Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with Target = 'Ultraspiracle'
TargetUltraspiracle isoform-A(Yellowfever mosquito)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50178988BDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  25nMAssay Description:Binding affinity to Aedes aegypti EcRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488539BDBM50488539(Muristerone A)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488539BDBM50488539(Muristerone A)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488539BDBM50488539(Muristerone A)
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488539BDBM50488539(Muristerone A)
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle protein(Fall armyworm)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50326777BDBM50326777((2beta,3beta,5beta,22R)-2,3,14,20,22,25-hexahydrox...)
Affinity DataIC50: 166nMAssay Description:Binding affinity to Spodoptera frugiperda (fall armyworm) EcRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50326776BDBM50326776(2,3,14,20,22-PENTAHYDROXYCHOLEST-7-EN-6-ONE | Pona...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50326776BDBM50326776(2,3,14,20,22-PENTAHYDROXYCHOLEST-7-EN-6-ONE | Pona...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50326776BDBM50326776(2,3,14,20,22-PENTAHYDROXYCHOLEST-7-EN-6-ONE | Pona...)
Affinity DataIC50: 250nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50326776BDBM50326776(2,3,14,20,22-PENTAHYDROXYCHOLEST-7-EN-6-ONE | Pona...)
Affinity DataIC50: 280nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50326777BDBM50326777((2beta,3beta,5beta,22R)-2,3,14,20,22,25-hexahydrox...)
Affinity DataIC50: 1.05E+3nMAssay Description:Binding affinity to Nezara viridula EcRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle isoform B(Colorado potato beetle)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50226672BDBM50226672(makisterone A | CHEMBL255034)
Affinity DataIC50: 1.74E+3nMAssay Description:Binding affinity to Leptinotarsa decemlineata EcRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle isoform-A(Yellowfever mosquito)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488437BDBM50488437(CHEMBL2286416)
Affinity DataEC50:  2.14E+3nMAssay Description:Agonist activity at Aedes aegypti ecdysone receptor expressed in mammalian cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50326777BDBM50326777((2beta,3beta,5beta,22R)-2,3,14,20,22,25-hexahydrox...)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle isoform B(Colorado potato beetle)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50178988BDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  2.51E+3nMAssay Description:Binding affinity to Leptinotarsa decemlineata EcRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50326777BDBM50326777((2beta,3beta,5beta,22R)-2,3,14,20,22,25-hexahydrox...)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50326777BDBM50326777((2beta,3beta,5beta,22R)-2,3,14,20,22,25-hexahydrox...)
Affinity DataIC50: 3.00E+3nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50326777BDBM50326777((2beta,3beta,5beta,22R)-2,3,14,20,22,25-hexahydrox...)
Affinity DataIC50: 4.50E+3nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle isoform-A(Yellowfever mosquito)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488477BDBM50488477(CHEMBL2286417)
Affinity DataEC50:  5.01E+3nMAssay Description:Agonist activity at Aedes aegypti ecdysone receptor expressed in mammalian cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414646BDBM50414646(INOKOSTERONE)
Affinity DataKi:  6.00E+3nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414646BDBM50414646(INOKOSTERONE)
Affinity DataKi:  6.70E+3nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414646BDBM50414646(INOKOSTERONE)
Affinity DataIC50: 7.00E+3nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414646BDBM50414646(INOKOSTERONE)
Affinity DataIC50: 8.00E+3nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50178988BDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  1.68E+4nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50178988BDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  2.00E+4nMAssay Description:Binding affinity to Nezara viridula EcR10More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50178988BDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataIC50: 2.00E+4nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50178988BDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  2.39E+4nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50178988BDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  2.51E+4nMAssay Description:Binding affinity to Nezara viridula EcRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50178988BDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  2.51E+4nMAssay Description:Binding affinity to Nezara viridula EcR11More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50178988BDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataIC50: 2.80E+4nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414651BDBM50414651(ECDYSONE)
Affinity DataKi:  5.04E+4nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414651BDBM50414651(ECDYSONE)
Affinity DataKi:  5.11E+4nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414651BDBM50414651(ECDYSONE)
Affinity DataIC50: 6.00E+4nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR11More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetUltraspiracle(Southern green stink bug)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414651BDBM50414651(ECDYSONE)
Affinity DataIC50: 6.00E+4nMAssay Description:Displacement of [3H]PonA from recombinant Nezara viridula EcR10More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed