Report error Found 346 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 4 group A member 1'
Affinity DataEC50: 0.115nMAssay Description:Agonist activity at nuclear orphan receptor Nur77 expressed in human BGC823 cells co-transfected with fused GAL4-LBD assessed as transactivation afte...More data for this Ligand-Target Pair
Affinity DataEC50: 0.115nMAssay Description:Inhibition of Gal4-fused Nur77-LBD in human BGC-823 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.278nMAssay Description:Agonist activity at nuclear orphan receptor Nur77 expressed in human BGC823 cells co-transfected with fused GAL4-Nur77 assessed as transactivation af...More data for this Ligand-Target Pair
Affinity DataEC50: 0.278nMAssay Description:Inhibition of Gal4-fused full length Nur77 in human BGC-823 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 33nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77-LBD (367 to 598 residues) expressed in Escherichia coli BL21 DE3 by surface plasmon...More data for this Ligand-Target Pair
Affinity DataKd: 36nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77-LBD (367 to 598 residues) expressed in Escherichia coli BL21 DE3 by surface plasmon...More data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Agonist activity at human Nur77 LBD transiently transfected in HEK293T cells incubated for 16 hrs by Gal4-hybrid reporter gene based Dual-glo lucifer...More data for this Ligand-Target Pair
Affinity DataKd: 66nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77-LBD (367 to 598 residues) expressed in Escherichia coli BL21 DE3 by flourescence qu...More data for this Ligand-Target Pair
Affinity DataKd: 66nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77-LBD (367 to 598 residues) expressed in Escherichia coli BL21 DE3 by flourescence qu...More data for this Ligand-Target Pair
Affinity DataKd: 91nMAssay Description:Binding affinity to His-tagged Nur77 ligand binding domain (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKd: 110nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77-LBD (367 to 598 residues) expressed in Escherichia coli BL21 DE3 by surface plasmon...More data for this Ligand-Target Pair
Affinity DataKd: 121nMAssay Description:Binding affinity to Nur77 ligand binding domain (unknown origin) by fluorescence quenching assayMore data for this Ligand-Target Pair
Affinity DataEC50: 140nMAssay Description:Agonist activity at human Nur77 LBD transiently transfected in HEK293T cells incubated for 16 hrs by Gal4-hybrid reporter gene based Dual-glo lucifer...More data for this Ligand-Target Pair
Affinity DataKd: 154nMAssay Description:Binding affinity to wild type Nur77 ligand binding domain (unknown origin) assessed as decrease in fluorescence intensity incubated for 30 secs by fl...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 195nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (San Diego, CA) NIH Molecular Libraries Screening Cen...More data for this Ligand-Target Pair
Affinity DataKd: 217nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77-LBD (367 to 598 residues) expressed in Escherichia coli BL21 DE3 by flourescence qu...More data for this Ligand-Target Pair
Affinity DataKd: 220nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Affinity DataKd: 270nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Affinity DataKd: 290nMAssay Description:Binding affinity to Nur77 LBD (unknown origin) expressed in Escherichia coli incubated for 3 hrs by circular dichroism analysisMore data for this Ligand-Target Pair
Affinity DataKd: 290nMAssay Description:Binding affinity to Nur77 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 290nMAssay Description:Binding affinity to purified Nur77 LBD (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 320nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Affinity DataKd: 354nMAssay Description:Binding affinity to Nur77 ligand binding domain (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Affinity DataKd: 354nMAssay Description:Binding affinity to His-tagged Nur77 ligand binding domain (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataEC50: 480nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
Affinity DataIC50: 493nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (San Diego, CA) NIH Molecular Libraries Screening Cen...More data for this Ligand-Target Pair
Affinity DataKd: 520nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Affinity DataEC50: 540nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
Affinity DataIC50: 558nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (San Diego, CA) NIH Molecular Libraries Screening Cen...More data for this Ligand-Target Pair
Affinity DataEC50: 620nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
Affinity DataEC50: 670nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
Affinity DataKd: 720nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Affinity DataIC50: 725nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (San Diego, CA) NIH Molecular Libraries Screening Cen...More data for this Ligand-Target Pair
Affinity DataKd: 740nMAssay Description:Binding affinity to Nur77 receptor expressed in human BGC823 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 783nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (San Diego, CA) NIH Molecular Libraries Screening Cen...More data for this Ligand-Target Pair
Affinity DataKd: 800nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Affinity DataKd: 830nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Affinity DataKd: 870nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Affinity DataEC50: 940nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
Affinity DataKd: 960nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Affinity DataIC50: 963nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (San Diego, CA) NIH Molecular Libraries Screening Cen...More data for this Ligand-Target Pair
Affinity DataEC50: 1.03E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
Affinity DataEC50: 1.05E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
Affinity DataIC50: 1.07E+3nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (San Diego, CA) NIH Molecular Libraries Screening Cen...More data for this Ligand-Target Pair
Affinity DataIC50: 1.08E+3nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (San Diego, CA) NIH Molecular Libraries Screening Cen...More data for this Ligand-Target Pair
Affinity DataIC50: 1.13E+3nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (San Diego, CA) NIH Molecular Libraries Screening Cen...More data for this Ligand-Target Pair
Affinity DataKd: 1.17E+3nMAssay Description:Binding affinity to Nur77 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 1.17E+3nMAssay Description:Binding affinity to His-tagged Nur77 ligand binding domain (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataEC50: 1.20E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
Affinity DataKd: 1.34E+3nMAssay Description:Binding affinity to His-tagged Nur77 ligand binding domain (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair

3D Structure (crystal)



































