Report error Found 311 Enz. Inhib. hit(s) with Target = 'Dynamin-1'
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 500nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
Affinity DataIC50: 720nMAssay Description:The GTPase activity of Drp1 was assayed using a colorimetric assay similar to as described previously by Leonard M. et al. Robust colorimetric assays...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 750nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 750nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 750nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 750nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 750nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 750nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 750nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 750nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 750nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 750nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 750nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
TargetDynamin-1-like protein [1-699] and Mitochondrial dynamics protein MID49 [126-454](Human)
Astellas Engineered Small Molecules US
US Patent
Astellas Engineered Small Molecules US
US Patent
Affinity DataIC50: 750nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
Affinity DataIC50: 910nMAssay Description:The GTPase activity of Drp1 was assayed using a colorimetric assay similar to as described previously by Leonard M. et al. Robust colorimetric assays...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of phosphotidylserine liposome-stimulated Dynamin 1 (unknown origin) GTPase activity by malachite green assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of phosphotidylserine liposome-stimulated Dynamin 1 (unknown origin) GTPase activity by malachite green assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.20E+3nMAssay Description:The GTPase activity of Drp1 was assayed using a colorimetric assay similar to as described previously by Leonard M. et al. Robust colorimetric assays...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:The GTPase activity of Drp1 was assayed using a colorimetric assay similar to as described previously by Leonard M. et al. Robust colorimetric assays...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:The GTPase activity of Drp1 was assayed using a colorimetric assay similar to as described previously by Leonard M. et al. Robust colorimetric assays...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:The GTPase activity of Drp1 was assayed using a colorimetric assay similar to as described previously by Leonard M. et al. Robust colorimetric assays...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of phosphotidylserine liposome-stimulated Dynamin 1 (unknown origin) GTPase activity by malachite green assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.60E+3nMAssay Description:The GTPase activity of Drp1 was assayed using a colorimetric assay similar to as described previously by Leonard M. et al. Robust colorimetric assays...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:The GTPase activity of Drp1 was assayed using a colorimetric assay similar to as described previously by Leonard M. et al. Robust colorimetric assays...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:The GTPase activity of Drp1 was assayed using a colorimetric assay similar to as described previously by Leonard M. et al. Robust colorimetric assays...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against dynamin1 GTPase expressed in sheep brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against dynamin1 GTPase expressed in sheep brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against dynamin1 GTPase expressed in sheep brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against dynamin1 GTPase expressed in sheep brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:The GTPase activity of Drp1 was assayed using a colorimetric assay similar to as described previously by Leonard M. et al. Robust colorimetric assays...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:The GTPase activity of Drp1 was assayed using a colorimetric assay similar to as described previously by Leonard M. et al. Robust colorimetric assays...More data for this Ligand-Target Pair
