Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase Nek2 [T175A]'
TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259811BDBM259811(US9505766, 11)
Affinity DataIC50: 109nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259836BDBM259836(US9505766, 40)
Affinity DataIC50: 189nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259819BDBM259819(US9505766, 20)
Affinity DataIC50: 200nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259818BDBM259818(US9505766, 18)
Affinity DataIC50: 211nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259832BDBM259832(US9505766, 36)
Affinity DataIC50: 440nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259810BDBM259810(US9505766, 10)
Affinity DataIC50: 900nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259825BDBM259825(US9505766, 29)
Affinity DataIC50: 1.00E+3nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259822BDBM259822(US9505766, 23)
Affinity DataIC50: 1.00E+3nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259820BDBM259820(US9505766, 21)
Affinity DataIC50: 1.00E+3nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259837BDBM259837(US9505766, 41)
Affinity DataIC50: 1.14E+3nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259815BDBM259815(US9505766, 15)
Affinity DataIC50: 3.00E+3nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259812BDBM259812(US9505766, 12)
Affinity DataIC50: 3.00E+3nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259813BDBM259813(US9505766, 13)
Affinity DataIC50: 3.00E+3nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259838BDBM259838(US9505766, 42)
Affinity DataIC50: 3.80E+3nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259824BDBM259824(US9505766, 25)
Affinity DataIC50: 6.50E+3nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259821BDBM259821(US9505766, 22)
Affinity DataIC50: 8.00E+3nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259829BDBM259829(US9505766, 33)
Affinity DataIC50: 1.00E+4nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259817BDBM259817(US9505766, 17)
Affinity DataIC50: 1.00E+4nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259814BDBM259814(US9505766, 14)
Affinity DataIC50: 1.00E+4nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259827BDBM259827(US9505766, 31)
Affinity DataIC50: 4.00E+4nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase Nek2 [T175A](Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 259826BDBM259826(US9505766, 30)
Affinity DataIC50: 3.00E+5nMpH: 7.6 T: 2°CAssay Description:For RSK2 kinase assays, see Example 64 above. Full-length human T175A NEK2 (referred to as NEK2) was expressed and purified as previously described (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2017
Entry Details
US Patent