Compile Data Set for Download or QSAR
Report error Found 4373 Enz. Inhib. hit(s) with Target = 'Macrophage colony-stimulating factor 1'
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644089BDBM50644089(CHEMBL5574726)
Affinity DataKd:  0.00200nMAssay Description:Binding affinity to recombinant human CSF-1R assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775143BDBM775143(US12435062, Compound 55)
Affinity DataIC50: 0.00300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775185BDBM775185(US12435062, Compound 69)
Affinity DataIC50: 0.00300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775146BDBM775146(US12435062, Compound 56)
Affinity DataIC50: 0.00400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775128BDBM775128(US12435062, Compound 48)
Affinity DataIC50: 0.00500nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775125BDBM775125(US12435062, Compound 47)
Affinity DataIC50: 0.00500nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775173BDBM775173(US12435062, Compound 65)
Affinity DataIC50: 0.00500nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775110BDBM775110(US12435062, Compound 42)
Affinity DataIC50: 0.00500nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775206BDBM775206(US12435062, Compound 76)
Affinity DataIC50: 0.00500nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775113BDBM775113(US12435062, Compound 43)
Affinity DataIC50: 0.00600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775116BDBM775116(US12435062, Compound 44)
Affinity DataIC50: 0.00700nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775182BDBM775182(US12435062, Compound 68)
Affinity DataIC50: 0.00700nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775203BDBM775203(US12435062, Compound 75)
Affinity DataIC50: 0.00800nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775158BDBM775158(US12435062, Compound 60)
Affinity DataIC50: 0.00800nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775119BDBM775119(US12435062, Compound 45)
Affinity DataIC50: 0.00900nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775167BDBM775167(US12435062, Compound 63)
Affinity DataIC50: 0.00900nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775200BDBM775200(US12435062, Compound 74)
Affinity DataIC50: 0.00900nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775191BDBM775191(US12435062, Compound 71)
Affinity DataIC50: 0.0100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775197BDBM775197(US12435062, Compound 73)
Affinity DataIC50: 0.0110nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775055BDBM775055(US12435062, Compound 38)
Affinity DataIC50: 0.0120nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775122BDBM775122(US12435062, Compound 46)
Affinity DataIC50: 0.0120nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775194BDBM775194(US12435062, Compound 72)
Affinity DataIC50: 0.0140nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775104BDBM775104(US12435062, Compound 40)
Affinity DataIC50: 0.0160nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775170BDBM775170(US12435062, Compound 64)
Affinity DataIC50: 0.0160nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775221BDBM775221(1,2-dimethyl-N-(5-((2-(1-methyl-1H-pyrazol-4-yl)py...)
Affinity DataIC50: 0.0190nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775164BDBM775164(US12435062, Compound 62)
Affinity DataIC50: 0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775224BDBM775224(N-(5-((2-(1H-pyrazol-4-yl)pyridin-4-yl)oxy)pyridin...)
Affinity DataIC50: 0.0210nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775131BDBM775131(US12435062, Compound 49)
Affinity DataIC50: 0.0230nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775149BDBM775149(US12435062, Compound 57)
Affinity DataIC50: 0.0240nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775107BDBM775107(US12435062, Compound 41)
Affinity DataIC50: 0.0270nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775188BDBM775188(US12435062, Compound 70)
Affinity DataIC50: 0.0320nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775179BDBM775179(US12435062, Compound 67)
Affinity DataIC50: 0.0330nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775101BDBM775101(US12435062, Compound 39)
Affinity DataIC50: 0.0330nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775161BDBM775161(US12435062, Compound 61)
Affinity DataIC50: 0.0450nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775212BDBM775212(US12435062, Compound 120)
Affinity DataIC50: 0.0520nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775176BDBM775176(US12435062, Compound 66)
Affinity DataIC50: 0.0540nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775218BDBM775218(US12435062, Compound 122)
Affinity DataIC50: 0.0550nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775137BDBM775137(US12435062, Compound 51)
Affinity DataIC50: 0.0560nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775152BDBM775152(US12435062, Compound 58)
Affinity DataIC50: 0.0690nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775134BDBM775134(US12435062, Compound 50)
Affinity DataIC50: 0.0780nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775155BDBM775155(US12435062, Compound 59)
Affinity DataIC50: 0.121nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 775140BDBM775140(US12435062, Compound 53)
Affinity DataIC50: 0.135nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 789791BDBM789791(3-(4-(4-(Benzyl(methyl)amino)-7H-pyrrolo[2,3-d]pyr...)
Affinity DataIC50: 0.200nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
3/11/2026
Entry Details US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50640578BDBM50640578(CHEMBL5563269 | US20250353857, Compound SH-01-59)
Affinity DataIC50: 0.200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/11/2026
Entry Details US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617728BDBM50617728(CHEMBL5415149 | US20250353857, Compound TIA05-014)
Affinity DataIC50: 0.200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2026
Entry Details US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 789810BDBM789810(Dimethyl(4-(4-(methyl(3-methylbenzyl)amino)-7H-pyr...)
Affinity DataIC50: 0.200nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
3/11/2026
Entry Details US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617728BDBM50617728(CHEMBL5415149 | US20250353857, Compound TIA05-014)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of CSF1R (unknown origin) using FRET-peptide as substrate incubated in presence of ATP by FRET based Z-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50640596BDBM50640596(CHEMBL5573671 | US20250353857, Compound HHMT1-170)
Affinity DataIC50: 0.200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/11/2026
Entry Details US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622233BDBM50622233(CHEMBL5415647 | US20250353857, Compound FAB01-23)
Affinity DataIC50: 0.200nMMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
3/11/2026
Entry Details US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50640575BDBM50640575(CHEMBL5556952 | US20250353857, Compound TIA05-032)
Affinity DataIC50: 0.200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/11/2026
Entry Details US Patent

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