Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with Target = 'Cell division related protein kinase 2'
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397589BDBM50397589(CHEMBL2171517)
Affinity DataIC50: 5nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397590BDBM50397590(CHEMBL2171516)
Affinity DataIC50: 20nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397588BDBM50397588(CHEMBL2171518)
Affinity DataIC50: 60nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397592BDBM50397592(CHEMBL2171514)
Affinity DataIC50: 240nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397593BDBM50397593(CHEMBL2171513)
Affinity DataIC50: 260nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397591BDBM50397591(CHEMBL2171515)
Affinity DataIC50: 510nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 47658BDBM47658(cid_1477566 | 1-(4-methylphenyl)-3-(2-pyridin-3-yl...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397595BDBM50397595(CHEMBL2171512)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 78336BDBM78336(CHEMBL1328065 | (6E)-6-[4-(3-pyridinylmethylamino)...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed