Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with Target = 'Cryptochrome-2'
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356658BDBM356658(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  79nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356696BDBM356696(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  79nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356935BDBM356935(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  128nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 50453623BDBM50453623(CHEMBL4211895)
Affinity DataEC50:  149nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356933BDBM356933(2-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  163nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356668BDBM356668(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  164nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 50453622BDBM50453622(CHEMBL4216091)
Affinity DataEC50:  167nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356645BDBM356645(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  171nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356636BDBM356636(US10214507, Compound 71 | US10759777, Compound 71)
Affinity DataEC50:  188nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356640BDBM356640(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  192nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356663BDBM356663(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  194nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356714BDBM356714(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  199nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356653BDBM356653(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  208nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356721BDBM356721(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  224nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 50453635BDBM50453635(CHEMBL4210175)
Affinity DataEC50:  246nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356687BDBM356687(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  261nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356951BDBM356951(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  330nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356694BDBM356694(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  332nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356639BDBM356639(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  363nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 50453619BDBM50453619(CHEMBL4217664)
Affinity DataEC50:  397nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 50453637BDBM50453637(CHEMBL4207485)
Affinity DataEC50:  406nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 50453627BDBM50453627(CHEMBL4208268)
Affinity DataEC50:  417nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356672BDBM356672(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  417nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356704BDBM356704(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  424nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356947BDBM356947(4-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  447nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356670BDBM356670(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  463nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356943BDBM356943(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  487nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356674BDBM356674(US10214507, Compound 86 | US10759777, Compound 86)
Affinity DataEC50:  497nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356684BDBM356684(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  528nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356725BDBM356725(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  541nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356679BDBM356679(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  547nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 50453632BDBM50453632(CHEMBL4207319)
Affinity DataEC50:  565nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356686BDBM356686(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  605nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356650BDBM356650(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  620nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356646BDBM356646(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  625nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356671BDBM356671(US10214507, Compound 85 | US10759777, Compound 85)
Affinity DataEC50:  667nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356956BDBM356956(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  716nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356644BDBM356644(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  719nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 50453633BDBM50453633(CHEMBL4214995)
Affinity DataEC50:  742nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 50453630BDBM50453630(CHEMBL4210300)
Affinity DataEC50:  833nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 50453634BDBM50453634(CHEMBL4218474)
Affinity DataEC50:  855nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 56256BDBM56256(N-(3-carbazol-9-yl-2-hydroxypropyl)-N-(furan-2-ylm...)
Affinity DataEC50:  870nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356923BDBM356923(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  1.03E+3nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356641BDBM356641(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  1.06E+3nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 50453615BDBM50453615(CHEMBL4211699)
Affinity DataEC50:  1.12E+3nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 50453618BDBM50453618(CHEMBL4218453)
Affinity DataEC50:  1.14E+3nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 356700BDBM356700(1-(3-(3,6-difluoro- 9H-carbazol-9-yl)-2- hydroxypr...)
Affinity DataEC50:  1.15E+3nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 50453644BDBM50453644(CHEMBL4215504)
Affinity DataEC50:  1.19E+3nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCryptochrome-2(Human)TBA
LigandChemical structure of BindingDB Monomer ID 50453624BDBM50453624(CHEMBL4214381)
Affinity DataEC50:  1.36E+3nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50453614BDBM50453614(CHEMBL4217929)
Affinity DataEC50:  1.49E+3nMAssay Description:Modulation activity at CRY2/PER2 in human U2OS cells harboring per2-dLuc assessed as activation of per2 activity measured every 100 mins for 5 days b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
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