Report error Found 456 Enz. Inhib. hit(s) with Target = 'RAC-alpha serine/threonine-protein kinase [E17K]'
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 2nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 50nMAssay Description:Purified human recombinant kinase full-length AKT1 E17K was expressed in insect cells and activated in vitro by PDPK1. UlightTM-CREBtide (PerkinElmer...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 80nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataKi: 94nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K]/RAC-beta serine/threonine-protein kinase(Human)
Terremoto Biosciences
US Patent
Terremoto Biosciences
US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Human)
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent

3D Structure (crystal)













































