Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with Target = 'Proprotein convertase subtilisin/kexin type 4'
TargetProprotein convertase subtilisin/kexin type 4(Human)
Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270054BDBM50270054(TPRARRRKKRT | CHEMBL502642)
Affinity DataKi:  441nMAssay Description:Inhibition of human recombinant PC4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 4(Human)
Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270060BDBM50270060(TPQRARRRKKRT | CHEMBL455792)
Affinity DataKi:  515nMAssay Description:Inhibition of human recombinant PC4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 4(Human)
Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269901BDBM50269901(TPRARRRKKRI | CHEMBL525748)
Affinity DataKi:  562nMAssay Description:Inhibition of human recombinant PC4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 4(Human)
Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270069BDBM50270069(TPQRARRRKKRY | CHEMBL499438)
Affinity DataKi:  624nMAssay Description:Inhibition of human recombinant PC4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 4(Human)
Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270068BDBM50270068(TPQRARRRKKRF | CHEMBL500184)
Affinity DataKi:  772nMAssay Description:Inhibition of human recombinant PC4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 4(Human)
Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270067BDBM50270067(TPQRARRRKKRW | CHEMBL503520)
Affinity DataKi:  952nMAssay Description:Inhibition of human recombinant PC4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed