Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with Target = 'Formyl peptide receptor-related sequence 1'
TargetFormyl peptide receptor-related sequence 1(Mouse)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50097567BDBM50097567(CHEMBL3588871)
Affinity DataEC50:  240nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetFormyl peptide receptor-related sequence 1(Mouse)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50050937BDBM50050937(N-formylmethionine-leucine-phenylalanine | (S)-2-[...)
Affinity DataKd: >300nMAssay Description:Binding affinity to mouse FPR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2016
Entry Details Article
PubMed
TargetFormyl peptide receptor-related sequence 1(Mouse)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186957BDBM50186957(1-(3-tert-butyl-2-methyl-5-oxo-1-phenyl-2,5-dihydr...)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at mouse FPR3 expressed in CHO-A12 cells assessed as cAMP level incubated for 1.5 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetFormyl peptide receptor-related sequence 1(Mouse)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50097570BDBM50097570(CHEMBL3590074)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetFormyl peptide receptor-related sequence 1(Mouse)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50097565BDBM50097565(CHEMBL3589947)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetFormyl peptide receptor-related sequence 1(Mouse)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50097560BDBM50097560(CHEMBL3590072)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetFormyl peptide receptor-related sequence 1(Mouse)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50097569BDBM50097569(CHEMBL3590075)
Affinity DataEC50:  2.30E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetFormyl peptide receptor-related sequence 1(Mouse)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50097564BDBM50097564(CHEMBL3589948)
Affinity DataEC50:  2.30E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetFormyl peptide receptor-related sequence 1(Mouse)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50097568BDBM50097568(CHEMBL3590076)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetFormyl peptide receptor-related sequence 1(Mouse)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50097563BDBM50097563(CHEMBL3590069)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetFormyl peptide receptor-related sequence 1(Mouse)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50097559BDBM50097559(CHEMBL3590073)
Affinity DataEC50:  2.80E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetFormyl peptide receptor-related sequence 1(Mouse)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50097562BDBM50097562(CHEMBL3590070)
Affinity DataEC50:  3.80E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetFormyl peptide receptor-related sequence 1(Mouse)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50097561BDBM50097561(CHEMBL3590071)
Affinity DataEC50:  3.90E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetFormyl peptide receptor-related sequence 1(Mouse)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50097566BDBM50097566(CHEMBL3589946)
Affinity DataEC50:  4.90E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetFormyl peptide receptor-related sequence 1(Mouse)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50071956BDBM50071956(CHEMBL3407845)
Affinity DataEC50:  9.00E+3nMAssay Description:Induction of calcium release in mouse FPR2 receptor-expressed HEK cell by cytosolic-free calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2016
Entry Details Article
PubMed