Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily E member 1'
LigandChemical structure of BindingDB Monomer ID 50392995BDBM50392995(CHEMBL2152523)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of IKs (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50343721BDBM50343721(3-(4-(4-(2-fluoro-4-methylphenyl)-5-(4-methoxyphen...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of IKrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50343722BDBM50343722(3-(4-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-4-(2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of IKrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50355405BDBM50355405(CHEMBL1835153)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Iks channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50045833BDBM50045833(CHEMBL3314349)
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of human cardiac slowly activating delayed rectifier K+ channel expressed in CHO cells by electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50468128BDBM50468128(CHEMBL4282052)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of IKs (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50523763BDBM50523763(CHEMBL4438854)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of IKs (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50385309BDBM50385309(CHEMBL2035983)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Iks ion channel by voltage clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103543BDBM50103543(CHEMBL3358006)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of IKs channel (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50246769BDBM50246769(CHEMBL4064608)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of IKs (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50524101BDBM50524101(CHEMBL4474619)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human KCNE1 by Ion-work electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50524102BDBM50524102(CHEMBL4542281)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human KCNE1 by Ion-work electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50523766BDBM50523766(CHEMBL4476275)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of IKs (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50045831BDBM50045831(CHEMBL3314352)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human cardiac slowly activating delayed rectifier K+ channel expressed in CHO cells by electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50045830BDBM50045830(CHEMBL3314362)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human cardiac slowly activating delayed rectifier K+ channel expressed in CHO cells by electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50523773BDBM50523773(CHEMBL4475999)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of IKs (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50524103BDBM50524103(CHEMBL4563459)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human KCNE1 by Ion-work electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E member 1(Rabbit)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403104BDBM50403104(CHEMBL2216904)
Affinity DataIC50: 5.25E+4nMAssay Description:Inhibition of Iks tail current in rabbit ventricular myocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50523765BDBM50523765(CHEMBL4437013)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of IKs (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed