Compile Data Set for Download or QSAR
Report error Found 297 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4 [44-164]'
TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425214BDBM425214(US10519177, Compound P-0092 | benzyl 4-[[5-(3,5- d...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425213BDBM425213(US10519177, Compound P-0091)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425212BDBM425212(US10519177, Compound P-0090)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425211BDBM425211(US10519177, Compound P-0089)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425206BDBM425206(US10519177, Compound P-0084)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425207BDBM425207(US10519177, Compound P-0085 | 4-[3-[dicyclopropyl-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425200BDBM425200(US10519177, Compound P-0080)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425199BDBM425199(US10519177, Compound P-0079)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425202BDBM425202(US10519177, Compound P-0081)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425230BDBM425230(US10519177, Compound P-0109)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425229BDBM425229(US10519177, Compound P-0108)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425232BDBM425232(US10519177, Compound P-0111 | 3,5-dimethyl-4-[3-(1...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425231BDBM425231(US10519177, Compound P-0110 | 4-[1-(benzenesulfony...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425226BDBM425226(US10519177, Compound P-0104 | 4-[1-(benzenesulfony...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425225BDBM425225(US10519177, Compound P-0103 | 4-[1-cyclopentyl- su...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425228BDBM425228(US10519177, Compound P-0106 | 1-[4-[[5-(3,5- dimet...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425227BDBM425227(US10519177, Compound P-0105 | 4-[1-cyclopentylsulf...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425223BDBM425223(US10519177, Compound P-0101 | (4,4- difluorocycloh...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425220BDBM425220(US10519177, Compound P-0098)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425246BDBM425246(US10519177, Compound P-0125 | 4-[3-(1-ethylpyrazol...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425245BDBM425245(US10519177, Compound P-0124 | 4-[1-(benzenesulfony...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425248BDBM425248(US10519177, Compound P-0127 | 4-[3-(1-allylpyrazol...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425247BDBM425247(US10519177, Compound P-0126 | 4-[3-(1-allylpyrazol...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425242BDBM425242(US10519177, Compound P-0121 | 4-[1-(2-fluorophenyl...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425241BDBM425241(US10519177, Compound P-0120 | 1-[4[[5-(3,5- dimeth...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425244BDBM425244(US10519177, Compound P-0123 | 4-[1-(4-fluorophenyl...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425243BDBM425243(US10519177, Compound P-0122 | 4-[1-(3-fluorophenyl...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425238BDBM425238(US10519177, Compound P-0117 | 4-[[5-(3,5- dimethyl...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425237BDBM425237(US10519177, Compound P-0116 | 4-[3-[(1-ethylsulfon...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425239BDBM425239(US10519177, Compound P-0118 | 4-[3-[1-(4,4- difluo...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425234BDBM425234(US10519177, Compound P-0113)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425233BDBM425233(US10519177, Compound P-0112 | 4-[1-cyclopentyl- su...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425236BDBM425236(US10519177, Compound P-0115 | [4-[[5-(3,5- dimethy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425235BDBM425235(US10519177, Compound P-0114 | 4-[[5-(3,5- dimethyl...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425262BDBM425262(US10519177, Compound P-0141)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425261BDBM425261(US10519177, Compound P-0140 | 4-[3-(1-allylpyrazol...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425264BDBM425264(US10519177, Compound P-0143)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425263BDBM425263(US10519177, Compound P-0142)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425258BDBM425258(US10519177, Compound P-0137 | 4-[3-(1-allylpyrazol...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425257BDBM425257(US10519177, Compound P-0136 | 4-[3-[1-(difluoro- m...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425260BDBM425260(US10519177, Compound P-0139 | 4-[3-(1-allylpyrazol...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425259BDBM425259(US10519177, Compound P-0138 | 4-[3-(1-allylpyrazol...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425254BDBM425254(US10519177, Compound P-0133 | 4-[1-cyclopentylsulf...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425253BDBM425253(US10519177, Compound P-0132 | 4-[3-[1-(difluoromet...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425256BDBM425256(US10519177, Compound P-0135 | 4-[3-[1-(difluoro- m...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425255BDBM425255(US10519177, Compound P-0134 | 4-[1-cyclobutyl- sul...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425250BDBM425250(US10519177, Compound P-0129 | 4-[3-(1-allylpyrazol...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425249BDBM425249(US10519177, Compound P-0128 | 4-[3-(1-allylpyrazol...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425252BDBM425252(US10519177, Compound P-0131 | 4-[1-(benzenesulfony...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetBromodomain-containing protein 4 [44-164](Human)
Plexxikon

US Patent
LigandChemical structure of BindingDB Monomer ID 425278BDBM425278(US10519177, Compound P-0157)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding of compounds of formula (I) with bromodomain 2, 3 4 was assessed using Alphascreen binding assay. The inhibition of the interaction between b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

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