Compile Data Set for Download or QSAR
Report error Found 186 Enz. Inhib. hit(s) with Target = 'Taste receptor type 2 member 1'
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211090BDBM211090(US9247759, 5-11)
Affinity DataIC50: 14nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211181BDBM211181(US9247759, 5-128)
Affinity DataIC50: 36nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211114BDBM211114(US9247759, 5-37)
Affinity DataIC50: 54nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613033BDBM50613033(CHEMBL5279691)
Affinity DataEC50:  72nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211099BDBM211099(US9247759, 5-20)
Affinity DataIC50: 83nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211176BDBM211176(US9247759, 5-123)
Affinity DataIC50: 92nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613028BDBM50613028(CHEMBL5285591)
Affinity DataEC50:  98nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613041BDBM50613041(CHEMBL5275180)
Affinity DataEC50:  100nMAssay Description:Partial agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211179BDBM211179(US9247759, 5-126)
Affinity DataIC50: 109nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613023BDBM50613023(CHEMBL5273955)
Affinity DataEC50:  150nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613032BDBM50613032(CHEMBL5274304)
Affinity DataEC50:  160nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613021BDBM50613021(CHEMBL5277615)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613040BDBM50613040(CHEMBL5280542)
Affinity DataEC50:  180nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211119BDBM211119(US9247759, 5-43)
Affinity DataIC50: 188nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50124575BDBM50124575(CHEMBL3623735)
Affinity DataEC50:  190nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613015BDBM50613015(CHEMBL5279381)
Affinity DataEC50:  190nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 60947BDBM60947(US9247759, compound C | BDBM50443972)
Affinity DataIC50: 200nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 60947BDBM60947(US9247759, compound C | BDBM50443972)
Affinity DataIC50: 220nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613019BDBM50613019(CHEMBL3088246)
Affinity DataEC50:  230nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211101BDBM211101(US9247759, 5-22)
Affinity DataIC50: 240nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 55311BDBM55311(cid_1518966 | N-(1,3-benzodioxol-5-yl)-1,3-dimethy...)
Affinity DataIC50: 264nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211237BDBM211237(US9247759, 6-24)
Affinity DataIC50: 292nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613038BDBM50613038(CHEMBL5277281)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613018BDBM50613018(CHEMBL5278834)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613014BDBM50613014(CHEMBL5278171)
Affinity DataEC50:  330nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211169BDBM211169(US9247759, 5-115)
Affinity DataIC50: 334nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211127BDBM211127(US9247759, 5-51)
Affinity DataIC50: 342nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211159BDBM211159(US9247759, 5-153 | US9247759, 5-101)
Affinity DataIC50: 345nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211159BDBM211159(US9247759, 5-153 | US9247759, 5-101)
Affinity DataIC50: 345nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613030BDBM50613030(CHEMBL5274470)
Affinity DataEC50:  360nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613024BDBM50613024(CHEMBL5278477)
Affinity DataEC50:  380nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613016BDBM50613016(CHEMBL5275001)
Affinity DataEC50:  390nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50320146BDBM50320146(4-((N-benzyl-4-chlorophenylsulfonamido)methyl)benz...)
Affinity DataIC50: 394nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211162BDBM211162(US9247759, 5-156 | US9247759, 5-104)
Affinity DataIC50: 406nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211162BDBM211162(US9247759, 5-156 | US9247759, 5-104)
Affinity DataIC50: 406nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613022BDBM50613022(CHEMBL5289590)
Affinity DataEC50:  420nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211161BDBM211161(US9247759, 5-155 | US9247759, 5-103)
Affinity DataIC50: 429nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211161BDBM211161(US9247759, 5-155 | US9247759, 5-103)
Affinity DataIC50: 429nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 17636BDBM17636(2-{[3-(trifluoromethyl)phenyl]amino}benzoic acid |...)
Affinity DataEC50:  430nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211121BDBM211121(US9247759, 5-45)
Affinity DataIC50: 459nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211218BDBM211218(US9247759, 6-2)
Affinity DataIC50: 499nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211180BDBM211180(US9247759, 5-127)
Affinity DataIC50: 499nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613036BDBM50613036(CHEMBL5280688)
Affinity DataEC50:  540nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211081BDBM211081(US9247759, 5-2)
Affinity DataIC50: 590nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613020BDBM50613020(CHEMBL5286379)
Affinity DataEC50:  640nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613034BDBM50613034(CHEMBL5268924)
Affinity DataEC50:  640nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 50613025BDBM50613025(CHEMBL5279341)
Affinity DataEC50:  670nMAssay Description:Agonist activity at human TAS2R14 transfected in HEK293T cells assessed as IP1 accumulation measured after 150 mins by IP1 accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211173BDBM211173(US9247759, 5-119)
Affinity DataIC50: 672nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211115BDBM211115(US9247759, 5-39)
Affinity DataIC50: 678nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

TargetTaste receptor type 2 member 14(Human)
Senomyx

US Patent
LigandChemical structure of BindingDB Monomer ID 211221BDBM211221(US9247759, 6-6)
Affinity DataIC50: 706nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2017
Entry Details
US Patent

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