Compile Data Set for Download or QSAR
Report error Found 2324 Enz. Inhib. hit(s) with Target = 'WD repeat-containing protein 5'
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605331BDBM50605331(CHEMBL5190578)
Affinity DataKi: <0.0200nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605330BDBM50605330(CHEMBL5201192)
Affinity DataKi: <0.0200nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605332BDBM50605332(CHEMBL5195031)
Affinity DataKi: <0.0200nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605336BDBM50605336(CHEMBL5202831)
Affinity DataKi: <0.0200nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520141BDBM50520141(CHEMBL4462065)
Affinity DataKd: <0.0200nMAssay Description:Competitive inhibition of human N-terminal His6-SUMO tagged WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold(DE3) cells using 10-mer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605343BDBM50605343(CHEMBL5190556)
Affinity DataKi:  0.0200nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520138BDBM50520138(CHEMBL4463776)
Affinity DataKd: <0.0200nMAssay Description:Competitive inhibition of human N-terminal His6-SUMO tagged WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold(DE3) cells using 10-mer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 468736BDBM468736(US10807959, Example 5)
Affinity DataKi:  0.0200nMAssay Description:A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50631541BDBM50631541(CHEMBL5412813)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520131BDBM50520131(CHEMBL4588661)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells assessed as inhibition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50631547BDBM50631547(CHEMBL5418460)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50631548BDBM50631548(CHEMBL5418271)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50631545BDBM50631545(CHEMBL5414839)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50631546BDBM50631546(CHEMBL5411289)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605323BDBM50605323(CHEMBL5174357)
Affinity DataKi: <0.0200nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50631549BDBM50631549(CHEMBL5432148)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605325BDBM50605325(CHEMBL5199203)
Affinity DataKi: <0.0200nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50631550BDBM50631550(CHEMBL5421916)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520131BDBM50520131(CHEMBL4588661)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50631539BDBM50631539(CHEMBL5417425)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50631540BDBM50631540(CHEMBL5422217)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605355BDBM50605355(CHEMBL5170717)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50631538BDBM50631538(CHEMBL5409903)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605347BDBM50605347(CHEMBL5174178)
Affinity DataKi: <0.0200nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605346BDBM50605346(CHEMBL5177738)
Affinity DataKi: <0.0200nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520131BDBM50520131(CHEMBL4588661)
Affinity DataKd: <0.0200nMAssay Description:Competitive inhibition of human N-terminal His6-SUMO tagged WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold(DE3) cells using 10-mer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605349BDBM50605349(CHEMBL5191181)
Affinity DataKi: <0.0200nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605348BDBM50605348(CHEMBL5183319)
Affinity DataKi: <0.0200nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605350BDBM50605350(CHEMBL5177656)
Affinity DataKi: <0.0200nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605353BDBM50605353(CHEMBL5190717)
Affinity DataKi: <0.0200nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605352BDBM50605352(CHEMBL5198319)
Affinity DataKi: <0.0200nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 473225BDBM473225(US10844044, Example 283)
Affinity DataKi:  0.0200nMAssay Description:A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2021
Entry Details
US Patent

TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605350BDBM50605350(CHEMBL5177656)
Affinity DataKi: <0.0200nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605356BDBM50605356(CHEMBL5170071)
Affinity DataKi: <0.0200nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605355BDBM50605355(CHEMBL5170717)
Affinity DataKi: <0.0200nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 468925BDBM468925(US10807959, Example B64)
Affinity DataKi:  0.0210nMAssay Description:FPA Assay protocol adopted from Karatas et al. (J. Med. Chem. 2010, 5179.; J. Amer. Chem. Soc. 2013, 669.): WDR5 (Δ23, residues 24-334), is expr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605322BDBM50605322(CHEMBL5169425)
Affinity DataKi:  0.0220nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50631535BDBM50631535(CHEMBL5398730)
Affinity DataKi:  0.0230nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605327BDBM50605327(CHEMBL5181314)
Affinity DataKi:  0.0230nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520135BDBM50520135(CHEMBL4463486)
Affinity DataKd:  0.0230nMAssay Description:Competitive inhibition of human N-terminal His6-SUMO tagged WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold(DE3) cells using 10-mer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605329BDBM50605329(CHEMBL5186072)
Affinity DataKi:  0.0250nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50631534BDBM50631534(CHEMBL5398302)
Affinity DataKi:  0.0260nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50631544BDBM50631544(CHEMBL5405792)
Affinity DataKi:  0.0270nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520120BDBM50520120(CHEMBL4476662)
Affinity DataKd:  0.0270nMAssay Description:Competitive inhibition of human N-terminal His6-SUMO tagged WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold(DE3) cells using 10-mer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605337BDBM50605337(CHEMBL5192283)
Affinity DataKi:  0.0280nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605339BDBM50605339(CHEMBL5171051)
Affinity DataKi:  0.0280nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605354BDBM50605354(CHEMBL5179388)
Affinity DataKi:  0.0280nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605351BDBM50605351(CHEMBL5180435)
Affinity DataKi:  0.0290nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605324BDBM50605324(CHEMBL5182982)
Affinity DataKi:  0.0290nMAssay Description:Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Frederick National Laboratory For Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50520126BDBM50520126(CHEMBL4557848)
Affinity DataKd:  0.0300nMAssay Description:Competitive inhibition of human N-terminal His6-SUMO tagged WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold(DE3) cells using 10-mer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
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