Compile Data Set for Download or QSAR
Report error Found 73 Enz. Inhib. hit(s) with Target = 'Carnitine O-palmitoyltransferase 1, muscle isoform'
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50403039(CHEMBL2216778)
Affinity DataIC50: 16nMAssay Description:Inhibition of CPT1B (unknown origin) in KB cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50403040(CHEMBL2216779)
Affinity DataIC50: 21nMAssay Description:Inhibition of CPT1B (unknown origin) in KB cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403039(CHEMBL2216778)
Affinity DataIC50: 30nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403029(CHEMBL2216792)
Affinity DataIC50: 40nMAssay Description:Inhibition of rat CPT1B expressed in intact Saccharomyces cerevisiae using [methyl-3H]carnitine by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403040(CHEMBL2216779)
Affinity DataIC50: 55nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403037(CHEMBL2216774)
Affinity DataIC50: 130nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403041(CHEMBL2216776)
Affinity DataIC50: 150nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50403031(CHEMBL2216771)
Affinity DataIC50: 160nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403038(CHEMBL2216777)
Affinity DataIC50: 180nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50403028(CHEMBL2216769)
Affinity DataIC50: 360nMAssay Description:Inhibition of CPT1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50260111(CHEBI:15531 | MALONYL-COENZYME A)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM80613(SMR000674573 | cid_9926449 | 1-(2,3,4-Trimethoxy-b...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of CPT1A in rat myocardiumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM80613(SMR000674573 | cid_9926449 | 1-(2,3,4-Trimethoxy-b...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of rat CPT1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50122839([3-Carboxy-2-(3-tetradecyl-ureido)-propyl]-trimeth...)
Affinity DataIC50: 1.45E+3nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101594([3-Carboxy-2-(decane-1-sulfonylamino)-propyl]-trim...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50046145(2-[6-hydroxy-4,4-dimethyl-6-pentadecyl-(2R,6S)-1,4...)
Affinity DataKi:  2.80E+3nMAssay Description:Compound was evaluated for its ability to inhibit carnitine palmitoyltransferase I activity in intact mitochondria from rat heartMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101604([3-Carboxy-2-(dodecane-1-sulfonylamino)-propyl]-tr...)
Affinity DataIC50: 3.40E+3nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50403039(CHEMBL2216778)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101598([3-Carboxy-2-(dodecane-1-sulfonylamino)-propyl]-tr...)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50403038(CHEMBL2216777)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101589([3-Carboxy-2-(nonylaminosulphonyl-amino)-propyl]-t...)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50122839([3-Carboxy-2-(3-tetradecyl-ureido)-propyl]-trimeth...)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50403032(CHEMBL2216785)
Affinity DataIC50: 5.44E+3nMAssay Description:Inhibition of CPT1B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101591([3-Carboxy-2-(undecylaminosulphonyl-amino)-propyl]...)
Affinity DataIC50: 5.80E+3nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101591([3-Carboxy-2-(undecylaminosulphonyl-amino)-propyl]...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50403043(CHEMBL2216780)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101600([3-Carboxy-2-(undecylaminosulphonyl-amino)-propyl]...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101600([3-Carboxy-2-(undecylaminosulphonyl-amino)-propyl]...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101598([3-Carboxy-2-(dodecane-1-sulfonylamino)-propyl]-tr...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101604([3-Carboxy-2-(dodecane-1-sulfonylamino)-propyl]-tr...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50260115(CHEMBL4097976)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM61402(perhexiline maleate | (Z)-but-2-enedioic acid;2-(2...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50118093((4-Hydroxy-phenyl)-oxo-acetic acid | CHEMBL129918)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of CPT1B in heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50260105(CHEMBL1592481)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of Wistar rat heart mitochondrial CPT-1 assessed as reduction in conversion of palmitoyl CoA and L-carnitine into palmitoylcarnitine prein...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50403031(CHEMBL2216771)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of CPT1B (unknown origin) in KB cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50403045(CHEMBL2216773)
Affinity DataIC50: 1.68E+4nMAssay Description:Inhibition of CPT1B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50260109(CHEMBL4077250)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50403033(CHEMBL1231507)
Affinity DataIC50: 2.17E+4nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403034(CHEMBL2114397)
Affinity DataIC50: 2.73E+4nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50260108(CHEMBL4082420)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50122839([3-Carboxy-2-(3-tetradecyl-ureido)-propyl]-trimeth...)
Affinity DataIC50: 4.34E+4nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50260104(CHEMBL4081530)
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50122827([3-Carboxy-2-(3-nonyl-ureido)-propyl]-trimethyl-am...)
Affinity DataIC50: 4.62E+4nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50403030(CHEMBL2216768)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CPT1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50118093((4-Hydroxy-phenyl)-oxo-acetic acid | CHEMBL129918)
Affinity DataIC50: 6.03E+4nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50260105(CHEMBL1592481)
Affinity DataIC50: 7.70E+4nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50122833((3-Carboxy-2-octyloxycarbonylamino-propyl)-trimeth...)
Affinity DataIC50: 8.01E+4nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101590([3-Carboxy-2-(3-nonyl-ureido)-propyl]-trimethyl-am...)
Affinity DataIC50: 8.32E+4nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50403032(CHEMBL2216785)
Affinity DataIC50: 8.53E+4nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50260112(CHEMBL4068222)
Affinity DataIC50: 8.80E+4nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
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