Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with Target = 'H2-K region expressed gene 2, rat orthologue'
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079824BDBM50079824(((S)-1-{(S)-1-[(S)-(S)-1-(1-Carbamoyl-3-methyl-but...)
Affinity DataIC50: 1nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079829BDBM50079829(((S)-1-{(S)-1-[(S)-1-((S)-1-Carbamoyl-3-methyl-but...)
Affinity DataIC50: 1nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079854BDBM50079854((S)-2-(3-Cyclohexyl-propylamino)-pentanoic acid [(...)
Affinity DataIC50: 25nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079848BDBM50079848((S)-2-(3-Cyclohexyl-propylamino)-2-methyl-pentanoi...)
Affinity DataIC50: 100nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079845BDBM50079845((S)-2-[(R)-3-(3-Cyclohexyl-propylamino)-2-oxo-3-pr...)
Affinity DataIC50: 150nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079846BDBM50079846(N-Butyl-N'-{(S)-2-[(R)-3-(3-cyclohexyl-propylamino...)
Affinity DataIC50: 160nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079850BDBM50079850(N-Butyl-N'-{(S)-2-[(R)-3-(3-cyclohexyl-propylamino...)
Affinity DataIC50: 210nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079844BDBM50079844(N-Butyl-N'-{(S)-2-[(R)-3-(3-cyclohexyl-propylamino...)
Affinity DataIC50: 240nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079826BDBM50079826((S)-2-{(S)-2-[2-(3-Cyclohexyl-propylamino)-2-methy...)
Affinity DataIC50: 260nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079823BDBM50079823(((S)-1-{(S)-1-[(S)-1-((S)-1-Carbamoyl-3-methyl-but...)
Affinity DataIC50: 270nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079827BDBM50079827([(S)-1-((S)-1-{[(S)-1-((S)-1-Carbamoyl-3-methyl-bu...)
Affinity DataIC50: 320nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079837BDBM50079837((S)-2-[(R)-3-((E)-3-Cycloheptyl-allylamino)-2-oxo-...)
Affinity DataIC50: 340nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079833BDBM50079833((S)-2-[(R)-3-(3-Cyclohexyl-propylamino)-2-oxo-pyrr...)
Affinity DataIC50: 760nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079833BDBM50079833((S)-2-[(R)-3-(3-Cyclohexyl-propylamino)-2-oxo-pyrr...)
Affinity DataIC50: 760nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079842BDBM50079842(N-Butyl-N'-{(S)-2-[(R)-3-(3-cyclohexyl-propylamino...)
Affinity DataIC50: 780nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079828BDBM50079828([(S)-1-(1-{(S)-1-[((S)-(S)-1-Carbamoyl-3-methyl-bu...)
Affinity DataIC50: 1.20E+3nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079847BDBM50079847(1-(3-Cyclohexyl-propylamino)-cyclopentanecarboxyli...)
Affinity DataIC50: 1.26E+3nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079852BDBM50079852((S)-2-[(S)-3-(3-Cyclohexyl-propylamino)-2-oxo-3-pr...)
Affinity DataIC50: 1.80E+3nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079840BDBM50079840(((S)-1-{(S)-1-[(S)-1-((S)-1-Carbamoyl-3-methyl-but...)
Affinity DataIC50: 1.90E+3nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079821BDBM50079821((1-(S)-1-Benzyl-2-{1-[(S)-1-((S)-1-carbamoyl-3-met...)
Affinity DataIC50: 3.00E+3nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079836BDBM50079836((S)-2-Benzyl-N-{(S)-1-[(S)-1-((S)-1-carbamoyl-3-me...)
Affinity DataIC50: 3.10E+3nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079843BDBM50079843(N'-{(S)-2-[(R)-3-(3-Cyclohexyl-propylamino)-2-oxo-...)
Affinity DataIC50: 4.70E+3nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079839BDBM50079839([(S)-1-({(S)-1-[(S)-1-((S)-1-Carbamoyl-3-methyl-bu...)
Affinity DataIC50: 1.20E+4nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079834BDBM50079834((S)-2-[(S)-3-(3-Cyclohexyl-propylamino)-2-oxo-pyrr...)
Affinity DataIC50: 1.40E+4nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079834BDBM50079834((S)-2-[(S)-3-(3-Cyclohexyl-propylamino)-2-oxo-pyrr...)
Affinity DataIC50: 1.40E+4nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079838BDBM50079838((S)-2-Benzyl-N-{(R)-1-[(S)-1-((S)-1-carbamoyl-3-me...)
Affinity DataIC50: 2.40E+4nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079830BDBM50079830([(S)-1-((S)-1-{[(S)-1-((S)-1-Carbamoyl-3-methyl-bu...)
Affinity DataIC50: 4.50E+4nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079841BDBM50079841((R)-2-[(S)-3-(3-Cyclohexyl-propylamino)-2-oxo-3-pr...)
Affinity DataIC50: 5.00E+4nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079825BDBM50079825((S)-N-{(S)-1-[(S)-1-((S)-1-Carbamoyl-3-methyl-buty...)
Affinity DataIC50: 5.00E+4nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079851BDBM50079851(N'-{(S)-2-[(R)-3-(3-Cyclohexyl-propylamino)-2-oxo-...)
Affinity DataIC50: 5.00E+4nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079835BDBM50079835(((S)-2-{(R)-1-[(S)-1-((S)-1-Carbamoyl-3-methyl-but...)
Affinity DataIC50: 5.00E+4nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079853BDBM50079853((S)-2-[(R)-3-(3-Cyclohexyl-propylamino)-2-oxo-pyrr...)
Affinity DataIC50: 5.00E+4nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079849BDBM50079849((R)-2-[(R)-3-(3-Cyclohexyl-propylamino)-2-oxo-3-pr...)
Affinity DataIC50: 5.00E+4nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079831BDBM50079831((S)-2-{(S)-2-[(R)-2-(3-Cyclohexyl-propylamino)-but...)
Affinity DataIC50: 5.00E+4nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079832BDBM50079832((S)-N-{(R)-1-[(S)-1-((S)-1-Carbamoyl-3-methyl-buty...)
Affinity DataIC50: 5.00E+4nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetH2-K region expressed gene 2, rat orthologue(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079822BDBM50079822([(S)-1-((S)-1-{(S)-1-[((S)-1-Carbamoyl-3-methyl-bu...)
Affinity DataIC50: 8.80E+4nMAssay Description:Ability to inhibit binding of biotinylated rat myelin basic protein 13-mer peptide (RMBP 90-102, Major histocompatibility complex class II to purifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed