Compile Data Set for Download or QSAR
Report error Found 184 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase 1 [8-360]'
TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 193676BDBM193676(US9670208, Example 295 4-(3-(cyclopropylmethyl)-[1...)
Affinity DataIC50: 0.400nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 193385BDBM193385(US9670208, Example 57)
Affinity DataIC50: 0.5nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192361BDBM192361(US9187462, I-41)
Affinity DataIC50: 0.550nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192386BDBM192386(US9187462, I-66)
Affinity DataIC50: 0.600nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 193675BDBM193675(US9670208, Example 279 N-(1-methyl-1H-pyrazol-5-yl...)
Affinity DataIC50: 0.600nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192385BDBM192385(US9187462, I-65)
Affinity DataIC50: 0.600nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 193773BDBM193773(US9670208, Example 402 4-(3-(4-fluorobenzyl)-[1,2,...)
Affinity DataIC50: 0.600nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 236879BDBM236879(US9388171, I-8)
Affinity DataIC50: 0.748nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 191370BDBM191370(US9670208, Example 35)
Affinity DataIC50: 0.800nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 193672BDBM193672(US9670208, Example 278 4-(3-(pyridin-2-ylmethyl)-[...)
Affinity DataIC50: 0.800nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 193781BDBM193781(US9670208, Example 493 4-(3-((6-ethoxypyridin-3-yl...)
Affinity DataIC50: 0.800nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192322BDBM192322(US9187462, I-2)
Affinity DataIC50: 0.800nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 193381BDBM193381(US9670208, Example 49)
Affinity DataIC50: 0.800nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 193396BDBM193396(US9670208, Example 121)
Affinity DataIC50: 0.900nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 193412BDBM193412(US9670208, Example 276 N-(1-methyl-1H-pyrazol-5-yl...)
Affinity DataIC50: 0.900nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 193410BDBM193410(US9670208, Example 272 4-(3-((6-methoxypyridin-3-y...)
Affinity DataIC50: 0.900nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 193776BDBM193776(US9670208, Example 403 4-(3-(3-fluoro-4-methoxyben...)
Affinity DataIC50: 0.900nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 193756BDBM193756(US9670208, Example 317 4-(3-((4,4-difluorocyclohex...)
Affinity DataIC50: 0.900nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192364BDBM192364(US9187462, I-44)
Affinity DataIC50: 1nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192436BDBM192436(US9187462, II-46)
Affinity DataIC50: 1.10nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192352BDBM192352(US9187462, I-32)
Affinity DataIC50: 1.10nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192368BDBM192368(US9187462, I-48)
Affinity DataIC50: 1.10nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 236882BDBM236882(US9388171, I-24)
Affinity DataIC50: 1.15nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192403BDBM192403(US9187462, II-13)
Affinity DataIC50: 1.20nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192388BDBM192388(US9187462, I-68 | BDBM192402)
Affinity DataIC50: 1.20nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192389BDBM192389(US9187462, I-69)
Affinity DataIC50: 1.20nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192335BDBM192335(US9187462, I-15)
Affinity DataIC50: 1.20nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192359BDBM192359(US9187462, I-39)
Affinity DataIC50: 1.20nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192437BDBM192437(US9187462, II-47)
Affinity DataIC50: 1.30nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192388BDBM192388(US9187462, I-68 | BDBM192402)
Affinity DataIC50: 1.30nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192367BDBM192367(US9187462, I-47)
Affinity DataIC50: 1.40nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192332BDBM192332(US9187462, I-12)
Affinity DataIC50: 1.40nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192342BDBM192342(US9187462, I-22)
Affinity DataIC50: 1.40nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192438BDBM192438(US9187462, II-48)
Affinity DataIC50: 1.40nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192353BDBM192353(US9187462, I-33)
Affinity DataIC50: 1.5nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 193411BDBM193411(US9670208, Example 275 N-(1-methyl-1H-pyrazol-5-yl...)
Affinity DataIC50: 1.5nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192443BDBM192443(US9187462, II-53)
Affinity DataIC50: 1.5nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192356BDBM192356(US9187462, I-36)
Affinity DataIC50: 1.60nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192351BDBM192351(US9187462, I-31)
Affinity DataIC50: 1.70nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 193754BDBM193754(US9670208, Example 306 N-(1-methyl-1H-pyrazol-5-yl...)
Affinity DataIC50: 1.80nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 193780BDBM193780(US9670208, Example 467 N-(1-(3-chloro-4-fluorophen...)
Affinity DataIC50: 1.80nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192327BDBM192327(US9187462, I-7)
Affinity DataIC50: 1.80nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 236881BDBM236881(US9388171, I-21)
Affinity DataIC50: 1.86nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192442BDBM192442(US9187462, II-52)
Affinity DataIC50: 1.90nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192340BDBM192340(US9187462, I-20)
Affinity DataIC50: 2nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192355BDBM192355(US9187462, I-35)
Affinity DataIC50: 2nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192346BDBM192346(US9187462, I-26)
Affinity DataIC50: 2nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192381BDBM192381(US9187462, I-61)
Affinity DataIC50: 2nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192323BDBM192323(US9187462, I-3)
Affinity DataIC50: 2.10nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [8-360](Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 192350BDBM192350(US9187462, I-30)
Affinity DataIC50: 2.10nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an N-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
US Patent

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