Compile Data Set for Download or QSAR
Report error Found 165 Enz. Inhib. hit(s) with Target = 'Proprotein convertase subtilisin/kexin type 6'
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50264960BDBM50264960(CHEMBL4089819)
Affinity DataKi:  0.200nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50264892BDBM50264892(CHEMBL4065072)
Affinity DataKi:  0.300nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399749BDBM50399749(CHEMBL2179430)
Affinity DataKi:  0.340nMpH: 6.5Assay Description:Competitive inhibition of human recombinant PACE4 expressed in Drosophila S2 cells using pyroGlu-Arg-Val-Lys-Arg-methyl-coumaryl-7-amide as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50264931BDBM50264931(CHEMBL4084457)
Affinity DataKi:  0.400nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399753BDBM50399753(CHEMBL2179835)
Affinity DataKi:  0.400nMpH: 6.5Assay Description:Competitive inhibition of human recombinant PACE4 expressed in Drosophila S2 cells using pyroGlu-Arg-Val-Lys-Arg-methyl-coumaryl-7-amide as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265119BDBM50265119(CHEMBL4091099)
Affinity DataKi:  0.400nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265083BDBM50265083(CHEMBL4100996)
Affinity DataKi:  0.5nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303774BDBM50303774(phenylacetyl-Arg-Val-Arg-4-amidinobenzylamide | CH...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of human PACE4 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265384BDBM50265384(CHEMBL4104777)
Affinity DataKi:  0.600nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265344BDBM50265344(CHEMBL4070237)
Affinity DataKi:  0.900nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265130BDBM50265130(CHEMBL4064275)
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265091BDBM50265091(CHEMBL4083310)
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399754BDBM50399754(CHEMBL2179836)
Affinity DataKi:  1.10nMpH: 6.5Assay Description:Competitive inhibition of human recombinant PACE4 expressed in Drosophila S2 cells using pyroGlu-Arg-Val-Lys-Arg-methyl-coumaryl-7-amide as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399752BDBM50399752(CHEMBL2179429)
Affinity DataKi:  1.30nMpH: 6.5Assay Description:Competitive inhibition of human recombinant PACE4 expressed in Drosophila S2 cells using pyroGlu-Arg-Val-Lys-Arg-methyl-coumaryl-7-amide as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265145BDBM50265145(CHEMBL4073661)
Affinity DataKi:  1.30nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265141BDBM50265141(CHEMBL4094478)
Affinity DataKi:  1.5nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50264955BDBM50264955(CHEMBL4099961)
Affinity DataKi:  1.70nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265045BDBM50265045(CHEMBL4097940)
Affinity DataKi:  1.80nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50264969BDBM50264969(CHEMBL4096348)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265129BDBM50265129(CHEMBL4085824)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265131BDBM50265131(CHEMBL4093570)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265000BDBM50265000(CHEMBL4101342)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50264941BDBM50264941(CHEMBL4063327)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399751BDBM50399751(CHEMBL2179431)
Affinity DataKi:  2nMpH: 6.5Assay Description:Competitive inhibition of human recombinant PACE4 expressed in Drosophila S2 cells using pyroGlu-Arg-Val-Lys-Arg-methyl-coumaryl-7-amide as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265328BDBM50265328(CHEMBL4087970)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265331BDBM50265331(CHEMBL4103443)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265170BDBM50265170(CHEMBL4075692)
Affinity DataKi:  2.10nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265047BDBM50265047(CHEMBL4072949)
Affinity DataKi:  2.20nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303775BDBM50303775((S)-2-acetamido-N-((S)-1-((S)-1-(4-carbamimidoylbe...)
Affinity DataKi:  2.40nMAssay Description:Inhibition of human PACE4 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265048BDBM50265048(CHEMBL4065627)
Affinity DataKi:  2.5nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50466079BDBM50466079(CHEMBL4286124)
Affinity DataKi:  2.60nMAssay Description:Inhibition of recombinant human PACE4 using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50264970BDBM50264970(CHEMBL4059801)
Affinity DataKi:  2.80nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50264999BDBM50264999(CHEMBL4084913)
Affinity DataKi:  2.80nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50264971BDBM50264971(CHEMBL4089913)
Affinity DataKi:  3nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50264972BDBM50264972(CHEMBL4080551)
Affinity DataKi:  3nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265144BDBM50265144(CHEMBL4067772)
Affinity DataKi:  3nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265332BDBM50265332(CHEMBL4093266)
Affinity DataKi:  3nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303776BDBM50303776(N-((6S,9S,12S)-1,17-diamino-6-(4-carbamimidoylbenz...)
Affinity DataKi:  3nMAssay Description:Inhibition of human PACE4 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265092BDBM50265092(CHEMBL4063219)
Affinity DataKi:  3nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50446944BDBM50446944(CHEMBL3115771)
Affinity DataKi:  3.10nMAssay Description:Inhibition of human recombinant PACE4 expressed in drosophila schneider 2 cells using pyroGlu-Arg-Thr-Lys-Arg-AMC as substrate after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50533413BDBM50533413(CHEMBL3126388)
Affinity DataKi:  3.60nMAssay Description:Inhibition of recombinant C-terminal truncated human SPC4 expressed in drosophila Schneider 2 cells after 1 hr by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265162BDBM50265162(CHEMBL4076965)
Affinity DataKi:  3.70nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50264994BDBM50264994(CHEMBL4097058)
Affinity DataKi:  4nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50264930BDBM50264930(CHEMBL4077533)
Affinity DataKi:  4nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265140BDBM50265140(CHEMBL4066994)
Affinity DataKi:  4nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265185BDBM50265185(CHEMBL4092088)
Affinity DataKi:  4nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50264894BDBM50264894(CHEMBL4063459)
Affinity DataKi:  4nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265090BDBM50265090(CHEMBL4101304)
Affinity DataKi:  4nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265302BDBM50265302(CHEMBL4060537)
Affinity DataKi:  4nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 6(Human)
University of Gdansk

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265186BDBM50265186(CHEMBL4091172)
Affinity DataKi:  4.10nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
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