Compile Data Set for Download or QSAR
Report error Found 2289 Enz. Inhib. hit(s) with Target = 'Somatostatin receptor type 4'
TargetSomatostatin receptor type 4(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 82253BDBM82253(CAS_133073-82-2 | BIM 23052)
Affinity DataKi:  0.00200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 4(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 82253BDBM82253(CAS_133073-82-2 | BIM 23052)
Affinity DataKi:  0.00200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50097783BDBM50097783(SRIF-D-Trp8 | D-Trp8 SST-14 | CHEMBL438401 | SOMAT...)
Affinity DataKi:  0.00200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 4(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 82463BDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  0.00500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 84618BDBM84618(Leu8, D-Trp22, Tyr25 SST-28)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81767BDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataIC50: 0.0800nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor hSSTR4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50254239BDBM50254239(somatostatin-28)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2011
Entry Details
PubMed
TargetSomatostatin receptor type 4(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 82462BDBM82462(D-Nal-c[Cys-Tyr-D-Trp-Lys-Thr-Cys]-Thr-NH2 | BIM 2...)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 4(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 84630BDBM84630(BIM 23060)
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 311957BDBM311957(US10166214, Example 93 | US9789082, Example 93 | U...)
Affinity DataEC50:  0.100nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 311970BDBM311970(US10166214, Example 106 | US10675268, Example 106)
Affinity DataEC50:  0.100nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50474230BDBM50474230(CHEMBL3349516)
Affinity DataKi: <0.100nMAssay Description:Binding affinity towards human Somatostatin receptor type 4 (sst4) using Tyr11-[125I]-SRIF as radioligand was determined in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 82470BDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 4(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 82254BDBM82254(D-Nal-Cys-Tyr-D-Trp-Lys-Val-Cys-Thr-NH2 | DC-25-10...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 311957BDBM311957(US10166214, Example 93 | US9789082, Example 93 | U...)
Affinity DataEC50:  0.100nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50254239BDBM50254239(somatostatin-28)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50597579BDBM50597579(CHEMBL5197201)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 311970BDBM311970(US10166214, Example 106 | US10675268, Example 106)
Affinity DataEC50:  0.100nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50059090BDBM50059090(CHEMBL405598 | octreotide | 10-(4-Amino-butyl)-19-...)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2011
Entry Details
PubMed
TargetSomatostatin receptor type 4(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 82465BDBM82465(D-Phe-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-Abu-L-Cys(1)-L-...)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 4(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 84626BDBM84626(BIM 23034)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50474219BDBM50474219(CHEMBL3349522)
Affinity DataKi: <0.200nMAssay Description:Binding affinity towards human Somatostatin receptor type 4 (sst4) using Tyr11-[125I]-SRIF as radioligand was determined in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50474221BDBM50474221(CHEMBL3349521)
Affinity DataKi: <0.200nMAssay Description:Binding affinity towards human Somatostatin receptor type 4 (sst4) using Tyr11-[125I]-SRIF as radioligand was determined in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50597589BDBM50597589(CHEMBL5209180)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50537072BDBM50537072(CHEMBL440072)
Affinity DataKd:  0.200nMAssay Description:Displacement of [125I]somatostatin from human SSTR4 expressed in CHO-K1 cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 311971BDBM311971(US10166214, Example 107 | US9789082, Example 107 |...)
Affinity DataEC50:  0.200nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 523757BDBM523757(US11136312, Compound MM-I-87)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 311971BDBM311971(US10166214, Example 107 | US9789082, Example 107 |...)
Affinity DataEC50:  0.200nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50059090BDBM50059090(CHEMBL405598 | octreotide | 10-(4-Amino-butyl)-19-...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50097783BDBM50097783(SRIF-D-Trp8 | D-Trp8 SST-14 | CHEMBL438401 | SOMAT...)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50254239BDBM50254239(somatostatin-28)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 85246BDBM85246(Cortistatin | Cortistatin-17 | L-Asp-L-Arg-L-Met-L...)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Mouse)
Sandoz Pharma

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 82460BDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 85246BDBM85246(Cortistatin | Cortistatin-17 | L-Asp-L-Arg-L-Met-L...)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 311973BDBM311973(US10166214, Example 109 | US10675268, Example 109)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 312007BDBM312007(US10166214, Example 143 | US10675268, Example 143)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 311944BDBM311944(US10166214, Example 80 | US9789082, Example 80 | U...)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 312007BDBM312007(US10166214, Example 143 | US10675268, Example 143)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50597576BDBM50597576(CHEMBL5180543)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 311967BDBM311967(US10166214, Example 103 | US10675268, Example 103)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 311944BDBM311944(US10166214, Example 80 | US9789082, Example 80 | U...)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 311973BDBM311973(US10166214, Example 109 | US10675268, Example 109)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81767BDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 82460BDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 311967BDBM311967(US10166214, Example 103 | US10675268, Example 103)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 311994BDBM311994(US10166214, Example 130 | US10675268, Example 130)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 311994BDBM311994(US10166214, Example 130 | US10675268, Example 130)
Affinity DataEC50:  0.300nMAssay Description:The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2021
Entry Details
US Patent

TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 523756BDBM523756(US11136312, Compound MM-I-83)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50474231BDBM50474231(CHEMBL3349513)
Affinity DataKi: <0.316nMAssay Description:Binding affinity towards human Somatostatin receptor type 4 (sst4) using Tyr11-[125I]-SRIF as radioligand was determined in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 82547BDBM82547(SRIF-D-Trp8)
Affinity DataKi:  0.320nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/2/2012
Entry Details
PubMed
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