Compile Data Set for Download or QSAR
Report error Found 227 Enz. Inhib. hit(s) with Target = 'cAMP-dependent protein kinase catalytic subunit alpha/beta/gamma'
LigandChemical structure of BindingDB Monomer ID 50188913BDBM50188913(N-((S)-1-amino-3-(2,4-dichlorophenyl)propan-2-yl)-...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of PKAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of PKAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50044004BDBM50044004(CHEMBL3356433)
Affinity DataIC50: 1nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117503BDBM50117503(CHEMBL3613621)
Affinity DataIC50: 1nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117504BDBM50117504(CHEMBL3613620)
Affinity DataIC50: 1nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117489BDBM50117489(CHEMBL3613598)
Affinity DataIC50: 1nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117631BDBM50117631(CHEMBL3613610)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117632BDBM50117632(CHEMBL3613609)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117370BDBM50117370(CHEMBL3613599)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117299BDBM50117299(CHEMBL3613605)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117629BDBM50117629(CHEMBL3613612)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 4nMAssay Description:Inhibition of Protein kinase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117630BDBM50117630(CHEMBL3613611)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117301BDBM50117301(CHEMBL3613603)
Affinity DataIC50: 5.40nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117635BDBM50117635(CHEMBL3613606)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117300BDBM50117300(CHEMBL3613604)
Affinity DataIC50: 7nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 16nMAssay Description:Inhibition of Protein kinase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117634BDBM50117634(CHEMBL3613607)
Affinity DataIC50: 22nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117315BDBM50117315(CHEMBL3613600)
Affinity DataIC50: 24nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117633BDBM50117633(CHEMBL3613608)
Affinity DataIC50: 24nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 3153BDBM3153(CHEMBL52529 | 2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4...)
Affinity DataIC50: 30nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50285250BDBM50285250(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50: 30nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2005
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 3149BDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataIC50: 60nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2005
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50117627BDBM50117627(CHEMBL3613614)
Affinity DataIC50: 69nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 3152BDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50: 70nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50285251BDBM50285251(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50: 70nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2005
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 3149BDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataIC50: 80nMAssay Description:Inhibition of cAMP-dependent protein kinase (Protein kinase A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 80nMAssay Description:Inhibition of protein kinase A (PKA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117303BDBM50117303(CHEMBL3613601)
Affinity DataIC50: 81nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117302BDBM50117302(CHEMBL3613602)
Affinity DataIC50: 150nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50215105BDBM50215105(CHEMBL3143641)
Affinity DataEC50:  150nMAssay Description:Activation of cAMP dependent protein kinase (PKA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50117502BDBM50117502(CHEMBL3613622)
Affinity DataIC50: 332nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 3149BDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataIC50: 790nMAssay Description:Inhibition of cAMP-dependent protein kinase (Protein kinase A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50117505BDBM50117505(CHEMBL3613619)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117581BDBM50117581(CHEMBL3613618)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117598BDBM50117598(CHEMBL3613617)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192071BDBM50192071((13R,15S)-13-methyl-16-oxa-8,9,12,22,24-pentaazahe...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PKAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117501BDBM50117501(CHEMBL3613623)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117625BDBM50117625(CHEMBL3613616)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117500BDBM50117500(CHEMBL3613624)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117626BDBM50117626(CHEMBL3613615)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50117628BDBM50117628(CHEMBL3613613)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 3154BDBM3154(2-({2,6-dihydroxy-4-[({3-[(4-hydroxybenzene)amido]...)
Affinity DataIC50: 1.90E+3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2005
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 3158BDBM3158(2-{[2,6-dihydroxy-4-({[(4S)-3-[(4-hydroxybenzene)a...)
Affinity DataIC50: 2.00E+3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2005
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 2581BDBM2581(CHEMBL16958 | 3,13,23-triazahexacyclo[14.7.0.0^{2,...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Protein kinase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50213033BDBM50213033(CHEMBL329274)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of c-AMP dependent kinase (PKA) using histone II A proteinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 2672BDBM2672(6,7,12,13-Tetrahydro-5,7-dioxo-5H-indolo[2,3-a]pyr...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Protein kinase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50290416BDBM50290416({4-[1-(3-Amino-propyl)-1H-indol-4-yl]-pyrimidin-2-...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of protein kinase A.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50366348BDBM50366348(CHEMBL1233654)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of c-AMP dependent kinase (PKA) using histone II A proteinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 4078BDBM4078(Elagic Acid | CHEMBL6246 | 6,7,13,14-tetrahydroxy-...)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of PKAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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