinity DataIC50: 60.2nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205450BDBM205450(IBETx2-PEG3 (32))
Affinity DataIC50: 64.6nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205445BDBM205445(IBETx2-PEG2 (31))
Affinity DataIC50: 123nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205436BDBM205436(6S+IBET-PEG0 (17))
Affinity DataIC50: 148nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205448BDBM205448(IBETx2-PEG0 (29))
Affinity DataIC50: 203nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205449BDBM205449(IBETx2-PEG1 (30))
Affinity DataIC50: 203nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205443BDBM205443(2S+IBET-PEG0 (23))
Affinity DataIC50: 596nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed