Compile Data Set for Download or QSAR
Report error Found 136 Enz. Inhib. hit(s) with Target = 'RecQ-like DNA helicase BLM'
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440514BDBM50440514(CHEMBL2426190)
Affinity DataIC50: 100nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440527BDBM50440527(CHEMBL2426164)
Affinity DataIC50: 110nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440533BDBM50440533(CHEMBL2426169)
Affinity DataIC50: 300nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544291BDBM50544291(CHEMBL4633662)
Affinity DataKd:  760nMAssay Description:Binding affinity to wild-type His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by isothermal cal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544291BDBM50544291(CHEMBL4633662)
Affinity DataIC50: 800nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50619887BDBM50619887(CHEMBL5423610)
Affinity DataIC50: 800nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440528BDBM50440528(CHEMBL2426165)
Affinity DataIC50: 910nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50505091BDBM50505091(CHEMBL4075790)
Affinity DataIC50: 950nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in BLM helicase unwinding activity using...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440538BDBM50440538(CHEMBL2426174)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440517BDBM50440517(CHEMBL2426193)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50619881BDBM50619881(CHEMBL5440285)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544262BDBM50544262(CHEMBL4647093)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 48721BDBM48721(SMR000178207 | 1-(3,4-Dichloro-phenyl)-3-(5-pyridi...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544291BDBM50544291(CHEMBL4633662)
Affinity DataKd:  1.40E+3nMAssay Description:Binding affinity to His-tagged BLM H996A mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by isothermal calorimetric titration ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50505091BDBM50505091(CHEMBL4075790)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440519BDBM50440519(CHEMBL2426195)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50044626BDBM50044626(CHEMBL1374426)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of BLM (unknown origin) ATPase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544277BDBM50544277(CHEMBL4646986)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440531BDBM50440531(CHEMBL2426168)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440541BDBM50440541(CHEMBL2426177)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50505091BDBM50505091(CHEMBL4075790)
Affinity DataKd:  1.80E+3nMAssay Description:Binding affinity to His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544261BDBM50544261(CHEMBL4636576)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544269BDBM50544269(CHEMBL4642601)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440524BDBM50440524(CHEMBL2426161)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440531BDBM50440531(CHEMBL2426168)
Affinity DataIC50: 2.15E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in BLM helicase unwinding activity using...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544287BDBM50544287(CHEMBL4648936)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50619886BDBM50619886(CHEMBL5424781)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50619869BDBM50619869(CHEMBL5433468)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544264BDBM50544264(CHEMBL4649302)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544275BDBM50544275(CHEMBL4632583)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544289BDBM50544289(CHEMBL4647563)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50619885BDBM50619885(CHEMBL5437731)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544288BDBM50544288(CHEMBL4647503)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440531BDBM50440531(CHEMBL2426168)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of BLM helicase (unknown origin) binding to DNAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544266BDBM50544266(CHEMBL4649146)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440522BDBM50440522(CHEMBL2426159)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544263BDBM50544263(CHEMBL4637928)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544265BDBM50544265(CHEMBL4634966)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50651694BDBM50651694(5,5''-indigotindisulfonic acid | Blue x | Indigo c...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of BLM (unknown origin) ATPase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440506BDBM50440506(CHEMBL2426200)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544290BDBM50544290(CHEMBL4640219)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50619876BDBM50619876(CHEMBL5433068)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50505091BDBM50505091(CHEMBL4075790)
Affinity DataIC50: 3.95E+3nMAssay Description:Inhibition of 5'-biotin labeled duplex forked-DNA binding to BLM (unknown origin) assessed as increase in unbound DNA levels after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50619873BDBM50619873(CHEMBL5425282)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440509BDBM50440509(CHEMBL2426179)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544268BDBM50544268(CHEMBL4637736)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440510BDBM50440510(CHEMBL2426181)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50544273BDBM50544273(CHEMBL4642239)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50619884BDBM50619884(CHEMBL5405727)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440512BDBM50440512(CHEMBL2426187)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
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