Compile Data Set for Download or QSAR
Report error Found 252 Enz. Inhib. hit(s) with Target = 'Non-receptor tyrosine-protein kinase TNK1'
TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 0.584nMAssay Description:Inhibition of human TNK1 using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 130909BDBM130909(US8822500, Stauro- sporine | US9920060, Staurospor...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human TNK1 using poly[Glu:Tyr] (4:1) as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition and measured after 120 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419721BDBM419721(US10464919, Example 59)
Affinity DataIC50: 1.37nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human TNK1 using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 482158BDBM482158(TAE684 | BDBM50242742)
Affinity DataKd:  1.80nMAssay Description:Binding constant for TNK1 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31096BDBM31096(CHEMBL290084 | Staurosporine | cid_451705 | US2024...)
Affinity DataKd:  2.5nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2011
Entry Details
PCBioAssay
TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataKd:  2.5nMAssay Description:Binding constant for full-length TNK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2012
Entry Details Article
PubMed
TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataKd:  2.5nMAssay Description:Binding constant for TNK1 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419794BDBM419794(US10464919, Example 132)
Affinity DataIC50: 2.77nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419844BDBM419844(US10464919, Example 182)
Affinity DataIC50: 3.33nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419799BDBM419799(US10464919, Example 137)
Affinity DataIC50: 3.36nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419755BDBM419755(US10464919, Example 93)
Affinity DataIC50: 3.59nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419785BDBM419785(US10464919, Example 123)
Affinity DataIC50: 3.92nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50505541BDBM50505541(CHEMBL4465866)
Affinity DataKd:  4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged TNK1 (106 to 390 residues) expressed in baculovirus expression system using CSKtide as su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419797BDBM419797(US10464919, Example 135)
Affinity DataIC50: 4.04nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419796BDBM419796(US10464919, Example 134)
Affinity DataIC50: 4.15nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419804BDBM419804(US10464919, Example 142)
Affinity DataIC50: 4.42nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419718BDBM419718(US10464919, Example 56)
Affinity DataIC50: 4.96nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419781BDBM419781(US10464919, Example 119)
Affinity DataIC50: 5nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419751BDBM419751(US10464919, Example 89)
Affinity DataIC50: 5.07nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419791BDBM419791(US10464919, Example 129)
Affinity DataIC50: 5.56nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419761BDBM419761(US10464919, Example 99)
Affinity DataIC50: 5.59nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419731BDBM419731(US10464919, Example 69)
Affinity DataIC50: 5.77nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419803BDBM419803(US10464919, Example 141)
Affinity DataIC50: 5.82nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419807BDBM419807(US10464919, Example 145)
Affinity DataIC50: 6.29nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419758BDBM419758(US10464919, Example 96)
Affinity DataIC50: 6.77nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419784BDBM419784(US10464919, Example 122)
Affinity DataIC50: 7.28nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419842BDBM419842(US10464919, Example 180)
Affinity DataIC50: 8.05nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419746BDBM419746(US10464919, Example 84)
Affinity DataIC50: 8.46nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419759BDBM419759(US10464919, Example 97)
Affinity DataIC50: 8.81nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50308060BDBM50308060(CEP-701 | 16-hydroxy-16-(hydroxymethyl)-15-methyl-...)
Affinity DataKd:  9.30nMAssay Description:Binding affinity to TNK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50308060BDBM50308060(CEP-701 | 16-hydroxy-16-(hydroxymethyl)-15-methyl-...)
Affinity DataKd:  9.30nMAssay Description:Binding constant for TNK1 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419832BDBM419832(US10464919, Example 170)
Affinity DataIC50: 9.65nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419793BDBM419793(US10464919, Example 131)
Affinity DataIC50: 9.89nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419782BDBM419782(US10464919, Example 120)
Affinity DataIC50: 10.2nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419786BDBM419786(US10464919, Example 124)
Affinity DataIC50: 10.4nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419787BDBM419787(US10464919, Example 125)
Affinity DataIC50: 10.4nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419801BDBM419801(US10464919, Example 139)
Affinity DataIC50: 10.6nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419775BDBM419775(US10464919, Example 113)
Affinity DataIC50: 10.7nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419822BDBM419822(US10464919, Example 160)
Affinity DataIC50: 10.7nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419740BDBM419740(US10464919, Example 78)
Affinity DataIC50: 11nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419738BDBM419738(US10464919, Example 76)
Affinity DataIC50: 11.3nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419757BDBM419757(US10464919, Example 95)
Affinity DataIC50: 11.4nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419737BDBM419737(US10464919, Example 75)
Affinity DataIC50: 11.4nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419769BDBM419769(US10464919, Example 107)
Affinity DataIC50: 11.4nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419843BDBM419843(US10464919, Example 181)
Affinity DataIC50: 11.6nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419747BDBM419747(US10464919, Example 85)
Affinity DataIC50: 11.8nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419722BDBM419722(US10464919, Example 60)
Affinity DataIC50: 12.1nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419732BDBM419732(US10464919, Example 70)
Affinity DataIC50: 12.4nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TNK1(Human)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 419765BDBM419765(US10464919, Example 103)
Affinity DataIC50: 12.5nMAssay Description:The tankyrase-1 or tankyrase-2 enzyme inhibitory activities of the compounds of the present invention were assayed in the following manner by use of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2020
Entry Details
US Patent

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