1891 SMILES Strings for Sodium- and chloride-dependent glycine transporter 1

Compound Name
SMILES String
COCCCN1CCC(CC1)NC(=O)c1cc(Cl)c(N)c2CCOc12
O=S(=O)(CC1CC1)NCCOc1ccc2CCC([C@@H](Cc3ccccc3)c2c1)N1CCC1 |r|
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(C(Cc3cccc(F)c3)c2c1)N1CCCC1
COc1cc(cc(SC)c1C(=O)N[C@H]1COCC[C@H]1N1CCCC1)C(F)(F)F |r|
COc1cc(cc(SC)c1C(=O)N[C@H]1COCC[C@@H]1N1CCCC1)C(F)(F)F |r|
COc1cc(cc(SC)c1C(=O)N[C@H]1COCC[C@H]1NC1CCC1)C(F)(F)F |r|
COc1cc(cc(SC)c1C(=O)N[C@H]1COCC[C@@H]1NC1CCC1)C(F)(F)F |r|
COc1cc(cc(SC)c1C(=O)N[C@@H]1COCC[C@H]1N1CCCC1)C(F)(F)F |r|
COc1cc(cc(SC)c1C(=O)N[C@H]1COCC[C@@H]1N1CCC(O)C1)C(F)(F)F |r|
FC(F)(F)c1ccc(C(=O)N[C@@H]2COCC[C@H]2N2CCCC2)c(c1)C1CC1 |r|
CSc1cc(cc(c1C(=O)N[C@@H]1COCC[C@H]1N1CCCC1)C(F)(F)F)C(F)(F)F |r|
Cc1cc(cc(c1C(=O)N[C@@H]1COCC[C@H]1N1CCCC1)C(F)(F)F)C(F)(F)F |r|
COc1cc(cc(SC)c1C(=O)N[C@@H]1COCC[C@H]1NC1CCCC1)C(F)(F)F |r|
FC(F)(F)c1ccc(C(=O)N[C@@H]2COCC[C@H]2NC2CCCC2)c(c1)C1CC1 |r|
CSc1cc(cc(c1C(=O)N[C@@H]1COCC[C@H]1NC1CCCC1)C(F)(F)F)C(F)(F)F |r|
FC(F)(F)c1ccc(C(=O)N[C@@H]2COCC[C@H]2NC2CCCCC2)c(c1)C1CC1 |r|
FC(F)(F)c1cc(C2CC2)c(C(=O)N[C@@H]2COCC[C@H]2N2CCCC2)c(c1)C(F)(F)F |r|
CC(C)N[C@@H]1CCOC[C@H]1NC(=O)c1ccc(cc1C1CC1)C(F)(F)F |r|
FC(F)(F)c1ccc(C(=O)N[C@@H]2COCC[C@H]2NC2CCOCC2)c(c1)C1CC1 |r|
FC(F)(F)c1ccc(C(=O)N[C@@H]2COCC[C@H]2NCC2CC2)c(c1)C1CC1 |r|
FC(F)(F)c1ccc(C(=O)N[C@@H]2COCC[C@H]2N2CCCCC2)c(c1)C1CC1 |r|
FC(F)(F)c1ccc(C(=O)N[C@@H]2COCC[C@H]2NC2CC2)c(c1)C1CC1 |r|
Cc1cc(cc(C)c1C(=O)N[C@@H]1COCC[C@H]1N1CCCC1)C(F)(F)F |r|
COc1cc(cc(C)c1C(=O)N[C@@H]1COCC[C@H]1N1CCCC1)C(F)(F)F |r|
CCc1cc(cc(CC)c1C(=O)N[C@@H]1COCC[C@H]1N1CCCC1)C(F)(F)F |r|
CCc1cc(cc(OC)c1C(=O)N[C@@H]1COCC[C@H]1N1CCCC1)C(F)(F)F |r|
COc1cc(cc(SC)c1C(=O)N[C@@H]1COCC[C@H]1NC1(C)CCCCC1)C(F)(F)F |r|
CCc1cc(cc(C)c1C(=O)N[C@@H]1COCC[C@H]1N1CCCC1)C(F)(F)F |r|
COc1cc(cc(C2CC2)c1C(=O)N[C@@H]1COCC[C@H]1N1CCCC1)C(F)(F)F |r|
COc1cc(cc(SC)c1C(=O)N[C@@H]1COCC[C@H]1NC1(C)CCCC1)C(F)(F)F |r|
CC1(CCCC1)N[C@@H]1CCOC[C@H]1NC(=O)c1ccc(cc1C1CC1)C(F)(F)F |r|
CC(N[C@@H]1CCOC[C@H]1NC(=O)c1ccc(cc1C1CC1)C(F)(F)F)C1CC1 |r|
COc1cc(cc(SC)c1C(=O)N[C@@H]1COCC[C@H]1NC(C)C1CC1)C(F)(F)F |r|
FC(F)(F)c1ccc(C(=O)N[C@@H]2COCC[C@H]2NC2CCC2)c(c1)C1CC1
COc1cc(cc(SC)c1C(=O)N[C@@H]1COCC[C@H]1NC1CCC(O)CC1)C(F)(F)F |r,wU:18.20,wD:13.13,(1.33,3.08,;1.33,1.54,;2.67,.77,;4,1.54,;5.33,.77,;5.33,-.77,;4,-1.54,;4,-3.08,;5.33,-3.85,;2.67,-.77,;1.33,-1.54,;1.33,-3.08,;,-.77,;-1.33,-1.54,;-1.33,-3.08,;-2.67,-3.85,;-4,-3.08,;-4,-1.54,;-2.67,-.77,;-2.67,.77,;-4,1.54,;-4,3.08,;-5.33,3.85,;-6.67,3.08,;-8,3.85,;-6.67,1.54,;-5.33,.77,;6.67,1.54,;8,2.31,;6.67,3.08,;8,.77,)|
COc1cc(cc(SC)c1C(=O)N[C@@H]1COCC[C@H]1N1C[C@@H]2C[C@@H]2C1)C(F)(F)F |r|
FC(F)(F)c1ccc(C(=O)N[C@@H]2COCC[C@H]2N2C[C@@H]3C[C@@H]3C2)c(c1)C1CC1 |r|
OC1CCN(CC1)[C@@H]1CCOC[C@H]1NC(=O)c1ccc(cc1C1CC1)C(F)(F)F |r|
FC(F)(F)c1ccc(C(=O)N[C@H]2COCC[C@@H]2N2CCCC2)c(c1)C1CC1 |r|
Cc1cc(cc(c1C(=O)N[C@H]1COCC[C@@H]1N1CCCC1)C(F)(F)F)C(F)(F)F |r|
CSc1cc(cc(c1C(=O)N[C@H]1COCC[C@@H]1N1CCCC1)C(F)(F)F)C(F)(F)F |r|
FC(F)(F)c1ccc(C(=O)N[C@H]2COCC[C@@H]2NC2CCCC2)c(c1)C1CC1 |r|
COc1cc(cc(SC)c1C(=O)N[C@H]1COCC[C@@H]1NC1CCCC1)C(F)(F)F |r|
FC(F)(F)c1cc(C2CC2)c(C(=O)N[C@H]2COCC[C@@H]2N2CCCC2)c(c1)C(F)(F)F |r|
FC(F)(F)c1ccc(C(=O)N[C@H]2COCC[C@@H]2NC2CCCCC2)c(c1)C1CC1 |r|
Cc1cc(cc(C)c1C(=O)N[C@H]1COCC[C@@H]1N1CCCC1)C(F)(F)F |r|
COc1cc(cc(C)c1C(=O)N[C@H]1COCC[C@@H]1N1CCCC1)C(F)(F)F |r|
CCc1cc(cc(OC)c1C(=O)N[C@H]1COCC[C@@H]1N1CCCC1)C(F)(F)F |r|
COc1cc(cc(C2CC2)c1C(=O)N[C@H]1COCC[C@@H]1N1CCCC1)C(F)(F)F |r|
COc1cc(cc(SC)c1C(=O)N[C@@H]1COCC[C@H]1N1CCC2CC12)C(F)(F)F |r|
OC1CCN(C1)[C@@H]1CCOC[C@H]1NC(=O)c1ccc(cc1C1CC1)C(F)(F)F |r|
COc1cc(cc(SC)c1C(=O)N[C@@H]1CCOC[C@@H]1N1CCCC1)C(F)(F)F |r|
COc1cc(cc(SC)c1C(=O)N[C@H]1CCOC[C@H]1N1CCCC1)C(F)(F)F |r|
Cn1cnc(c1)S(=O)(=O)NCc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CC2CC2C1
Cn1cc(cn1)S(=O)(=O)NCCOc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CC2CC2C1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(C(Cc3ccccc3F)c2c1)N1CC2CC2C1
CCS(=O)(=O)NCc1ccc2CCC(NC3(COC3)C#N)C(Cc3ccccc3)c2c1
CCCS(=O)(=O)NCc1ccc2CCC(NC3(COC3)C#N)C(Cc3ccccc3)c2c1
O=S(=O)(NCc1ccc2CCC(NC3(COC3)C#N)C(Cc3ccccc3)c2c1)C1CCC1
O=S(=O)(CC1CC1)NCc1ccc2CCC(NC3(COC3)C#N)C(Cc3ccccc3)c2c1
Cn1cnc(c1)S(=O)(=O)NCCOc1cc2C(Cc3ccccc3)C(CCc2cc1[N+]#[C-])N1CC2CC2C1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNC(=O)c3ccc(Cl)cc3Cl)cc12
CS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNC(=O)c3ccccc3)cc12
CCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CC(C)C(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CC(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CC(C)CS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3ccc4ccccc4c3)cc12
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3cccnc3)cc12
FC(F)(F)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CS(=O)(=O)NCCOc1cc2C(NCCc2cc1F)C1(CCC1)c1ccc(Cl)cc1
Fc1cc2CCNC(c2cc1OCCNS(=O)(=O)c1ccccc1)C1(CCC1)c1ccc(Cl)cc1
Fc1cc2CCNC(c2cc1OCCNS(=O)(=O)c1cccnc1)C1(CCC1)c1ccc(Cl)cc1
CCCS(=O)(=O)NCCOc1cc2C(NCCc2cc1F)C1(CCC1)c1ccc(Cl)cc1
CCCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3cccs3)cc12
COc1ccccc1S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
COc1cccc(c1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3ccc(s3)-c3ccon3)cc12
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3ccccc3C#N)cc12
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3ccc(cc3)C#N)cc12
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3ccccc3Cl)cc12
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3cccc(Cl)c3)cc12
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3ccc(Cl)cc3)cc12
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)C3CC3)cc12
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3ccc(Cl)nc3)cc12
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3cccc4cccnc34)cc12
COc1ccc(cc1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)Cc3ccccc3)cc12
CCCNC(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNC(=O)Nc3ccccc3)cc12
Cc1nn(C)cc1S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CC(C)NC(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Cn1cc(cn1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CC(C)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CCCCS(=O)(=O)NCCOc1ccc2CCN(C(c2c1)C1(CCC1)c1ccc(Cl)cc1)C(=O)NCC
CCCCS(=O)(=O)NCCOc1ccc2CCN(C)C(c2c1)C1(CCC1)c1ccc(Cl)cc1
CCS(=O)(=O)N1CCN(CC1)c1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNC(=O)Nc3cccnc3)cc12
Cn1cc(cn1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CC(F)(F)C1)c1ccc(Cl)cc1
CCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CC(F)(F)C1)c1ccc(Cl)cc1
CCCS(=O)(=O)NCCN(CCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1)S(=O)(=O)CCC
CCCS(=O)(=O)NCCOc1ccc2CCN(C(c2c1)C1(CCC1)c1ccc(Cl)cc1)C(=N)NC#N
CCCS(=O)(=O)NCCOc1ccc2CCN(C(c2c1)C1(CCC1)c1ccc(Cl)cc1)C(N)=N
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCC(=O)N3CCNCC3)cc12
CCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1cccc(Cl)c1
CCCS(=O)(=O)NCCOc1ccc2CC[NH2+]C(c2c1)C1(CCC1)c1ccccc1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CC[NH2+]C(c2c1)C1(CCC1)c1ccc(Cl)cc1
Cc1nc(cn1C)S(=O)(=O)NCCOc1ccc2CC[NH2+]C(c2c1)C1(CCC1)c1ccc(Cl)cc1
CCOC(=O)N1CCN(CC1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)N3CCNCC3)cc12
CCCS(=O)(=O)N1CCN(CC1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3c[nH]cn3)cc12
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3ccc(NCc4ccccc4)nc3)cc12
CCCNc1ccc(cn1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CCCS(=O)(=O)NCCOc1ccc2CCNC(C(C(C)C)c3ccc(Cl)cc3)c2c1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)C3CCCNC3)cc12
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3ccccc3)cc12
CCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(F)cc1
Fc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3cccnc3)cc12
CCCS(=O)(=O)NCCOc1ccc2c(c1)C(NCC2(C)C)C1(CCC1)c1ccc(Cl)cc1
CCCS(=O)(=O)NCCOc1ccc2C(NCCc2c1)C1(CCC1)c1ccc(Cl)cc1
CCN(CC)S(=O)(=O)NCCOc1ccc2c(c1)C(NCC2(C)C)C1(CCC1)c1ccc(Cl)cc1
CCCS(=O)(=O)NCCOc1ccc2CCN(C(c2c1)C1(CCC1)c1ccc(F)cc1)C(=O)C(F)(F)F
CCCS(=O)(=O)NCCOc1ccc2CCN(CC(F)(F)F)C(c2c1)C1(CCC1)c1ccc(F)cc1
CCCS(=O)(=O)NCCOc1ccc2CCN(C(c2c1)C1(CCC1)c1ccc(F)cc1)C(N)=N
CCCS(=O)(=O)NCCOc1cc(Br)c2CCNC(c2c1)C1(CCC1)c1ccc(F)cc1
CCCS(=O)(=O)NCCOc1ccc2CCN(N=O)C(c2c1)C1(CCC1)c1ccc(F)cc1
CCCS(=O)(=O)NCCOc1ccc2CCN(N)C(c2c1)C1(CCC1)c1ccc(F)cc1
CCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1OC
CCCS(=O)(=O)NCCOc1ccc2CCN(CC#N)C(c2c1)C1(CCC1)c1cccc(Cl)c1
CCCS(=O)(=O)NCCOc1ccc2CCN(CCN)C(c2c1)C1(CCC1)c1cccc(Cl)c1
CCCS(=O)(=O)NCCOc1ccc2CCN(C(c2c1)C1(CCC1)c1ccc(F)cc1)c1ncc[nH]1
CCCS(=O)(=O)NCCOc1ccc2CCN(CC#N)C(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCCS(=O)(=O)N3CCOCC3)cc12
CCCNS(=O)(=O)CCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CCCS(=O)(=O)N1CCN(CC1)c1cc2CCN(C(c2cc1OC)C1(CCC1)c1ccc(Cl)cc1)S(=O)(=O)CCC
Clc1ccc(cc1)C1(CC1)C1NCCc2ccc(OCCNS(=O)(=O)c3cccnc3)cc12
Cn1cc(cn1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CC1)c1ccc(Cl)cc1
CCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CC1)c1ccc(Cl)cc1
CCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1cccc(F)c1
Fc1cccc(c1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3cccnc3)cc12
CC(C)(O)CS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Fc1cccc(c1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3cccs3)cc12
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(CNS(=O)(=O)c3cccnc3)cc12
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCCS(=O)(=O)Nc3ccccc3)cc12
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(Oc3ccccc3NS(=O)(=O)c3cccs3)cc12
CC(C)NS(=O)(=O)CCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CC(C)(C)NS(=O)(=O)CCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
COc1ccccc1NS(=O)(=O)CCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CC(C)(C)OC(=O)N1CCN(CC1)S(=O)(=O)CCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CC(C)(C)OC(=O)NCCNS(=O)(=O)CCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
NCCNS(=O)(=O)CCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CN(C)CCNS(=O)(=O)CCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCCS(=O)(=O)N3CCNCC3)cc12
COCCNS(=O)(=O)CCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)c(N)c1
CCCS(=O)(=O)NCCOc1ccc2CCNC(C(C)c3ccc(Cl)cc3)c2c1
NCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CC(C)(C)CS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Nc1ccc(cn1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1nc2sccn2c1S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C(O)(c1ccc(Cl)cc1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)CCN3C(=O)c4ccccc4C3=O)cc12
CN(C)CCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CCCN1CCN(CC1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CCCNCCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CCNCCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CCN(CC)CCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CC(C)NCCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)CCCN3CCCCC3)cc12
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)CCCN3CCOCC3)cc12
CCNC(=O)NCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
C\C=C\S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CCCS(=O)(=O)NCCNc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CCCS(=O)(=O)NCc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Cn1cc(cn1)S(=O)(=O)NCc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(cc12)C#N
Cn1cnc(c1)S(=O)(=O)NCc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
FCCCS(=O)(=O)NCc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CCCS(=O)(=O)NCc1ccc2CCNC(c2c1)C(C)(C)c1ccc(Cl)cc1
OCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccccn1
CCCS(=O)(=O)NCC(=O)Nc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Cn1cc(cn1)S(=O)(=O)NCc1ccc2CCNC(c2c1)C(C)(C)c1ccc(Cl)cc1
Cn1cnc(c1)S(=O)(=O)NCc1ccc2CCNC(c2c1)C(C)(C)c1ccc(Cl)cc1
FCCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccccn1
CCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1cccc(Cl)n1
CC(C)(C1NCCc2ccc(cc12)C#N)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCCS(=O)(=O)Nc3ccccn3)cc12
FCCc1ccc(cc1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Cn1cnc(c1)S(=O)(=O)NCC(=O)Nc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Cn1cc(cn1)S(=O)(=O)NCC(=O)Nc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
FCCCc1ccc(cc1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(Oc3ccc(NS(=O)(=O)c4cccs4)cc3)cc12
CCCS(=O)(=O)Nc1ccc(Oc2ccc3CCNC(c3c2)C2(CCC2)c2ccc(Cl)cc2)nc1
CCCS(=O)(=O)Oc1ccc2CCNC(c2c1)C1(CCC1)c1cccc(F)c1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(Oc3ccccc3NS(=O)(=O)c3cccnc3)cc12
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(Oc3ccc(NS(=O)(=O)c4cccs4)cn3)cc12
CCCS(=O)(=O)NCc1ccc2CCNC(c2c1)C1(CCC1)c1ccccn1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(Oc3ncccc3NS(=O)(=O)c3cccs3)cc12
CCCS(=O)(=O)Nc1cccnc1Oc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
N#Cc1ccc2CCNC(c2c1)C1(CCC1)c1ccccn1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(Oc3ccc(NS(=O)(=O)c4cccnc4)cn3)cc12
O=S(=O)(CC1CC1)NCc1ccc2CCNC(c2c1)C1(CCC1)c1ccccn1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(Oc3ncccc3NS(=O)(=O)c3cccnc3)cc12
NCCCNS(=O)(=O)CCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C(C)(C)c1ccc(Cl)cc1
FCCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CN(C)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
FC(F)(F)CCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Nc1ccc(cc1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)C3CCNC3)cc12
CN(C)CCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Nc1ncc(cn1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3cn[nH]c3)cc12
COc1ccc(cn1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Nc1cccc(c1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)CCN3CCCCC3)cc12
CNc1nnc(s1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Nc1ncc(s1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)C3CNC3)cc12
CC(C)NCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)C3CCN(C3)C(=O)OCc3ccccc3)cc12
CCCS(=O)(=O)NCCOc1ccc2CCN(C(c2c1)C1(CCC1)c1ccc(Cl)cc1)C(C)=O
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3ccc(Oc4ccccc4)nc3)cc12
CCCS(=O)(=O)N(CCN)CCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)C3CCN(Cc4ccccc4)CC3)cc12
CNCCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CC(=O)N1CC(C1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
NCCCCS(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CN1CCOc2cc(cnc12)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CC(=O)Nc1ncc(s1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3ccc(nc3)N3CCOCC3)cc12
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)C3CCNCC3)cc12
NC(=O)Nc1ccc(cc1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Cc1oncc1S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CCC1)C1NCCc2ccc(OCCNS(=O)(=O)c3ncn[nH]3)cc12
Nc1n[nH]c(n1)S(=O)(=O)NCCOc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
Cn1cnc(c1)S(=O)(=O)N1CCc2ccc(cc2C1)C(CN)Cc1ccccc1
Cn1cc(cn1)S(=O)(=O)N1CCc2ccc(cc2C1)C(CN)Cc1ccccc1
NCC(Cc1ccccc1)c1ccc2CCN(Cc2c1)S(=O)(=O)CC1CC1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CC[C@@H](CN)[C@@H](Cc3ccccc3)c2c1 |r|
CCS(=O)(=O)NCCOc1ccc2CC[C@@H](CN)[C@@H](Cc3ccccc3)c2c1 |r|
NC[C@@H]1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2[C@@H]1Cc1ccccc1 |r|
CNC[C@@H]1CCc2ccc(OCCNS(=O)(=O)c3cn(C)cn3)cc2[C@@H]1Cc1ccccc1 |r|
CCS(=O)(=O)NCCOc1ccc2CC[C@@H](CNC)[C@@H](Cc3ccccc3)c2c1 |r|
CNC[C@@H]1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2[C@@H]1Cc1ccccc1 |r|
CCS(=O)(=O)NCCOc1ccc2CC[C@@H](CN3CCC3)[C@@H](Cc3ccccc3)c2c1 |r|
O=S(=O)(CC1CC1)NCCOc1ccc2CC[C@@H](CN3CCC3)[C@@H](Cc3ccccc3)c2c1 |r|
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CC[C@@H](CN3CCC3)[C@@H](Cc3ccccc3)c2c1 |r|
Cn1cnc(c1)S(=O)(=O)NCc1ccc2CC[C@@H](CN3CCC3)[C@@H](Cc3ccccc3)c2c1 |r|
CCOC(=O)NC1CCc2ccc(OCCNC(=O)OC(C)(C)C)cc2C1Cc1ccc(Cl)c(Cl)c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3cn(C)cn3)cc2C1Cc1ccc(Cl)c(Cl)c1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(Cl)c(Cl)c3)c2c1
Cn1cc(cn1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(Cl)c(Cl)c3)c2c1
NC1CCc2ccc(OCCNS(=O)(=O)c3cccnc3)cc2C1Cc1ccc(Cl)c(Cl)c1
CCCS(=O)(=O)NCCOc1ccc2CCC(C(Cc3ccc(Cl)c(Cl)c3)c2c1)N(C)C
CCCS(=O)(=O)NCCOc1ccc2CCC(NC(=O)OCC)C(Cc3ccc(Cl)c(Cl)c3)c2c1
CCCS(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(Cl)c(Cl)c3)c2c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3cnn(C)c3)cc2C1Cc1ccc(Cl)c(Cl)c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3cccnc3)cc2C1Cc1ccc(Cl)c(Cl)c1
CCCS(=O)(=O)N(C)CCOc1ccc2CCC(N)C(Cc3ccc(Cl)c(Cl)c3)c2c1
CCOC(=O)NC1CCc2ccc(OCCNS(C)(=O)=O)cc2C1Cc1ccc(Cl)c(Cl)c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3ccccc3)cc2C1Cc1ccc(Cl)c(Cl)c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3cccs3)cc2C1Cc1ccc(Cl)c(Cl)c1
CS(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(Cl)c(Cl)c3)c2c1
NC1CCc2ccc(OCCNS(=O)(=O)c3ccccc3)cc2C1Cc1ccc(Cl)c(Cl)c1
NC1CCc2ccc(OCCNS(=O)(=O)c3cccs3)cc2C1Cc1ccc(Cl)c(Cl)c1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(NC(=O)C(F)(F)F)C(Cc3ccc(Cl)c(Cl)c3)c2c1
NC1CCc2ccc(OCCNS(=O)(=O)C3CCNC3)cc2C1Cc1ccc(Cl)c(Cl)c1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(NC=O)C(Cc3ccc(Cl)c(Cl)c3)c2c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3cc(C)cs3)cc2C1Cc1ccc(Cl)c(Cl)c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)CCCF)cc2C1Cc1ccc(Cl)c(Cl)c1
CCNC1CCc2ccc(OCCNS(=O)(=O)c3cn(C)cn3)cc2C1Cc1ccc(Cl)c(Cl)c1
Cc1csc(c1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(Cl)c(Cl)c3)c2c1
CN(C)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(Cl)c(Cl)c3)c2c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)CCC(F)(F)F)cc2C1Cc1ccc(Cl)c(Cl)c1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(Cl)cc3)c2c1
Cn1cc(cn1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(Cl)cc3)c2c1
CCOC(=O)NC1CCc2ccc(OS(=O)(=O)C(F)(F)F)cc2C1Cc1ccc(Cl)c(Cl)c1
NC1CCc2ccc(cc2C1Cc1ccc(Cl)cc1)C#N
NC1CCc2ccc(CNS(=O)(=O)CCCF)cc2C1Cc1ccccc1
CCOC(=O)NC1CCc2ccc(cc2C1Cc1ccc(Cl)c(Cl)c1)C#N
NC1CCc2ccc(OCCN3CCCS3(=O)=O)cc2C1Cc1cccc(Cl)c1
CC(C)(C)OC(=O)NC1CCc2ccc(cc2C1Cc1ccc(Cl)c(Cl)c1)C#N
NC1CCc2ccc(O)cc2C1Cc1ccc(Cl)c(Cl)c1
CC(C)(C)OC(=O)NC1CCc2ccc(OC(F)F)cc2C1Cc1ccc(Cl)cc1
Oc1ccc2CCC(NC(=O)OCc3ccccc3)C(Cc3ccc(Cl)cc3)c2c1
CC(C)(C)OC(=O)NC1CCc2ccc(CN)cc2C1Cc1ccc(Cl)c(Cl)c1
CCCS(=O)(=O)NCc1ccc2CCC(NC(=O)OC(C)(C)C)C(Cc3ccc(Cl)c(Cl)c3)c2c1
CCCS(=O)(=O)NCc1ccc2CCC(N)C(Cc3ccc(Cl)c(Cl)c3)c2c1
NC1CCc2ccc(CNS(=O)(=O)CCCF)cc2C1Cc1ccc(Cl)c(Cl)c1
CCCS(=O)(=O)NCc1ccc2CCC(N)C(Cc3ccccc3)c2c1
NC1CCc2ccc(CNS(=O)(=O)C3CCC3)cc2C1Cc1ccccc1
NC1CCc2ccc(CNS(=O)(=O)CC3CC3)cc2C1Cc1ccccc1
CCCS(=O)(=O)N(C)Cc1ccc2CCC(N)C(Cc3ccccc3)c2c1
CCOC(=O)NC1CCc2ccc(OCCNC(=O)OC(C)(C)C)cc2C1Cc1cccc(Cl)c1
Cn1cc(cn1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3sc(C)nc3C)cc2C1Cc1cccc(Cl)c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3cccs3)cc2C1Cc1cccc(Cl)c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3ccc(Cl)s3)cc2C1Cc1cccc(Cl)c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3cnc(C)s3)cc2C1Cc1cccc(Cl)c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3ccc(C)s3)cc2C1Cc1cccc(Cl)c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3cc(C)cs3)cc2C1Cc1cccc(Cl)c1
CCCS(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
NC1CCc2ccc(OCCNS(=O)(=O)c3cccs3)cc2C1Cc1cccc(Cl)c1
Cc1nc(C)c(s1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
Cc1ncc([nH]1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
NC1CCc2ccc(OCCNS(=O)(=O)c3ccc(Cl)s3)cc2C1Cc1cccc(Cl)c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3cc(C)sc3C)cc2C1Cc1cccc(Cl)c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3cnn(CC)c3)cc2C1Cc1cccc(Cl)c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3cnn(C)c3)cc2C1Cc1ccc(Cl)cc1Cl
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3cccs3)cc2C1Cc1ccc(Cl)cc1Cl
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3ccc(C)s3)cc2C1Cc1ccc(Cl)cc1Cl
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)CC)cc2C1Cc1cccc(Cl)c1
CCn1cc(cn1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
Cc1csc(c1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
Cc1ccc(s1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
Cc1cc(c(C)s1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
CCS(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
Cn1cc(cn1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(Cl)cc3Cl)c2c1
NC1CCc2ccc(OCCNS(=O)(=O)c3cccs3)cc2C1Cc1ccc(Cl)cc1Cl
Cc1ccc(s1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(Cl)cc3Cl)c2c1
CCCS(=O)(=O)NCCOc1ccc2CCC(NC(=O)OCC)C(Cc3ccc(Cl)cc3Cl)c2c1
CCCS(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(Cl)cc3Cl)c2c1
CCCS(=O)(=O)N(C)CCOc1ccc2CCC(NC(=O)OCC)C(Cc3ccc(Cl)cc3)c2c1
CCCS(=O)(=O)N(C)CCOc1ccc2CCC(N)C(Cc3ccc(Cl)cc3)c2c1
CCCS(=O)(=O)N(C)CCOc1ccc2CCC(NC(=O)OCC)C(Cc3cccc(Cl)c3)c2c1
CCCS(=O)(=O)N(C)CCOc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3cn(C)cn3)cc2C1Cc1cccc(Cl)c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3cnn(c3)C(F)F)cc2C1Cc1cccc(Cl)c1
CCCS(=O)(=O)OC[C@H]1CCCN1S(=O)(=O)CCC |r|
CCCS(=O)(=O)N1CC(C1)Oc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
CCS(=O)(=O)CCCOc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
NC1CCc2ccc(OCCNS(=O)(=O)C3CCCCC3)cc2C1Cc1ccc(Cl)c(Cl)c1
C[Si](C)(C)CCS(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(Cl)c(Cl)c3)c2c1
Cc1cc(CS(=O)(=O)NCCOc2ccc3CCC(N)C(Cc4ccc(Cl)c(Cl)c4)c3c2)no1
Clc1ccc(CC2C(CCc3ccc(OCCNS(=O)(=O)C4CCC4)cc23)N2CCCC2)cc1Cl
CN(CCOc1ccc2CCC(C(Cc3ccc(Cl)c(Cl)c3)c2c1)N1CCCC1)S(=O)(=O)c1cnn(C)c1
CCCCS(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(Cl)c(Cl)c3)c2c1
CC(C)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(Cl)c(Cl)c3)c2c1
CCOCCS(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(Cl)c(Cl)c3)c2c1
CN(CCOc1ccc2CCC(C(Cc3ccc(Cl)c(Cl)c3)c2c1)N1CCCC1)S(=O)(=O)C1CCC1
NC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccc(Cl)c(Cl)c1
CCCS(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(OC)cc3)c2c1
CN(CCOc1ccc2CCC(N)C(Cc3ccccc3)c2c1)S(=O)(=O)c1cn(C)cn1
NC1CCc2ccc(OCCNS(=O)(=O)c3ccccc3)cc2C1Cc1ccccc1
NC1CCc2ccc(OCCNS(=O)(=O)CCC(F)(F)F)cc2C1Cc1ccccc1
CN(CCOc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCCC1)S(=O)(=O)c1cn(C)cn1
NC1CCc2ccc(OCCNS(=O)(=O)C3CC3)cc2C1Cc1ccccc1
CCC(=O)NCCOc1ccc2CCC(N)C(Cc3ccccc3)c2c1
Cn1cnc(n1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(Cl)c(Cl)c3)c2c1
CN(CCOc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCC1)S(=O)(=O)c1cn(C)cn1
NC1CCc2ccc(OCCNS(=O)(=O)CC3CCC3)cc2C1Cc1ccc(Cl)c(Cl)c1
CCCS(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3cccc(F)c3)c2c1
CN(CCOc1ccc2CCC(N)C(Cc3ccc(Cl)c(Cl)c3)c2c1)S(=O)(=O)CC1CC1
CN(CCOc1ccc2CCC(N)C(Cc3ccccc3)c2c1)S(=O)(=O)c1cnn(C)c1
CCN(CCOc1ccc2CCC(N)C(Cc3ccc(Cl)c(Cl)c3)c2c1)S(=O)(=O)c1cnn(C)c1
CN(CCOc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCCC1)S(=O)(=O)c1cnn(C)c1
CN(CCOc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCC1)S(=O)(=O)c1cnn(C)c1
CCN(CCOc1ccc2CCC(N)C(Cc3ccccc3)c2c1)S(=O)(=O)c1cnn(C)c1
CCCCCS(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(Cl)c(Cl)c3)c2c1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCCC1
CCCS(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccc(F)c(Cl)c3)c2c1
NC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccccc1
NC1CCc2ccc(OCCNC(=O)CC3CC3)cc2C1Cc1ccc(Cl)c(Cl)c1
NC1CCc2ccc(OCCNC(=O)c3ccccc3)cc2C1Cc1ccc(Cl)c(Cl)c1
CCN(CCOc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCCC1)S(=O)(=O)c1cnn(C)c1
NC1CCc2ccc(OCCNS(=O)(=O)CCC3CC3)cc2C1Cc1ccc(Cl)c(Cl)c1
CN(CCOc1ccc2CCC(C(Cc3ccc(Cl)c(Cl)c3)c2c1)N1CCCC1)S(=O)(=O)CC1CC1
CN(CCOc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCCC1)S(=O)(=O)CC1CC1
NC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccc(Cl)cc1
CN(CCOc1ccc2CCC(N)C(Cc3ccc(Cl)cc3)c2c1)S(=O)(=O)CC1CC1
CN(CCOc1ccc2CCC(N)C(Cc3ccccc3)c2c1)S(=O)(=O)CC1CC1
NC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccc(F)c(F)c1
Clc1ccc(CC2C(CCc3ccc(OCCNS(=O)(=O)CC4CC4)cc23)N2CCCC2)cc1Cl
O=S(=O)(CC1CC1)NCCOc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCCC1
FC1CCN(C1)C1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccc(Cl)c(Cl)c1
Clc1ccc(CC2C(CCc3ccc(OCCNS(=O)(=O)CC4CC4)cc23)N2CCC2)cc1Cl
FC1CCN(C1)C1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccccc1
CNC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccccc1
Fc1cccc(CC2C(CCc3ccc(OCCNS(=O)(=O)CC4CC4)cc23)N2CCCC2)c1
Fc1cccc(CC2C(CCc3ccc(OCCNS(=O)(=O)CC4CC4)cc23)N2CCC2)c1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(C(Cc3cccc(F)c3)c2c1)N1CCC1
O=S(=O)(CC1CC1)NCCOc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCC1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCC1
O=S(=O)(NCCOc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCC1)C1CCC1
CCCS(=O)(=O)NCCOc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCC1
NC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1cc(F)cc(Cl)c1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3cc(F)cc(Cl)c3)c2c1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCC(F)C1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(C(Cc3cccc(c3)C#N)c2c1)N1CCCC1
CC(C)NC1CCc2ccc(OCCNS(=O)(=O)c3cn(C)cn3)cc2C1Cc1cccc(c1)C#N
O=S(=O)(CC1CC1)NCCOc1ccc2CCC(C(Cc3cccc(c3)C#N)c2c1)N1CCCC1
CC(C)NC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1cccc(c1)C#N
CCCS(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccccc3)c2c1
CNC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1cc(F)cc(Cl)c1
Fc1cc(Cl)cc(CC2C(CCc3ccc(OCCNS(=O)(=O)CC4CC4)cc23)N2CCC2)c1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(C(Cc3cc(F)cc(Cl)c3)c2c1)N1CCC1
CNC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccc(F)cc1
Cc1cccc(CC2C(CCc3ccc(OCCNS(=O)(=O)c4cn(C)cn4)cc23)N2CCCC2)c1
COc1cccc(CC2C(CCc3ccc(OCCNS(=O)(=O)c4cn(C)cn4)cc23)N2CCCC2)c1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3cccc(c3)C(F)(F)F)c2c1
CCCS(=O)(=O)NCc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
CS(=O)(=O)NCc1ccc2CCC(N)C(Cc3ccccc3)c2c1
NC1CCc2ccc(CNS(=O)(=O)c3ccccc3)cc2C1Cc1ccccc1
CCCS(=O)(=O)NCc1ccc2CCC(N)[C@@H](Cc3ccccc3)c2c1 |r|
CCCS(=O)(=O)NCc1ccc2CCC(N)[C@H](Cc3ccccc3)c2c1 |r|
CCCS(=O)(=O)NCc1ccc2CCC(N)C(Cc3cccc(F)c3)c2c1
Cn1cc(cn1)S(=O)(=O)NCc1ccc2CCC(N)C(Cc3ccccc3)c2c1
Cn1cnc(c1)S(=O)(=O)NCc1ccc2CCC(N)C(Cc3ccccc3)c2c1
NC1CCc2ccc(CNS(=O)(=O)C3CCC3)cc2C1Cc1ccc(F)cc1
CCCS(=O)(=O)NCc1ccc2CCC(N)C(Cc3ccc(F)cc3)c2c1
Cn1cnc(c1)S(=O)(=O)NCc1ccc2CCC(N)C(Cc3ccc(F)cc3)c2c1
Cn1cnc(c1)S(=O)(=O)NCc1ccc2CCC(N)C(Cc3cccc(F)c3)c2c1
Cn1cc(cn1)S(=O)(=O)NCc1ccc2CCC(N)C(Cc3cccc(F)c3)c2c1
Cc1cccc(c1)S(=O)(=O)NCc1ccc2CCC(N)C(Cc3ccccc3)c2c1
Cn1ccc(c1)S(=O)(=O)NCc1ccc2CCC(N)C(Cc3ccccc3)c2c1
NC1CCc2ccc(CNS(=O)(=O)c3cccnc3)cc2C1Cc1ccccc1
Cn1cc(c(n1)C(F)(F)F)S(=O)(=O)NCc1ccc2CCC(N)C(Cc3ccccc3)c2c1
Cn1ccc(n1)S(=O)(=O)NCc1ccc2CCC(N)C(Cc3ccccc3)c2c1
NC1CCc2ccc(CNS(=O)(=O)C3CCC3)cc2C1Cc1cccc(F)c1
NC1CCc2ccc(CNS(=O)(=O)CC3CC3)cc2C1Cc1ccc(F)c(F)c1
NC1CCc2ccc(CNS(=O)(=O)C3CCC3)cc2C1Cc1ccc(F)c(F)c1
CCCS(=O)(=O)NCc1ccc2CCC(NC)C(Cc3ccccc3)c2c1
CNC1CCc2ccc(CNS(=O)(=O)C3CCC3)cc2C1Cc1ccccc1
CNC1CCc2ccc(CNS(=O)(=O)c3cccc(C)c3)cc2C1Cc1ccccc1
CNC1CCc2ccc(CNS(=O)(=O)c3ccn(C)c3)cc2C1Cc1ccccc1
CNC1CCc2ccc(CNS(=O)(=O)c3ccn(C)n3)cc2C1Cc1ccccc1
CCCS(=O)(=O)NCc1ccc2CCC(NC(C)=O)C(Cc3ccccc3)c2c1
CC(=O)NC1CCc2ccc(CNS(=O)(=O)c3cn(C)cn3)cc2C1Cc1ccc(F)cc1
CCCS(=O)(=O)NCc1ccc2CCC(NCC)C(Cc3ccccc3)c2c1
CCNC1CCc2ccc(CNS(=O)(=O)c3cn(C)cn3)cc2C1Cc1ccc(F)cc1
CCNC1CCc2ccc(CNS(=O)(=O)c3cnn(C)c3)cc2C1Cc1cccc(F)c1
CCCS(=O)(=O)NCCCc1ccc2CCC(NC(=O)OC(C)(C)C)C(Cc3ccc(Cl)cc3)c2c1
NC1CCc2ccc(CCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccc(Cl)cc1
CCCS(=O)(=O)NCCCc1ccc2CCC(N)C(Cc3ccc(Cl)c(Cl)c3)c2c1
NC1CCc2ccc(CCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccc(F)c(F)c1
CCCS(=O)(=O)NCCCc1ccc2CCC(N)C(Cc3ccccc3)c2c1
CCCS(=O)(=O)NCCCc1ccc2CCC(N)C(Cc3ccc(F)c(F)c3)c2c1
NC1CCc2ccc(CCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccccc1
NC1CCc2ccc(CCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccc(F)cc1
CCCS(=O)(=O)NCCCc1ccc2CCC(N)C(Cc3cccc(F)c3)c2c1
NC1CCc2ccc(CCCNS(=O)(=O)CC3CC3)cc2C1Cc1cccc(F)c1
CCCS(=O)(=O)NCCCc1ccc2CCC(N)C(Cc3ccccc3Cl)c2c1
NC1CCc2ccc(CCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccccc1Cl
CCCS(=O)(=O)NCCCc1ccc2CCC(N)C(Cc3ccc(F)cc3)c2c1
CCCS(=O)(=O)NCCCc1ccc2CCC(NC(C)=O)C(Cc3cccc(F)c3)c2c1
CCCS(=O)(=O)NCCCc1ccc2CCC(NC(C)=O)C(Cc3ccc(F)cc3)c2c1
CC(=O)NC1CCc2ccc(CCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccccc1
CCCS(=O)(=O)NCCCc1ccc2CCC(NC(C)=O)C(Cc3ccccc3)c2c1
CC(=O)NC1CCc2ccc(CCCNS(=O)(=O)CC3CC3)cc2C1Cc1cccc(F)c1
CCCS(=O)(=O)NCCCc1ccc2CCC(NCC)C(Cc3cccc(F)c3)c2c1
CCCS(=O)(=O)NCCCc1ccc2CCC(NCC)C(Cc3ccc(F)cc3)c2c1
CCNC1CCc2ccc(CCCNS(=O)(=O)CC3CC3)cc2C1Cc1cccc(F)c1
CCCS(=O)(=O)NCCCc1ccc2CCC(NCC)C(Cc3ccccc3Cl)c2c1
CCCS(=O)(=O)NCCCc1ccc2CCC(NCC)C(Cc3ccccc3)c2c1
CCNC1CCc2ccc(CCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccccc1
CCCS(=O)(=O)NCCCc1ccc2CCC(NCC)C(Cc3ccc(F)c(F)c3)c2c1
CCNC1CCc2ccc(CCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccc(F)c(F)c1
CCCS(=O)(=O)N(C)CCCc1ccc2CCC(N)C(Cc3cccc(F)c3)c2c1
CN(CCCc1ccc2CCC(N)C(Cc3ccccc3Cl)c2c1)S(=O)(=O)CC1CC1
CCCS(=O)(=O)N(C)CCCc1ccc2CCC(N)C(Cc3ccccc3Cl)c2c1
CN(CCCc1ccc2CCC(N)C(Cc3cccc(F)c3)c2c1)S(=O)(=O)CC1CC1
CN(CCCc1ccc2CCC(N)C(Cc3ccc(F)cc3)c2c1)S(=O)(=O)CC1CC1
CCCS(=O)(=O)N(C)CCCc1ccc2CCC(N)C(Cc3ccc(F)cc3)c2c1
CN(CCCc1ccc2CCC(N)C(Cc3ccc(Cl)cc3)c2c1)S(=O)(=O)CC1CC1
CCCS(=O)(=O)N(C)CCCc1ccc2CCC(N)C(Cc3ccc(Cl)cc3)c2c1
NC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1cccc(F)c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3ccn(C)c3)cc2C1Cc1cc(F)cc(F)c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1cc(F)cc(F)c1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccccc3)c2c1
CNC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1cccc(F)c1
CNC1CCc2ccc(OCCNS(=O)(=O)c3ccn(C)c3)cc2C1Cc1cc(F)cc(F)c1
CNC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1cc(F)cc(F)c1
CCCS(=O)(=O)NCc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCC1
Cn1cc(cn1)S(=O)(=O)NCc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCC1
Cn1ccc(c1)S(=O)(=O)NCc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCC1
Cn1cnc(c1)S(=O)(=O)NCc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCC1
O=S(=O)(NCc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCC1)c1ccccn1
O=S(=O)(NCc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCC1)c1cccs1
Cn1cnc(c1)S(=O)(=O)NCc1ccc2CCC(C(Cc3cccc(F)c3)c2c1)N1CCC1
Cn1cnc(c1)S(=O)(=O)NCc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCOCC1
Cn1cc(cn1)S(=O)(=O)NCc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCOCC1
O=S(=O)(CC1CC1)NCc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCOCC1
CCCS(=O)(=O)NCc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCOCC1
O=S(=O)(NCc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCOCC1)C1CCC1
Cn1cnc(c1)S(=O)(=O)NCc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCCC1
Cn1cnc(c1)S(=O)(=O)NCc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCCC1=O
COc1ccc2CCC(C(Cc3cccc(Cl)c3)c2c1)N1CCCC1
CCCS(=O)(=O)NCCCc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCCC1
O=S(=O)(CC1CC1)NCCCc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCCC1
Oc1ccc2CCC(C(Cc3cccc(F)c3)c2c1)N1CCCC1
Cn1ccc(c1)S(=O)(=O)NCCOc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCC1
Cn1ccc(c1)S(=O)(=O)NCCOc1ccc2CCC(C(Cc3cccc(F)c3)c2c1)N1CCC1
CCC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3ccn(C)c3)cc2C1Cc1ccccc1
Cn1ccc(c1)S(=O)(=O)NCCOc1ccc2CCC(NC=O)C(Cc3cc(F)cc(F)c3)c2c1
CCCS(=O)(=O)NCCCc1ccc2CCC(NC(C)C)C(Cc3ccc(Cl)c(Cl)c3)c2c1
CCCS(=O)(=O)NCCCc1ccc2CCC(NC(C)C)C(Cc3ccccc3)c2c1
CCN(CC)C1CCc2ccc(CCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccc(Cl)cc1
CCCS(=O)(=O)N(C)Cc1ccc2CCC(NC)C(Cc3ccccc3)c2c1
CCCS(=O)(=O)NCC#Cc1ccc2CCC(NC(C)=O)C(Cc3ccccc3)c2c1
CCCS(=O)(=O)N(CCOc1ccc2CCC(NC(=O)OCC)C(Cc3cccc(Cl)c3)c2c1)C1CC1
CCCS(=O)(=O)N(CCOc1ccc2CCC(NC(=O)OCC)C(Cc3ccccc3)c2c1)C1CC1
CCCS(=O)(=O)N(CCOc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1)C1CC1
CCCS(=O)(=O)N(CCOc1ccc2CCC(N)C(Cc3ccccc3)c2c1)C1CC1
CCCS(=O)(=O)N1CC(C1)c1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
CCCS(=O)(=O)N1CC(C1)c1ccc2CCC(N)C(Cc3ccccc3)c2c1
CCCS(=O)(=O)N1CC(COc2ccc3CCC(NC(=O)OCC)C(Cc4cccc(Cl)c4)c3c2)C1
CCCS(=O)(=O)N1CC(COc2ccc3CCC(N)C(Cc4cccc(Cl)c4)c3c2)C1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1cccc(Cl)c1
NC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1cccc(Cl)c1
CCOC(=O)NC1CCc2ccc(OCC3CN(C3)S(=O)(=O)CC3CC3)cc2C1Cc1cccc(Cl)c1
CCOC(=O)NC1CCc2ccc(OCCN(C)S(=O)(=O)CC3CC3)cc2C1Cc1cccc(Cl)c1
CN(CCOc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1)S(=O)(=O)CC1CC1
CCCS(=O)(=O)N1CC(COc2ccc3CCC(N)C(Cc4ccccc4)c3c2)C1
CCCS(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccccc3Cl)c2c1
NC1CCc2ccc(OCCNS(=O)(=O)C3CC3)cc2C1Cc1ccccc1Cl
NC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccccc1Cl
NC1CCc2ccc(CCCNS(=O)(=O)CC3CC3)cc2C1Cc1cccc(Cl)c1
CCCS(=O)(=O)NCCCc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3cn(C)cn3)cc2C1Cc1ccccc1Cl
CCOC(=O)NC1CCc2ccc(OCCNS(=O)(=O)c3cnn(C)c3)cc2C1Cc1ccccc1Cl
CNC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1cccc(Cl)c1
Cn1cc(cn1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccccc3Cl)c2c1
CNC1CCc2ccc(OCCNS(=O)(=O)c3cnn(C)c3)cc2C1Cc1ccccc1Cl
CNC1CCc2ccc(OCCNS(=O)(=O)c3cn(C)cn3)cc2C1Cc1ccccc1Cl
CCCS(=O)(=O)NCCc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3ccccc3Cl)c2c1
CC(=O)NC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1cccc(Cl)c1
CCNC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1cccc(Cl)c1
CCCS(=O)(=O)NCCCc1ccc2CCC(NC)C(Cc3cccc(Cl)c3)c2c1
CCCS(=O)(=O)NCCc1ccc2CCC(NC)C(Cc3cccc(Cl)c3)c2c1
NC1CCc2ccc(CCNS(=O)(=O)CC3CC3)cc2C1Cc1cccc(Cl)c1
CCCS(=O)(=O)NCCOc1ccc2CCC(NC)C(Cc3ccccc3F)c2c1
CNC1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccccc1F
CNC1CCc2ccc(CCNS(=O)(=O)c3cn(C)cn3)cc2C1Cc1cccc(Cl)c1
CCCS(=O)(=O)NCCOc1ccc2CCC(NC)C(CC3CCCCC3)c2c1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(C(Cc3ccccc3Cl)c2c1)N1CCCC1
Cc1nc(cn1C)S(=O)(=O)NCCOc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
Clc1cccc(CC2C(CCc3ccc(OCCNS(=O)(=O)CC4CC4)cc23)N2CCCC2)c1
Cn1cc(cn1)S(=O)(=O)NCCOc1ccc2CCC(C(Cc3cccc(Cl)c3)c2c1)N1CCCC1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(C(Cc3cccc(Cl)c3)c2c1)N1CCCC1
Clc1cccc(CC2C(CCc3ccc(OCCNS(=O)(=O)CC4CC4)cc23)N2CCC2)c1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CCC(C(Cc3cccc(Cl)c3)c2c1)N1CCC1
Cn1cc(cn1)S(=O)(=O)NCCOc1ccc2CCC(C(Cc3cccc(Cl)c3)c2c1)N1CCC1
CCCS(=O)(=O)NCCOc1ccc2CCC(C(Cc3cccc(Cl)c3)c2c1)N1CCCC1
Cn1cc(cn1)S(=O)(=O)NCCOc1ccc2CCC(C(Cc3ccccc3)c2c1)N1CCC1
CCCS(=O)(=O)CCc1ccc2CCC(N)C(Cc3ccccc3)c2c1
CCCS(=O)(=O)CCc1ccc2CCC(N)C(Cc3cccc(Cl)c3)c2c1
Fc1cccc(C2CN(CCN2C(=O)C2CCS(=O)(=O)CC2)c2ncc(cn2)C(F)(F)F)c1F
Fc1cccc([C@@H]2CN(CCN2C(=O)C2CCS(=O)(=O)CC2)c2ncc(cn2)C(F)(F)F)c1F |r|
Fc1cccc([C@H]2CN(CCN2C(=O)C2CCS(=O)(=O)CC2)c2ncc(cn2)C(F)(F)F)c1F |r|
Fc1cccc(c1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C(F)(F)F
Fc1cccc(c1)[C@@H]1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C(F)(F)F |r|
Fc1cccc(c1)[C@H]1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C(F)(F)F |r|
Fc1ccccc1C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C(F)(F)F
Fc1ccccc1[C@@H]1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C(F)(F)F |r|
Fc1ccccc1[C@H]1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C(F)(F)F |r|
Fc1ccc(cc1F)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C(F)(F)F
Fc1ccc(cc1F)[C@@H]1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C(F)(F)F |r|
Fc1ccc(cc1F)[C@H]1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C(F)(F)F |r|
Fc1ccc(C2CN(CCN2C(=O)C2CCS(=O)(=O)CC2)c2ncc(cn2)C(F)(F)F)c(F)c1
Fc1ccc([C@@H]2CN(CCN2C(=O)C2CCS(=O)(=O)CC2)c2ncc(cn2)C(F)(F)F)c(F)c1 |r|
Fc1ccc([C@H]2CN(CCN2C(=O)C2CCS(=O)(=O)CC2)c2ncc(cn2)C(F)(F)F)c(F)c1 |r|
Fc1ccc(nc1)N1CCN(C(C1)c1cccc(F)c1)C(=O)C1CCS(=O)(=O)CC1
Fc1cccc(c1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(F)cn1
Fc1cccc(C2CN(CCN2C(=O)C2CCS(=O)(=O)CC2)c2cc(on2)C(F)(F)F)c1F
Fc1cccc(c1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncccn1
Fc1cccc(c1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ccccn1
Fc1cccc(C2CN(CCN2C(=O)C2CCS(=O)(=O)CC2)c2ccc(cn2)C(F)(F)F)c1F
Fc1cnc(nc1)N1CCN(C(C1)c1cccc(F)c1F)C(=O)C1CCS(=O)(=O)CC1
Fc1cccc(C2CN(CCN2C(=O)C2CCS(=O)(=O)CC2)c2ncccn2)c1F
Fc1cccc(C2CN(CCN2C(=O)C2CCS(=O)(=O)CC2)c2ccccn2)c1F
Fc1ccc(nc1)N1CCN(C(C1)c1cccc(F)c1F)C(=O)C1CCS(=O)(=O)CC1
Fc1cccc(C2CN(CCN2C(=O)C2CCS(=O)(=O)CC2)c2cnc(cn2)C(F)(F)F)c1F
Fc1ccc(nc1)N1CCN(C(C1)c1ccc(F)cc1F)C(=O)C1CCS(=O)(=O)CC1
Fc1ccc(C2CN(CCN2C(=O)C2CCS(=O)(=O)CC2)c2ccccn2)c(F)c1
Fc1ccc(nc1)N1CCN(C(C1)c1ccc(F)c(F)c1)C(=O)C1CCS(=O)(=O)CC1
Fc1ccc(cc1F)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ccccn1
Fc1ccc(C2CN(CCN2C(=O)C2CCS(=O)(=O)CC2)c2cc(on2)C(F)(F)F)c(F)c1
Fc1ccc(cc1F)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cc(on1)C(F)(F)F
Cc1cnc(s1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ccc(cn1)C(F)(F)F
Fc1ccc(C2CN(CCN2C(=O)C2CCS(=O)(=O)CC2)c2cnc(cn2)C(F)(F)F)c(F)c1
Fc1ccc(C2CN(CCN2C(=O)C2CCS(=O)(=O)CC2)c2ccc(cn2)C(F)(F)F)c(F)c1
Fc1ccc(C2CN(CCN2C(=O)C2CCS(=O)(=O)CC2)c2ncccn2)c(F)c1
Fc1cnc(nc1)N1CCN(C(C1)c1ccc(F)cc1F)C(=O)C1CCS(=O)(=O)CC1
Fc1ccc(cc1F)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cnc(cn1)C(F)(F)F
Fc1ccc(cc1F)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ccc(cn1)C(F)(F)F
Fc1ccc(cc1F)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncccn1
Fc1cnc(nc1)N1CCN(C(C1)c1ccc(F)c(F)c1)C(=O)C1CCS(=O)(=O)CC1
Fc1ccc(cc1)[C@@H]1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ccc(cn1)C(F)(F)F |r|
Fc1ccc(cc1)[C@H]1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ccc(cn1)C(F)(F)F |r|
Fc1ccc(cc1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ccccn1
Fc1ccc(cc1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ccc(F)cn1
Fc1ccc(nc1)N1CCN(C(C1)c1ccccc1F)C(=O)C1CCS(=O)(=O)CC1
Fc1ccccc1C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ccccn1
Fc1cnc(nc1)N1CCN(C(C1)c1ccccc1F)C(=O)C1CCS(=O)(=O)CC1
Fc1ccccc1C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncccn1
Fc1ccc(cc1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cc(on1)C(F)(F)F
Fc1ccc(cc1)[C@@H]1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cc(on1)C(F)(F)F |r|
Fc1ccc(cc1)[C@H]1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cc(on1)C(F)(F)F |r|
Fc1ccc(cc1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncccn1
Fc1ccc(cc1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(F)cn1
Cc1ccc(nc1)N1CCN(C(C1)c1ccc(F)cc1)C(=O)C1CCS(=O)(=O)CC1
Cc1ccc(cn1)N1CCN(C(C1)c1ccc(F)cc1)C(=O)C1CCS(=O)(=O)CC1
Fc1ccc(cc1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ccc(nc1)C1CC1
Fc1cccc(c1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ccc(nc1)C1CC1
Fc1ccc(cc1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cnc(cn1)C(F)(F)F
Fc1ccc(cc1)[C@@H]1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cnc(cn1)C(F)(F)F |r|
Fc1ccc(cc1)[C@H]1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cnc(cn1)C(F)(F)F |r|
Clc1ccc(s1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cnc(nc1)C1CC1
Cc1ccc(cn1)N1CCN(C(C1)c1cccc(F)c1)C(=O)C1CCS(=O)(=O)CC1
Cc1ccc(nc1)N1CCN(C(C1)c1cccc(F)c1)C(=O)C1CCS(=O)(=O)CC1
Fc1ccc(cc1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cnc(nc1)C1CC1
Cc1ccc(nc1)N1CCN(C(C1)c1ccccc1F)C(=O)C1CCS(=O)(=O)CC1
Cc1ccc(cn1)N1CCN(C(C1)c1ccccc1F)C(=O)C1CCS(=O)(=O)CC1
Fc1ccccc1C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cnc(nc1)C1CC1
Cc1cnc(s1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1nnc(s1)C(F)(F)F
Fc1cccc(c1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cnc(nc1)C1CC1
FC(F)c1nc(no1)N1CCN(C(C1)c1ccc(Cl)s1)C(=O)C1CCS(=O)(=O)CC1
Cc1cnc(s1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cnc(cn1)C(F)(F)F
Fc1ccc(cc1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C(F)(F)F
Fc1ccc(cc1)[C@@H]1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C(F)(F)F |r|
Fc1ccc(cc1)[C@H]1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C(F)(F)F |r|
Fc1ccccc1C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cc(on1)C(F)(F)F
Fc1ccc(s1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cc(on1)C(F)(F)F
O=C(C1CCS(=O)(=O)CC1)N1CCN(CC1c1ccc(s1)C1CC1)c1cnc(cn1)C1CC1
FC(F)(F)c1cc(no1)N1CCN(C(C1)c1ccc(Cl)s1)C(=O)C1CCS(=O)(=O)CC1
Fc1ccc(cc1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cnc(nc1)C(F)(F)F
Fc1ccccc1C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cnc(cn1)C1CC1
Fc1cccc(c1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C1CC1
FC(F)(F)c1ncc(cn1)N1CCN(C(C1)c1ccc(Cl)s1)C(=O)C1CCS(=O)(=O)CC1
Fc1ccc(s1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cnc(nc1)C(F)(F)F
Fc1cccc(c1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cnc(nc1)C(F)(F)F
Cc1cnc(cn1)N1CCN(C(C1)c1cccc(F)c1)C(=O)C1CCS(=O)(=O)CC1
Cc1cnc(cn1)N1CCN(C(C1)c1ccc(F)s1)C(=O)C1CCS(=O)(=O)CC1
Cc1cnc(cn1)N1CCN(C(C1)c1ccccc1F)C(=O)C1CCS(=O)(=O)CC1
Cc1cnc(cn1)N1CCN(C(C1)c1ccc(Cl)s1)C(=O)C1CCS(=O)(=O)CC1
Fc1ccc(s1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1nnc(o1)C(F)(F)F
Cc1cnc(cn1)N1CCN(C(C1)c1ccc(F)cc1)C(=O)C1CCS(=O)(=O)CC1
Cc1cnc(nc1)N1CCN(C(C1)c1ccc(Cl)s1)C(=O)C1CCS(=O)(=O)CC1
Clc1ccc(s1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C1CC1
Fc1ccccc1C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C1CC1
Fc1ccccc1C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cnc(nc1)C(F)(F)F
Fc1ccc(s1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cnc(cn1)C(F)(F)F
Fc1ccc(s1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C1CC1
Fc1ccc(s1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1nnc(s1)C(F)(F)F
Fc1ccc(s1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C(F)(F)F
Cc1cnc(nc1)N1CCN(C(C1)c1ccc(F)s1)C(=O)C1CCS(=O)(=O)CC1
Fc1ccc(cc1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C1CC1
FC(F)(F)c1cnc(nc1)N1CCN([C@@H](C1)c1ccc(Cl)s1)C(=O)C1CCS(=O)(=O)CC1 |r|
FC(F)(F)c1cnc(nc1)N1CCN([C@H](C1)c1ccc(Cl)s1)C(=O)C1CCS(=O)(=O)CC1 |r|
Cc1cnc(nc1)N1CCN(C(C1)c1cccc(F)c1)C(=O)C1CCS(=O)(=O)CC1
Cc1cnc(nc1)N1CCN(C(C1)c1ccccc1F)C(=O)C1CCS(=O)(=O)CC1
Fc1ccccc1C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1noc(n1)C(F)(F)F
FC(F)c1nc(no1)N1CCN(C(C1)c1ccccc1F)C(=O)C1CCS(=O)(=O)CC1
Cc1cnc(nc1)N1CCN(C(C1)c1ccc(F)cc1)C(=O)C1CCS(=O)(=O)CC1
Fc1ccccc1C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cnc(cn1)C(F)(F)F
Fc1cccc(c1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cnc(cn1)C(F)(F)F
FC(F)(F)c1cnc(cn1)N1CCN(C(C1)c1ccc(Cl)s1)C(=O)C1CCS(=O)(=O)CC1
Fc1ccccc1C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1nnc(o1)C(F)(F)F
Fc1ccc(cc1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1noc(n1)C(F)(F)F
FC(F)c1nc(no1)N1CCN(C(C1)c1ccc(F)cc1)C(=O)C1CCS(=O)(=O)CC1
Fc1ccccc1C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1nc(co1)C(F)(F)F
Fc1ccc(cc1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1nc(co1)C(F)(F)F
Fc1cccc(c1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1cc(on1)C(F)(F)F
Fc1ccccc1C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1nnc(s1)C(F)(F)F
FC(F)(F)c1cccc(c1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C(F)(F)F
Fc1ccc(cc1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1nnc(s1)C(F)(F)F
FC(F)(F)c1ccc(cc1)N1CCN(C(C1)c1ccccc1)C(=O)C1CCS(=O)(=O)CC1
Clc1ccc(cc1)N1CCN(C(C1)c1ccccc1)C(=O)C1CCS(=O)(=O)CC1
Clc1ccc(cc1)N1CCN(C(C1)c1cccs1)C(=O)C1CCS(=O)(=O)CC1
COc1ccc(cc1C(F)(F)F)N1CCN(C(C1)c1ccccc1)C(=O)C1CCS(=O)(=O)CC1
O=C(C1CCS(=O)(=O)CC1)N1CCN(CC1c1ccccc1)c1ccc2ccccc2c1
FC(F)(F)c1ccc(cc1)N1CCN(C(C1)c1cccs1)C(=O)C1CCS(=O)(=O)CC1
O=C(C1CCS(=O)(=O)CC1)N1CCN(CC1c1ccccc1)c1nc2ccccc2s1
Clc1cccc(c1)N1CCN(C(C1)c1cccs1)C(=O)C1CCS(=O)(=O)CC1
O=C(C1CCS(=O)(=O)CC1)N1CCN(CC1c1cccs1)c1ccccc1
FC(F)(F)c1cc(ccc1Cl)N1CCN(C(C1)c1ccccc1)C(=O)C1CCS(=O)(=O)CC1
COc1ccc(cc1C(F)(F)F)N1CCN(C(C1)c1cccs1)C(=O)C1CCS(=O)(=O)CC1
FC(F)(F)c1cccc(c1)N1CCN(C(C1)c1ccccc1)C(=O)C1CCS(=O)(=O)CC1
Cc1ccc2nc([nH]c2c1)N1CCN(C(C1)c1ccccc1)C(=O)C1CCS(=O)(=O)CC1
COc1cccc(c1)N1CCN(C(C1)c1ccccc1)C(=O)C1CCS(=O)(=O)CC1
Clc1cccc(c1)N1CCN(C(C1)c1ccccc1)C(=O)C1CCS(=O)(=O)CC1
O=C(C1CCS(=O)(=O)CC1)N1CCN(CC1c1cccs1)c1ccc2ccccc2c1
FC(F)(F)c1cccc(c1)N1CCN(C(C1)c1cccs1)C(=O)C1CCS(=O)(=O)CC1
COc1cccc(c1)N1CCN(C(C1)c1cccs1)C(=O)C1CCS(=O)(=O)CC1
Clc1cc2nc([nH]c2cc1Cl)N1CCN(C(C1)c1ccccc1)C(=O)C1CCS(=O)(=O)CC1
FC(F)(F)c1cccc2[nH]c(nc12)N1CCN(C(C1)c1ccccc1)C(=O)C1CCS(=O)(=O)CC1
O=C(C1CCS(=O)(=O)CC1)N1CCN(CC1c1cccs1)c1cccnc1
O=C(C1CCS(=O)(=O)CC1)N1CCN(CC1c1ccccc1)c1cnccn1
O=C(C1CCS(=O)(=O)CC1)N1CCN(CC1c1cccs1)c1cccc2ccccc12
Clc1cc(Cl)c2nc([nH]c2c1)N1CCN(C(C1)c1ccccc1)C(=O)C1CCS(=O)(=O)CC1
Cc1cc2[nH]c(nc2cc1Cl)N1CCN(C(C1)c1ccccc1)C(=O)C1CCS(=O)(=O)CC1
FC(F)(F)c1ccc2nc([nH]c2c1)N1CCN(C(C1)c1ccccc1)C(=O)C1CCS(=O)(=O)CC1
FC(F)(F)c1nnc(s1)N1CCN([C@@H](C1)c1ccc(Cl)s1)C(=O)C1CCS(=O)(=O)CC1 |r|
FC(F)(F)c1nnc(s1)N1CCN([C@H](C1)c1ccc(Cl)s1)C(=O)C1CCS(=O)(=O)CC1 |r|
FC(F)(F)c1cc(no1)N1CCN(C(C1)c1ccccc1)C(=O)C1CCS(=O)(=O)CC1
FC(F)(F)c1cnc(nc1)N1CCN(C(C1)c1ccc(s1)C1CC1)C(=O)C1CCS(=O)(=O)CC1
FC(F)(F)c1cc(no1)N1CCN(C(C1)c1ccc(s1)C(F)(F)F)C(=O)C1CCS(=O)(=O)CC1
FC(F)(F)c1coc(n1)N1CCN(C(C1)c1ccc(s1)C(F)(F)F)C(=O)C1CCS(=O)(=O)CC1
FC(F)(F)c1ccc(s1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1nnc(s1)C(F)(F)F
FC(F)(F)c1ccc(s1)[C@@H]1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1nnc(s1)C(F)(F)F |r|
FC(F)(F)c1ccc(s1)[C@H]1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1nnc(s1)C(F)(F)F |r|
Fc1cccc(c1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ccc(cn1)C(F)(F)F
Cc1ccc(s1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ccc(cn1)C(F)(F)F
Cc1ccc(s1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ncc(cn1)C(F)(F)F
Cc1ccc(s1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1nnc(s1)C(F)(F)F
Cc1ccc(s1)C1CN(CCN1C(=O)C1CCS(=O)(=O)CC1)c1ccc(nn1)C(F)(F)F
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc(F)c(c1)C(CN)Cc1ccccc1
Cn1cc(cn1)S(=O)(=O)NCCOc1cccc(c1)C(CN)Cc1cccc(Cl)c1
Cn1cc(cn1)S(=O)(=O)NCCOc1cc(ccc1F)C(CN)Cc1ccccc1
Cn1cnc(c1)S(=O)(=O)NCCOc1cc(ccc1F)C(CN)Cc1ccccc1
Cn1cnc(c1)S(=O)(=O)NCCOc1cccc(c1)C(CN)Cc1ccccc1
Cn1cc(cn1)S(=O)(=O)NCCOc1cccc(c1)C(CN)Cc1ccccc1
Cn1cc(cn1)S(=O)(=O)NCCOc1cccc(c1)C(CN)Cc1cc(F)cc(F)c1
Cn1cc(cn1)S(=O)(=O)NCCOc1cccc(c1)C(CN)Cc1ccc(Cl)cc1
Cn1cnc(c1)S(=O)(=O)NCCOc1cccc(c1)C(CN)Cc1cccc(Cl)c1
Cn1cc(cn1)S(=O)(=O)NCCOc1cccc(c1)C(CN)Cc1cccc(c1)C(F)(F)F
Cn1cnc(c1)S(=O)(=O)NCCOc1cccc(c1)C(CN)Cc1cc(F)cc(F)c1
Cn1cnc(c1)S(=O)(=O)NCCOc1cccc(c1)C(CN)Cc1cccc(c1)C(F)(F)F
NC(=O)C(Cc1ccccc1)c1cccc(CNS(=O)(=O)CC2CC2)c1
NCC(Cc1ccccc1)c1cccc(CNS(=O)(=O)CC2CC2)c1
Cn1cc(cn1)S(=O)(=O)NCc1cccc(c1)C(Cc1ccccc1)C(N)=O
Cn1cnc(c1)S(=O)(=O)NCc1cccc(c1)C(Cc1ccccc1)C(N)=O
Cn1cnc(c1)S(=O)(=O)NCc1cccc(c1)C(Cc1ccccc1)C(=O)N1CCOCC1
Cn1cc(cn1)S(=O)(=O)NCc1cccc(c1)C(CN)Cc1ccccc1
Cn1cnc(c1)S(=O)(=O)NCc1cccc(c1)C(CN)Cc1ccccc1
Cn1cnc(c1)S(=O)(=O)NCc1cccc(c1)C(CN1CCOCC1)Cc1ccccc1
Cn1cc(cn1)S(=O)(=O)NCc1cccc(c1)C(CN1CCOCC1)Cc1ccccc1
O=S(=O)(CC1CC1)NCc1cccc(c1)C(CN1CCOCC1)Cc1ccccc1
CN(C)CC(Cc1ccccc1)c1cc(OCCNS(=O)(=O)c2cn(C)cn2)ccc1F
CN(C)CC(Cc1ccccc1)c1cccc(OCCNS(=O)(=O)c2cnn(C)c2)c1
CN(C)CC(Cc1ccccc1)c1cccc(OCCNS(=O)(=O)c2cn(C)cn2)c1
CN(C)CC(Cc1ccccc1)c1cccc(CNS(=O)(=O)c2cn(C)cn2)c1
CN(C)CC(Cc1ccccc1)c1cccc(CNS(=O)(=O)c2cnn(C)c2)c1
CN(C)CC(Cc1cccc(c1)C(F)(F)F)c1cccc(OCCNS(=O)(=O)c2cnn(C)c2)c1
CN(C)CC(Cc1cccc(c1)C(F)(F)F)c1cccc(OCCNS(=O)(=O)c2cn(C)cn2)c1
CN(C)CC(Cc1ccccc1)c1cc(OCCNS(=O)(=O)c2cnn(C)c2)ccc1Cl
CN(C)CC(Cc1ccccc1)c1ccc(F)c(OCCNS(=O)(=O)c2cnn(C)c2)c1
CN(C)CC(Cc1ccccc1)c1ccc(F)c(OCCNS(=O)(=O)c2cn(C)cn2)c1
CN(C)CC(Cc1ccccc1)c1cc(OCCNS(=O)(=O)c2cnn(C)c2)ccc1F
Cn1cc(cn1)S(=O)(=O)NCCOc1cccc(c1)C(CN1CCCC1)Cc1ccccc1
Cn1cnc(c1)S(=O)(=O)NCCOc1cccc(c1)C(CN1CCCC1)Cc1ccccc1
Cn1cc(cn1)S(=O)(=O)NCCOc1cccc(c1)C(CN1CCC1)Cc1ccccc1
Cn1cc(cn1)S(=O)(=O)NCc1cccc(c1)C(CN1CCC1)Cc1ccccc1
CN(Cc1cccc(c1)C(CNC(=O)OC(C)(C)C)C1(CCC1)c1ccc(Cl)cc1)S(=O)(=O)c1cnn(C)c1
CCCS(=O)(=O)N(C)Cc1cccc(c1)C(CNC(=O)OC(C)(C)C)C1(CCC1)c1ccc(Cl)cc1
CN(Cc1cccc(c1)C(CNC(=O)OC(C)(C)C)C1(CCC1)c1ccc(Cl)cc1)S(=O)(=O)c1cn(C)cn1
CCCS(=O)(=O)N(C)Cc1cccc(c1)C(CN)C1(CCC1)c1ccc(Cl)cc1
CN(Cc1cccc(c1)C(CN)C1(CCC1)c1ccc(Cl)cc1)S(=O)(=O)CCCF
CN(Cc1cccc(c1)C(CN)C1(CCC1)c1ccc(Cl)cc1)S(=O)(=O)c1cn(C)cn1
CN(Cc1cccc(c1)C(CN)C1(CCC1)c1ccc(Cl)cc1)S(=O)(=O)c1cnn(C)c1
CCOC(=O)N1CC(Cc2ccccc2)(C1)c1cccc(OCCNS(=O)(=O)c2cnn(C)c2)c1
CCOC(=O)N1CC(Cc2ccccc2)(C1)c1cccc(OCCNS(=O)(=O)c2cn(C)cn2)c1
CCOC(=O)N1CC(Cc2ccccc2)(C1)c1cccc(OCCNS(=O)(=O)CC2CC2)c1
O=S(=O)(CC1CC1)NCCOc1cccc(c1)C1(Cc2ccccc2)CNC1
Cn1cc(cn1)S(=O)(=O)NCCOc1cccc(c1)C1(Cc2ccccc2)CNC1
Cn1cnc(c1)S(=O)(=O)NCCOc1cccc(c1)C1(Cc2ccccc2)CNC1
CN1CC(Cc2ccccc2)(C1)c1ccc(F)c(OCCNS(=O)(=O)c2cn(C)cn2)c1
CN(CCOc1cc(ccc1F)C1(Cc2ccccc2)CN(C)C1)S(=O)(=O)c1cn(C)cn1
Cn1cnc(c1)S(=O)(=O)NCCOc1cccc(c1)C1(Cc2ccccc2)CN(CC(F)(F)F)C1
Cn1cnc(c1)S(=O)(=O)NCCOc1cccc(c1)C1(Cc2ccccc2)CN(CC(F)F)C1
Cn1cnc(c1)S(=O)(=O)NCCOc1cccc(c1)C1(Cc2ccccc2)CNC(=O)C1
O=C1CC(Cc2ccccc2)(CN1)c1cccc(OCCNS(=O)(=O)CC2CC2)c1
Cn1cc(cn1)S(=O)(=O)NCCOc1cccc(c1)C1(Cc2ccccc2)CNC(=O)C1
O=S(=O)(CC1CC1)NCCOc1cccc(c1)C1(Cc2ccccc2)CCNC1
Cn1cc(cn1)S(=O)(=O)NCCOc1cccc(c1)C1(Cc2ccccc2)CCNC1
Cn1cnc(c1)S(=O)(=O)NCCOc1cccc(c1)C1(Cc2ccccc2)CCNC1
CN1CCCC(Cc2ccccc2)(C1)c1cccc(OCCNS(=O)(=O)c2cn(C)cn2)c1
CN1CCCC(Cc2ccccc2)(C1)c1cccc(OCCNS(=O)(=O)c2cnn(C)c2)c1
CN1CCCC(Cc2ccccc2)(C1)c1cccc(OCCNS(=O)(=O)CC2CC2)c1
Cn1cc(cn1)S(=O)(=O)NCc1cccc(c1)C1(Cc2ccccc2)CNC(=O)C1
Cn1cc(cn1)S(=O)(=O)NCc1cccc(c1)C1(Cc2ccccc2)CCNC1
O=S(=O)(CC1CC1)NCc1cccc(c1)C1(Cc2ccccc2)CCNC1
CN1CCC(Cc2ccccc2)(C1)c1cccc(CNS(=O)(=O)c2cnn(C)c2)c1
CN1CCC(Cc2ccccc2)(C1)c1cccc(OCCNS(=O)(=O)c2cn(C)cn2)c1
Cn1cnc(c1)S(=O)(=O)NCCOc1cccc(c1)C1(Cc2ccccc2)CCN(C1)C(=O)C(F)F
Cn1cnc(c1)S(=O)(=O)NCCOc1cccc(c1)C1(Cc2ccccc2)CN(CCF)C1
COCCN1CC(Cc2ccccc2)(C1)c1cccc(OCCNS(=O)(=O)c2cn(C)cn2)c1
CN(CCOc1cccc(c1)C1(Cc2ccccc2)CCN(C)C1)S(=O)(=O)c1cn(C)cn1
Cn1cnc(c1)S(=O)(=O)NCCOc1cccc(c1)C1(Cc2ccccc2)CCN(CCF)C1
Cn1cnc(c1)S(=O)(=O)NCCOc1cccc(c1)C1(Cc2ccccc2)CCN(CC(C)(C)C)C1
CC(C)N1CCC(Cc2ccccc2)(C1)c1cccc(OCCNS(=O)(=O)c2cn(C)cn2)c1
CN1CC(Cc2ccccc2)(C1)c1cccc(OCCNS(=O)(=O)c2cn(C)cn2)c1
OC(=O)CN1CCN(CC1)C(c1ccc(Cl)cc1)c1ccc(Cl)cc1
C[C@@H]1CN(CCN1CC(O)=O)[C@@H](c1ccccc1)c1cccc(Br)c1
C[C@@H]1CN(CCN1CC(O)=O)[C@H](c1ccccc1)c1cccc(c1)-c1ccccc1
CSc1cccc(c1)[C@H](N1CCN(CC(O)=O)[C@H](C)C1)c1ccccc1
C[C@@H]1CN(CCN1CC(O)=O)[C@H](c1ccccc1)c1ccc(cc1)-c1ccc(C)cc1
C[C@@H]1CN(CCN1CC(O)=O)C(C1CC1)c1cccc(c1)C(F)(F)F
C[C@@H]1CN(CCN1CC(O)=O)C(c1ccccc1)c1ccccc1
C[C@@H]1CN(CCN1CC(O)=O)[C@H](c1ccccc1)c1cccc(c1)C(F)(F)F
C[C@@H]1CN(CCN1CC(O)=O)[C@H](c1ccccc1)c1cccc(C)c1
C[C@@H]1CN(CCN1CC(O)=O)[C@H](c1ccccc1)c1ccc(cc1)-c1cccc(C)c1
C[C@@H]1CN(CCN1CC(O)=O)[C@H](c1ccccc1)c1ccc(cc1)C#Cc1ccccc1
C[C@@H]1CN(CCN1CC(O)=O)C(c1ccc(Cl)cc1)c1ccc(Cl)cc1
C[C@@H]1CN(CCN1CC(O)=O)[C@H](c1ccccc1)c1cccc(Br)c1
C[C@H](N1CCN(C(c2ccc(Cl)cc2)c2ccc(Cl)cc2)[C@H](C)C1)C(O)=O
C[C@@H]1CN(CCN1CC(O)=O)[C@H](c1ccccc1)c1cccc(c1)-c1cccs1
C[C@@H](N1CCN(C[C@H]1C)C(c1ccc(Cl)cc1)c1ccc(Cl)cc1)C(O)=O
C[C@@H]1CN(CCN1CC(O)=O)[C@@H](c1cccs1)c1cccc(c1)C(F)(F)F
CN(CC[C@H](c1ccc(cc1)F)Oc2ccc(cc2)c3ccccc3)CC(=O)O
CN(CCC(Oc1ccc(cc1)C(=O)c1ccc(C)cc1)c1ccccc1)CC(O)=O
CC(C)C1CCCN1C[C@@H](O)CNS(=O)(=O)c1cccc2ccccc12
CC(C)C1CCCCN1C[C@@H](O)CNS(=O)(=O)c1cccc2ccccc12
CC(C)CC1CCCN1C[C@@H](O)CNS(=O)(=O)c1cccc2ccccc12
CCC1CCCN1C[C@@H](O)CNS(=O)(=O)c1cccc2ccccc12
O[C@@H](CNS(=O)(=O)c1cccc2ccccc12)CN1CCCC1C1CCCCC1
CC(C)(C)C1CCCN1C[C@@H](O)CNS(=O)(=O)c1cccc2ccccc12
O[C@@H](CNS(=O)(=O)c1cccc2ccccc12)CN1CCCC1C1CC1
COc1cc(cc(SC)c1C(=O)N[C@]1(CCCN(C)C1)c1ccccc1)C(F)(F)F |r|
COc1cc(cc(SC)c1C(=O)NC1(CCCN(C)C1)c1ccccc1)C(F)(F)F
COc1cc(cc(SC)c1C(=O)NC1(CCCN(C)C1)c1cccc(Cl)c1)C(F)(F)F
COc1cc(cc(SC)c1C(=O)NC1(CCCN(C)C1)c1ccc(F)cc1)C(F)(F)F
COc1cc(cc(SC)c1C(=O)NC1(CCCN(C)C1)c1ccc(Cl)cc1)C(F)(F)F
COc1cc(cc(SC)c1C(=O)NC1(CCCN(C)C1)c1cccc(F)c1)C(F)(F)F
COc1cc(cc(SC)c1C(=O)NC1(CCCN(C)C1)c1cccnc1)C(F)(F)F
COc1cc(cc(SC)c1C(=O)NC1(CCCN(C)C1)c1ccncc1)C(F)(F)F
CSc1cc(ccc1C(=O)NC1(CCCN(C)C1)c1ccccc1)C(F)(F)F
COc1cccc(c1)C1(CCCN(C)C1)NC(=O)c1c(OC)cc(cc1SC)C(F)(F)F
COc1ccc(cc1)C1(CCCN(C)C1)NC(=O)c1c(OC)cc(cc1SC)C(F)(F)F
COc1cc(cc(SC)c1C(=O)N[C@@]1(CCCN(C)C1)c1ccccc1)C(F)(F)F |r|
COc1cc(cc(SC)c1C(=O)NC1(CCCN(C)C1)c1ccc(F)cn1)C(F)(F)F
CCN1CCCC(C1)(NC(=O)c1c(OC)cc(cc1C(F)(F)F)C(F)(F)F)c1ccccc1
COc1cc(cc(c1C(=O)NC1(CCCN(C1)C(C)C)c1ccccc1)C(F)(F)F)C(F)(F)F
COc1cc(cc(SC)c1C(=O)NC1(CCCN(C)C1)c1ccc(C)cc1)C(F)(F)F
COc1cc(cc(c1C(=O)NC1(CCCN(C1)C1CCCC1)c1ccccc1)C(F)(F)F)C(F)(F)F
CN1CCCC(C1)(NC(=O)c1ccc(cc1Br)C(F)(F)F)c1ccccc1
CN1CCCC(C1)(NC(=O)c1ccc(cc1C)C(F)(F)F)c1ccccc1
COc1cc(cc(c1C(=O)NC1(CCCN(CC2CC2)C1)c1ccccc1)C(F)(F)F)C(F)(F)F
CN1CCCC(C1)(NC(=O)c1ccc(cc1C(F)(F)F)C(F)(F)F)c1ccccc1
COc1cc(cc(c1C(=O)NC1(CCCNC1)c1ccccc1)C(F)(F)F)C(F)(F)F
CN1CCCC(C1)(NC(=O)c1ccc(Cl)cc1Cl)c1ccccc1
COc1cccc(c1C(=O)NC1(CCCN(C)C1)c1ccccc1)C(F)(F)F
COc1cc(cc(SC)c1C(=O)NC1(CCCN(C)C1)c1cnccn1)C(F)(F)F
COc1cc(cc(SC)c1C(=O)NC1(CCCN(C)C1)c1ccncn1)C(F)(F)F
COc1cc(ccc1C(=O)NC1(CCCN(C)C1)c1ccccc1)C(F)(F)F
COc1cc(cc(c1C(=O)NC1(CCCN(Cc2ccccc2)C1)c1ccccc1)C(F)(F)F)C(F)(F)F
CN1CCCC(C1)(NC(=O)c1ccc(cc1F)C(F)(F)F)c1ccccc1
COc1cc(cc(c1C(=O)NC1(CCCN(C)C1)c1ccccc1)C(F)(F)F)C(F)(F)F
COc1cc(cc(c1C(=O)NC1(CCCN(C1)C(C)=O)c1ccccc1)C(F)(F)F)C(F)(F)F
COc1cc(cc(c1C(=O)NC1(CCCN(C1)C(=O)c1ccccc1)c1ccccc1)C(F)(F)F)C(F)(F)F
COc1cc(cc(c1C(=O)NC1(CCCN(C1)S(C)(=O)=O)c1ccccc1)C(F)(F)F)C(F)(F)F
CN1CCCC(C1)(NC(=O)c1ccc(cc1)C(F)(F)F)c1ccccc1
CN1CCCC(C1)(NC(=O)c1ccc(cc1C#N)C(F)(F)F)c1ccccc1
COc1cc(cc(SC)c1C(=O)NC1(CCCN(C)C1)c1ncccn1)C(F)(F)F
CCCCOc1c(OC)cc(cc1OC)C(=O)NCC1(CCCC1)N(C)C
CN(C)C1(CCCC1)CNC(=O)c2cc(c(c(c2)OC)OCc3ccccc3)OC
COc1cc(cc(OC)c1OCc1ccccc1)C(=O)NCC1(CCCCC1)N(C)C
CCCCOc1c(OC)cc(cc1OC)C(=O)NCC1(CCCCC1)N(C)C
FC(F)(F)c1ccc(cc1)N1CNC(=O)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
CCCCCCN1CNC(=O)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
COc1ccc(cc1)N1CNC(=O)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
O=C1NCN(c2ccccc2)C11CCN(Cc2ccccc2)CC1
CCCN1CNC(=O)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
O=C1NCN(C2CCCCC2)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
Cc1ccc(cc1)[C@@H]1CCCC[C@@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1
O=C1NCN(CC2CCCCC2)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
COc1ccc(cc1)[C@@H]1CCCC[C@@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1
O=C1NCN(CCN2CCCCC2)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
Fc1ccc(cc1)N1CNC(=O)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
CCCCCN1CNC(=O)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
O=C1NCN(C2CCC2)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
O=C1NCN(CCC2CCCCC2)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
COCCN1CNC(=O)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
O=C1NCN(c2ccccc2)C11CCN(CCc2ccccc2)CC1
O=C1NCN(CCc2ccccc2)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
Fc1ccc(cc1)[C@@H]1CCCC[C@@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1
O=C1NCN(c2ccccc2)C11CCN(CC1)[C@@H]1CCCC[C@H]1c1ccccc1
Clc1ccc(cc1)[C@@H]1CCCC[C@@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1
O=C1NCN(C2CCCC2)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
CN1CNC(=O)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
O=C1NCN(c2ccccc2)C11CCN(CC1)[C@H]1CCC[C@H]1c1ccccc1
CCN1CNC(=O)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
O=C1NCN(c2ccccc2)C11CCN(CC1)[C@H]1CCCCC[C@H]1c1ccccc1
CC(C)(Cc1ccccc1)N1CCC2(CC1)N(CNC2=O)c1ccccc1
O=C1NCN(c2ccccc2)C11CCN(CC1)[C@@H]1CCCC[C@@H]1c1ccccc1
Clc1ccc(cc1)N1CNC(=O)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
CC(C)(CN1CCC2(CC1)N(CNC2=O)c1ccccc1)c1ccccc1
O=C1NCN(c2ccccc2)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
Cc1ccc(cc1)N1CNC(=O)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
FC(F)(F)c1cc(ccc1Cl)[C@@H]1CCCC[C@@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1
O=C1NCN(C2CC2)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
Cc1ccccc1[C@@H]1CCCC[C@@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1
O=C1NCN(c2ccccc2)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccn1
O=C1NCN(Cc2ccccc2)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
Clc1cccc(c1)[C@@H]1CCCC[C@@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1
Clc1ccc(cc1Cl)[C@@H]1CCCC[C@@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1
O[C@]1(CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1)C1CCCCC1
O[C@]1(CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1)c1ccccn1
COc1cccc(c1)[C@]1(O)CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1
O[C@]1(COCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1)c1ccccc1
O[C@@]1(Cc2ccccc2)CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1
Cc1ccccc1[C@]1(O)CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1
COc1ccc(cc1)N1CNC(=O)C11CCN(CC1)[C@@H]1CCCC[C@@]1(O)c1ccc(Cl)cc1
O[C@]1(CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccc(F)cc1)c1ccc(Cl)cc1
O[C@]1(CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1)c1ccc(F)cc1
O[C@]1(CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1)c1cccnc1
CCCN1CNC(=O)C11CCN(CC1)[C@@H]1CCCC[C@@]1(O)c1ccccc1
CC(C)[C@]1(O)CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1
Cc1ccc(cc1)[C@]1(O)CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1
COc1ccc(cc1)[C@]1(O)CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1
O[C@]1(CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1)c1ccccc1
O[C@]1(CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1)c1ccc(Cl)cc1
CC(C)(C)[C@]1(O)CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1
O[C@]1(CCOC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1)c1ccccc1
O[C@]1(CCCC[C@@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1)c1ccccc1
C[C@]1(O)CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1
O[C@]1(CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccc(F)cc1)c1ccc(F)cc1
O[C@]1(CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1)c1ccncc1
O[C@]1(CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1)c1ccc(Cl)c(Cl)c1
O[C@]1(CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccc(Cl)cc1)c1ccc(F)cc1
O[C@]1(CCCC[C@H]1N1CCC2(CC1)N(CNC2=O)c1ccccc1)c1cccc(Cl)c1
COc1cc2C(=O)C(CCN(C)CC(O)=O)(C(=O)c2c(Cl)c1Cl)c1ccccc1
CN(CCC1(C(=O)c2ccc(Cl)cc2C1=O)c1ccccc1)CC(O)=O
CN(CCC1(C(=O)c2cccc(F)c2C1=O)c1ccccc1)CC(O)=O
COc1cc2C(=O)C(CCN(C)[C@H](C(O)=O)c3ccccc3)(C(=O)c2c(Cl)c1Cl)c1ccc(F)cc1
COc1cc2C(=O)C(CCN(C)C(C)(C)C(O)=O)(C(=O)c2c(Cl)c1Cl)c1ccc(F)cc1
COc1cc2C(=O)C(CCN(C)[C@@H](CO)C(O)=O)(C(=O)c2c(Cl)c1Cl)c1ccccc1
COc1cc2C(=O)C(CCN(C)[C@@H](C)C(O)=O)(C(=O)c2c(Cl)c1Cl)c1ccccc1
COc1cc2C(=O)C(CCN(C)CC(O)=O)(C(=O)c2c(Cl)c1Cl)c1ccc(F)cc1
CN(CCCC1(C(=O)c2ccccc2C1=O)c1ccccc1)CC(O)=O
CN(CCC1(C(=O)c2cc(Cl)c(Cl)cc2C1=O)c1ccccc1)CC(O)=O
COc1cc2C(=O)C(CCN(C)[C@H](C)C(O)=O)(C(=O)c2c(Cl)c1Cl)c1ccccc1
CC[C@@H](C)N(C)CCC1(C(=O)c2cc(OC)c(Cl)c(Cl)c2C1=O)c1ccc(F)cc1
COc1cc2C(=O)C(CCN3CCC[C@H]3C(O)=O)(C(=O)c2c(Cl)c1Cl)c1ccccc1
CN(CCCCC1(C(=O)c2ccccc2C1=O)c1ccccc1)CC(O)=O
CN(CCC1(C(=O)c2ccccc2C1=O)c1ccccc1)CC(O)=O
OC(=O)[C@H]1CCCN1CCOc1ccccc1Sc1cccc(Cl)c1
CCN(CCOc1ccccc1Sc1cccc(Cl)c1)C(C)C(O)=O
C[C@@H](COc1ccccc1Sc1cccc(F)c1)N(C)CC(O)=O
COc1cccc(c1)-c1ccc(OCCN2CCC[C@H]2C(O)=O)c(Sc2cccc(F)c2)c1
COc1ccc(cc1)-c1ccc(OCCN2CCC[C@H]2C(O)=O)c(Sc2cccc(F)c2)c1
CCC(COc1ccccc1Sc1cccc(F)c1)N(C)CC(O)=O
CN(CCOc1ccccc1Sc1ccc(C)cc1)CC(O)=O
CN(CCOc1ccccc1Sc1ccc(F)cc1)CC(O)=O
CCN(CCOc1ccccc1Sc1cccc(Cl)c1)CC(O)=O
CC(N(C)CCOc1ccccc1Sc1cccc(Cl)c1)C(O)=O
CN(CCOc1ccccc1Sc1ccc(cc1)C(C)(C)C)CC(O)=O
CN(CCOc1ccccc1Sc1ccc(NC(C)=O)cc1)CC(O)=O
C[C@H](COc1ccccc1Sc1cccc(F)c1)N(C)CC(O)=O
OC(=O)[C@@H]1CCCN1CCOc1ccc(cc1Sc1cccc(F)c1)-c1ccccc1
CC(C)C(COc1ccccc1Sc1cccc(F)c1)N(C)CC(O)=O
OC(=O)[C@@H]1CCCN1CCOc1cc(ccc1Sc1cccc(F)c1)-c1ccccc1
OC(=O)[C@@H]1CCCN1CCOc1ccc(Cl)cc1Sc1cccc(F)c1
OC(=O)[C@@H]1CCCN1CCOc1cccc(Cl)c1Sc1cccc(F)c1
OC(=O)[C@@H]1CCCN1CCOc1ccccc1Sc1cccc(Cl)c1
CN(CCOc1ccccc1Sc1ccc(Cl)cc1)CC(O)=O
OC(=O)[C@@H]1CCCN1CCOc1c(Cl)cccc1Sc1cccc(F)c1
CN(CCOc1ccccc1Sc1cccc(F)c1)CC(O)=O
OC(=O)[C@@H]1CCCN1CCOc1cc(Cl)ccc1Sc1cccc(F)c1
OC(=O)[C@@H]1CCCN1CCOc1ccc(cc1Sc1cccc(F)c1)-c1ccsc1
CN(CCOc1ccccc1Sc1cccc(Cl)c1)CC(O)=O
COc1ccc(Sc2ccccc2OCCN(C)CC(O)=O)cc1
OC(=O)[C@@H]1CCCN1CCOc1ccc(cc1Sc1cccc(F)c1)-c1ccc(Cl)cc1
CN(CCOc1ccccc1Sc1ccccc1)CC(O)=O
CC(C)(C)c1ccc(cc1)C1(O)CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccc(F)cc1
OC1(CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccccc1)c1cccc(F)c1
COc1cccc(c1)C1(O)CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccccc1
Cc1ccccc1C1(O)CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccc(F)cc1
OC1(CCCCC1N1CCC2(CC1)N(CNC2=O)c1ccccc1)c1ccc(F)cc1
OC1(CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccc(F)cc1)c1ccc(cc1)C#N
OC1(CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccc(F)cc1)c1ccccc1OC(F)(F)F
COc1ccc(cc1)C1(O)CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccc(F)cc1
OC1(CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccccc1)c1ccc(F)cc1
CS(=O)(=O)c1ccc(cc1)C1(O)CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccc(F)cc1
OC1(CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccc(F)cc1)c1ccccc1F
OC1(CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccc(F)cc1)c1cccc(F)c1
Cc1ccc(cc1)C1(O)CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccc(F)cc1
O=C1NC[C@@H](c2ccccc2)C11CCN(CC1)[C@@H]1CCCC[C@@H]1c1ccccc1
OC1(CCCCC1N1CCC2(CC1)N(CNC2=O)c1ccccc1)c1ccccc1
OC1(CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccc(F)cc1)c1cccc(Cl)c1
COc1cccc(c1)C1(O)CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccc(F)cc1
O=C1NCN(c2ccccc2)C11CCN(CC1)C1CCCCC1c1ccccc1
CC1CC2(CCN1C1CCCCC1(O)c1cccc(F)c1)C(CNC2=O)c1ccc(F)cc1
Cc1cccc(c1)C1(O)CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccc(F)cc1
COc1ccc(cc1)C1(O)CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccccc1
OC1(CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccc(F)cc1)c1ccc(cc1)C(F)(F)F
Fc1ccc(cc1)[C@H]1CNC(=O)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccc(F)cc1
Fc1ccc(cc1)[C@H]1CNC(=O)C11CCN(CC1)[C@@H]1CCCC[C@@H]1c1ccc(F)cc1
Fc1ccc(cc1)C1CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccccc1
COc1ccc(cc1)C1CNC(=O)C11CCN(CC1)C1CCCCC1c1ccc(C)cc1
Fc1ccc(cc1)[C@@H]1CNC(=O)C11CCN(CC1)[C@@H]1CCCC[C@@H]1c1ccc(F)cc1
O=C1NC[C@H](c2ccccc2)C11CCN(CC1)[C@@H]1CCCC[C@@H]1c1ccccc1
COc1ccc(cc1)C1CNC(=O)C11CCN(CC1)C1CCCCC1c1ccc(F)cc1
O=C1NC[C@H](c2ccccc2)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
Fc1ccc(cc1)[C@@H]1CNC(=O)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccc(F)cc1
O=C1NCC(c2ccccc2)C11CCN(CC1)C1CCCCC1c1ccccc1
O=C1NC[C@@H](c2ccccc2)C11CCN(CC1)[C@H]1CCCC[C@H]1c1ccccc1
Fc1ccc(cc1)C1CNC(=O)C11CCN(CC1)C1CCCCC1c1ccc(cc1)C(F)(F)F
Fc1ccc(cc1)C1CCCCC1N1CCC2(CC1)C(CNC2=O)c1ccc(Cl)c(Cl)c1
CCN(Cc1cccc(OCc2noc(n2)-c2ccccc2F)c1)C1CCN(C1)C1CC(C)C(C)C1 |w:24.26,29.32,31.35,33.37|
OCC1(CCCC1)N1CCN(CC1)C1CCc2ccc(OCc3noc(n3)-c3ccc(Cl)cc3)cc12 |w:13.14|
OCC1CCCN(CCCC2CCCc3ccc(OCc4ccc(cn4)-c4ccccc4F)cc23)C1 |w:2.1,10.9|
CC1CC(CC1C)N1CCN(CC1)C1CCc2ccc(OCc3noc(n3)-c3ccc(Cl)cc3)cc12 |w:13.14,3.7,1.0,5.6|
OCC1CCCN(CCCC2CCCc3ccc(OCc4noc(n4)-c4ccccc4F)cc23)C1 |w:10.9,2.1|
CC(C)N1CCN(CC1)C1CCc2ccc(OCc3noc(n3)-c3ccc(Cl)cc3)cc12 |w:9.9|
OCC1CCCN(CCCC2CCCc3ccc(OCc4noc(n4)-c4ccc(Cl)cc4)cc23)C1 |w:10.9,2.1|
CN1CCN(CC1)c1cccc2ccc(OCc3noc(n3)-c3ccc(Cl)cc3)cc12
OCC1(CCCC1)NCCCC1CCc2ccc(OCc3noc(n3)-c3ccc(Cl)cc3)cc12 |w:11.11|
OCC1(CCCC1)N1CCN(CC1)C1CCc2ccc(OCc3noc(n3)-c3ccccc3F)cc12 |w:13.14|
Fc1ccccc1-c1nc(COc2ccc3CCC(N4CCN(CC4)C4CCCC4)c3c2)no1 |w:18.19|
CN(CCOc1ccc(cc1-c1ccc(Cl)cc1)-c1ccccc1)CC(O)=O
CN(CCOc1ccc(cc1-c1ccccc1F)-c1ccccc1)CC(O)=O
CN(CCOc1ccc(cc1-c1cccs1)-c1ccc2OCCc2c1)CC(O)=O
CN(CCOc1ccc(cc1-c1ccccc1Cl)-c1ccc2OCCc2c1)CC(O)=O
CN(CCOc1ccc(cc1C(=O)c1cccs1)-c1ccccc1Cl)CC(O)=O
COc1ccccc1-c1cc(ccc1OCCN(C)CC(O)=O)-c1ccccc1
CN(CCOc1ccc(cc1C(=O)c1cccs1)-c1ccccc1)CC(O)=O
CN(CCOc1ccc(cc1-c1ccccc1C)-c1ccccc1)CC(O)=O
CN(CCOc1ccc(cc1-c1ccccc1Cl)-c1ccc2OCOc2c1)CC(O)=O
CN(CCOc1ccc(cc1-c1cccs1)-c1ccccc1)CC(O)=O
CN(CCOc1ccc(cc1-c1cccs1)-c1ccc2OCCOc2c1)CC(O)=O
CN(CCOc1ccc(cc1C(=O)c1ccccc1)-c1ccccc1)CC(O)=O
CN(CCOc1ccc(cc1Cc1ccccc1)-c1ccccc1)CC(O)=O
COc1ccc(cc1C)-c1ccc(OCCN(C)CC(O)=O)c(c1)-c1ccccc1Cl
CN(CCOc1ccc(cc1-c1cccs1)-c1ccc2OCOc2c1)CC(O)=O
CN(CCOc1ccc(cc1-c1ccccc1Cl)-c1ccccc1)CC(O)=O
CN(CCOc1ccc(cc1-c1cccc(Cl)c1)-c1ccccc1)CC(O)=O
CN(CCOc1ccc(cc1-c1ccccc1)-c1ccccc1)CC(O)=O
CN(CCOc1ccc(cc1-c1ccccc1Cl)-c1ccc2OCCOc2c1)CC(O)=O
CN(CCOc1ccc(cc1C(=O)C1CCCCC1)-c1ccccc1)CC(O)=O
CN(CCOc1ccc(cc1CC1CCCCC1)-c1ccccc1)CC(O)=O
CN(CCOc1ccc(cc1C1CCCCC1)-c1ccccc1)CC(O)=O
CN(CCOc1ccc(cc1-c1cccc2ccccc12)-c1ccccc1)CC(O)=O
COc1ccc(cc1OC)-c1ccc(OCCN(C)CC(O)=O)c(c1)C(=O)c1cccs1
CN(CCOc1ccc(cc1Cc1cccs1)-c1ccccc1)CC(O)=O
CN(CCOc1ccc(cc1C(=O)c1cccs1)-c1ccc2OCOc2c1)CC(O)=O
COc1ccc(cc1C)-c1ccc(OCCN(C)CC(O)=O)c(c1)-c1cccs1
CN(CCOc1ccc(cc1C(=O)c1cccs1)C(F)(F)F)CC(O)=O
CN(CCOc1ccc(cc1C(=O)c1cccs1)-c1cccc(Cl)c1)CC(O)=O
CN(CCOc1ccc(cc1-c1ccsc1)-c1ccccc1)CC(O)=O
CN(CCOc1ccc(cc1C(=O)c1cccs1)-c1ccc(C)c(C)c1)CC(O)=O
CN(CCOc1ccc(cc1-c1nccs1)-c1ccccc1)CC(O)=O
CN(CCOc1ccc(cc1C(=O)c1cccs1)-c1ccc(C)cc1)CC(O)=O
COc1cccc(c1)-c1ccc(OCCN(C)CC(O)=O)c(c1)C(=O)c1cccs1
COc1ccc(cc1)-c1ccc(OCCN(C)CC(O)=O)c(c1)C(=O)c1cccs1
COc1ccc(cc1C)-c1ccc(OCCN(C)CC(O)=O)c(c1)C(=O)c1cccs1
CN(CCOc1ccc(cc1C(=O)c1cccs1)-c1ccc(Cl)cc1)CC(O)=O
CN(CCOc1ccc(cc1C(=O)c1cccs1)-c1ccccc1C)CC(O)=O
CN(CCOc1ccc(cc1C(=O)c1cccs1)-c1cccc(C)c1)CC(O)=O
CC(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(ccc2NC2CCCCC2)[N+]([O-])=O)c(F)c1
CC(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(ccc2NCC2CCCCC2)[N+]([O-])=O)c(F)c1
CC(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(ccc2N2CCCCC2)[N+]([O-])=O)c(F)c1
CC(=O)c1ccc(N2CCN(CC2)C(=O)c2cccc(c2)[N+]([O-])=O)c(F)c1
CC(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(ccc2N2CCOCC2)S(=O)(=O)Cc2ccccc2)c(F)c1
[O-][N+](=O)c1ccc(N2CCOCC2)c(c1)C(=O)N1CCN(CC1)c1ncc(cc1Cl)C(F)(F)F
CS(=O)(=O)c1ccc(N2CCCCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1)C(F)(F)F
CS(=O)(=O)c1ccc(N2CCOCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1)C(F)(F)F
CC(C)Oc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1)C(F)(F)F)S(C)(=O)=O
CC(C)Oc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1F)C(C)=O)S(C)(=O)=O
CCC(C)Oc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1F)C(C)=O)S(C)(=O)=O
CC(C)Sc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1F)C(C)=O)S(C)(=O)=O
CC(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(ccc2OCC2CC2)S(C)(=O)=O)c(F)c1
[O-][N+](=O)c1ccc(N2CCOCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1F)C(F)(F)F
CC(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(Br)ccc2N2CCOCC2)c(F)c1
CC(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(ccc2-c2ccccc2)S(C)(=O)=O)c(F)c1
CC(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(C)ccc2N2CCOCC2)c(F)c1
[O-][N+](=O)c1ccc(N2CCOCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1C#N)C(F)(F)F
CS(=O)(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(ccc2-c2ccccc2)S(C)(=O)=O)c(F)c1
[O-][N+](=O)c1ccc(N2CCOCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(c(Cl)n1)C(F)(F)F
CS(=O)(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(ccc2OCC2CC2)S(C)(=O)=O)c(F)c1
[O-][N+](=O)c1ccc(N2CCOCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(c(F)c1)C(F)(F)F
CC(=O)c1ccc(N2CCN(CC2)C(=O)c2ccccc2N2CCOCC2)c(F)c1
CC(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(N)ccc2N2CCOCC2)c(F)c1
CCCS(=O)(=O)c1ccc(N2CCOCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1F)C(C)=O
CC(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(ccc2N2CCOCC2)S(N)(=O)=O)c(F)c1
[O-][N+](=O)c1ccc(N2CCOCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1)C#N
[O-][N+](=O)c1ccc(N2CCOCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1F)C#N
CS(=O)(=O)c1ccc(cc1)N1CCN(CC1)C(=O)c1cc(ccc1N1CCOCC1)[N+]([O-])=O
CC(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(ccc2N2CCOCC2)C(F)(F)F)c(F)c1
CS(=O)(=O)c1ccc(N2CCCCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1F)C#N
CS(=O)(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(ccc2N2CCOCC2)[N+]([O-])=O)c(F)c1
CC(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(ccc2N2CCOCC2)S(C)(=O)=O)c(F)c1
CS(=O)(=O)c1ccc(-c2ccccc2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1F)C#N
CC(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(ccc2N2CCOCC2)C#N)c(F)c1
CS(=O)(=O)c1ccc(OCC2CC2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1F)C#N
CS(=O)(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(ccc2N2CCCCC2)S(C)(=O)=O)c(F)c1
CNS(=O)(=O)c1ccc(N2CCOCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1F)C(C)=O
Cc1ccccc1N1CCN(CC1)C(=O)c1cc(ccc1N1CCOCC1)[N+]([O-])=O
COc1ccccc1N1CCN(CC1)C(=O)c1cc(ccc1N1CCOCC1)[N+]([O-])=O
[O-][N+](=O)c1ccc(N2CCOCC2)c(c1)C(=O)N1CCN(CC1)c1ccccc1Cl
CNc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1F)C(C)=O)[N+]([O-])=O
Cc1ccc(cc1)N1CCN(CC1)C(=O)c1cc(ccc1N1CCOCC1)[N+]([O-])=O
CS(=O)(=O)c1ccc(-c2ccccc2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1)C(F)(F)F
COc1ccc(cc1)N1CCN(CC1)C(=O)c1cc(ccc1N1CCOCC1)[N+]([O-])=O
CC(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(ccc2N)[N+]([O-])=O)c(F)c1
CS(=O)(=O)c1ccc(OCC2CC2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1)C(F)(F)F
[O-][N+](=O)c1ccc(N2CCOCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1)C(F)(F)F
CC(C)Nc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1F)C(C)=O)[N+]([O-])=O
CS(=O)(=O)c1ccc(C2CCCCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1)C(F)(F)F
[O-][N+](=O)c1ccc(N2CCOCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(Cl)cc1
CN(C)c1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1F)C(C)=O)[N+]([O-])=O
CS(=O)(=O)c1ccc(-c2ccc(F)cc2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1)C(F)(F)F
[O-][N+](=O)c1ccc(N2CCOCC2)c(c1)C(=O)N1CCN(CC1)c1ccccc1C(F)(F)F
Cc1cccc(c1)N1CCN(CC1)C(=O)c1cc(ccc1N1CCOCC1)[N+]([O-])=O
COc1cccc(c1)N1CCN(CC1)C(=O)c1cc(ccc1N1CCOCC1)[N+]([O-])=O
[O-][N+](=O)c1ccc(N2CCOCC2)c(c1)C(=O)N1CCN(CC1)c1cccc(c1)C(F)(F)F
[O-][N+](=O)c1ccc(N2CCOCC2)c(c1)C(=O)N1CCN(CC1)c1cccc(Cl)c1
CC(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(ccc2N2CCOCC2)[N+]([O-])=O)c(F)c1
CC(=O)c1ccc(N2CCN(CC2)C(=O)c2cc(ccc2-c2cccc(F)c2)S(C)(=O)=O)c(F)c1
CN1c2ccccc2C(CNC(=O)CNC(=O)c2ccc(F)cc2)c2ccccc2C1=O
COc1ccc(CCC(=O)NCC(=O)N2CC(=O)N(C)c3ccc(Cl)cc3C2c2ccccc2)cc1
CC(=O)NCC(=O)NC(c1ccccc1)c1ccc(Cl)cc1
Fc1ccc(cc1)C(=O)NCC(=O)NC(c1ccccc1)c1ccccc1
Fc1ccc(cc1)C(=O)NCC(=O)NC(c1ccccc1)c1ncccn1
Clc1ccc(cc1)C(NC(=O)CNC(=O)CCc1ccccc1)c1ccccc1
Fc1ccc(cc1)C(=O)NCC(=O)NC(c1cccc(F)c1)c1cccc(F)c1
Fc1ccc(cc1)C(=O)NCC(=O)NC(c1ccccc1)c1cccc(c1)C(F)(F)F
COc1ccc(cc1)C(NC(=O)CNC(=O)c1ccc(F)cc1)c1ccccc1
Fc1ccc(cc1)C(=O)NCC(=O)NCC1c2ccccc2Sc2ccc(Cl)cc12
Fc1ccc(cc1)C(=O)NCC(=O)NCC1c2ccccc2CCc2ccccc12
Fc1ccc(cc1)C(=O)NCC(=O)NCC1c2ccccc2COc2ccc(F)cc12
Clc1ccc(cc1)C(NC(=O)CNC(=O)c1ccncc1)c1ccccc1
Clc1ccc(cc1)C(NC(=O)CNC(=O)c1ccsc1)c1ccccc1
Clc1ccc(cc1)C(NC(=O)CNC(=O)C1CCCC1)c1ccccc1
Fc1ccc(cc1)C(=O)NCC(=O)NC(c1ccccc1)c1cccc(Cl)c1
Clc1ccc(cc1)C(NC(=O)CNC(=O)Cc1ccccc1)c1ccccc1
Fc1ccc(cc1)C(=O)NCC(=O)NC(c1nccs1)c1ccccc1
Clc1ccc(cc1)C(NC(=O)CNC(=O)c1ccccc1)c1ccccc1
Clc1ccc(cc1)C(NC(=O)CNC(=O)c1ccc(Cl)cc1)c1ccccc1
Fc1ccc(cc1)C(=O)NCC(=O)NC(c1ccccc1)c1ccc(Cl)cc1
Clc1ccc(cc1)C(NC(=O)CNC(=O)c1ccc(cc1)C#N)c1ccccc1
COc1ccc(cc1)C(NC(=O)CNC(=O)c1ccc(F)cc1)c1ccc(OC)cc1
CCC(NC(=O)CNC(=O)c1ccc(F)cc1)c1ccccc1
Fc1ccc(cc1)C(=O)NCC(=O)NC(c1ccccc1)c1ccncc1
Fc1ccc(cc1)C(=O)NCC(=O)NC(c1ccccc1)c1cccnn1
Cc1ccccc1C(NC(=O)CNC(=O)c1ccc(F)cc1)c1ccccc1
Cc1cccc(c1)C(NC(=O)CNC(=O)c1ccc(F)cc1)c1ccccc1
Cc1ccc(cc1)C(NC(=O)CNC(=O)c1ccc(F)cc1)c1ccccc1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1ccccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2cccc(Cl)c2)(CC1)c1ccccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2c(Cl)cccc2Cl)(CC1)c1ccccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2c(N)cccc2Cl)(CC1)c1ccccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)c(Cl)c2)(CC1)c1ccccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2c(F)ccc(F)c2Cl)(CC1)c1ccccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2)(CC1)c1cc(C)ccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2)(CC1)c1ccccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2F)(CC1)c1ccccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2C)(CC1)c1ccccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2Cl)(CC1)c1ccccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2)(CC1)c1ccccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2OC)(CC1)c1ccccc1
CCCS(=O)(=O)N1CCC(CC1)([C@H](C)NC(=O)c1ccccc1OC(F)(F)F)c1ccccn1 |r|
CCCS(=O)(=O)N1CCC(CC1)([C@H](C)NC(=O)c1c(N)cccc1Cl)c1ccccc1 |r|
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2Cl)(CC1)c1cccc(C)n1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1cccc(OC)n1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2)(CC1)c1cccc(n1)N1CCOCC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2Cl)(CC1)c1cccc(n1)N1CCOCC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1ccncc1
CCCS(=O)(=O)N1CCC(CC1)([C@@H](C)NC(=O)c1ccccc1OC(F)(F)F)c1ccccn1 |r|
CCCS(=O)(=O)N1CCC(CC1)([C@@H](C)NC(=O)c1ccc(Cl)cc1Cl)c1ccccn1 |r|
CCCS(=O)(=O)N1CCC(CC1)([C@@H](C)NC(=O)c1cc(F)cc(F)c1Cl)c1ccccn1 |r|
CCCS(=O)(=O)N1CCC(CC1)([C@H](C)NC(=O)c1ccc(Cl)cc1Cl)c1ccccn1 |r|
CCCS(=O)(=O)N1CCC(CC1)([C@H](C)NC(=O)c1cc(F)cc(F)c1Cl)c1ccccn1 |r|
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1cccnc1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1cccc(n1)N1CCOCC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2C)(CC1)C1CCCCN1C
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2Cl)(CC1)c1cc(C)ccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2OC(F)(F)F)(CC1)C1CCCCN1C
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1cc(C)ccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2Cl)(CC1)C1CCCCN1C
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2)(CC1)c1cccc(C)n1
CCCS(=O)(=O)N1CCC(CNC(=O)c2cccc(C)c2)(CC1)c1ccccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2C(F)(F)F)(CC1)c1ccccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2)(CC1)C1CCCCN1C
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2OC(F)(F)F)(CC1)c1ccccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2Cl)(CC1)c1cccc(OC)n1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)C1CCCCN1C
CCCS(=O)(=O)N1CCC(CNC(=O)c2cc(F)cc(F)c2Cl)(CC1)C1CCCCN1C
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1cccc(C)n1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2)(CC1)c1cccc(OC)n1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)N1CCC1
CCCS(=O)(=O)N1CCC(CCOC)(CNC(=O)c2ccc(Cl)cc2Cl)CC1
CC(O)CS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1ccccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC2CCCCO2)CC1
CCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1ccccn1
CS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1ccccn1
CC(F)CS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1ccccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)C1CCCCC1O
CCCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1ccccn1
FC(F)(F)CS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1ccccn1
FC(F)(F)S(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1ccccn1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)C1CCCCC1OC(C)=O
CN(C)S(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1ccccn1
CC(C)S(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1ccccn1
Clc1ccc(C(=O)NCC2(CCN(CC2)S(=O)(=O)C2CC2)c2ccccn2)c(Cl)c1
Fc1cccnc1C1(CNC(=O)c2ccc(Cl)cc2Cl)CCN(CC1)S(=O)(=O)c1cccs1
Cn1cnc(c1)S(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1ncccc1F
Cn1cc(cn1)S(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1ncccc1F
Cn1ncc(n1)S(=O)(=O)N1CC(CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)C1
CCn1cc(nn1)S(=O)(=O)N1CC(CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)C1
Cn1cc(nn1)S(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1ncccc1F
Cn1cc(nn1)S(=O)(=O)N1CC(CNC(=O)c2ccc(Cl)cc2Cl)(C1)c1ncccc1F
Fc1cccnc1C1(CNC(=O)c2ccc(Cl)cc2Cl)CCN(CC1)S(=O)(=O)c1cccnc1
Clc1ccc(C(=O)NCC2(CC3CC3)CN(C2)S(=O)(=O)c2cnn[nH]2)c(Cl)c1
Cn1nncc1S(=O)(=O)N1CC(CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)C1
CCn1cc(nn1)S(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1
Cn1cc(cn1)S(=O)(=O)N1CC(CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)C1
Cn1cnnc1S(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1
Cn1cc(cn1)S(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1
Cn1cc(nn1)S(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1
Cn1cc(cn1)S(=O)(=O)N1CC(CNC(=O)c2ccc(Cl)cc2Cl)(C1)c1ncccc1F
Fc1cccnc1C1(CNC(=O)c2ccc(Cl)cc2Cl)CCN(CC1)S(=O)(=O)CC1CC1
Cn1ncnc1S(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)c1ncccc1F
FC(F)(F)Cn1cc(nn1)S(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1
Cn1cc(nn1)S(=O)(=O)N1CC(CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)C1
Cn1cc(nn1)S(=O)(=O)[C@H]1CC[C@](CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1 |r,wU:12.13,9.9,wD:12.26,(-1.1,-10.55,;-1.99,-9.3,;-1.5,-7.84,;-2.75,-6.91,;-4,-7.81,;-3.53,-9.28,;-2.73,-5.37,;-1.19,-5.38,;-4.27,-5.37,;-2.8,-3.85,;-4.13,-3.1,;-4.12,-1.55,;-2.79,-.78,;-1.45,-.02,;-.13,-.8,;1.21,-.03,;1.22,1.51,;2.54,-.81,;2.53,-2.35,;3.85,-3.12,;5.19,-2.36,;6.52,-3.14,;5.2,-.81,;3.87,-.04,;3.87,1.5,;-4.13,-.01,;-4.13,1.53,;-3.36,2.87,;-4.9,2.87,;-1.46,-1.56,;-1.46,-3.09,)|
Cn1cc(nn1)S(=O)(=O)[C@H]1CC[C@@](CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1 |r,wU:12.26,9.9,wD:12.13,(28.49,-45.82,;27.6,-44.56,;28.09,-43.1,;26.85,-42.18,;25.6,-43.08,;26.06,-44.55,;26.86,-40.64,;28.4,-40.65,;25.32,-40.63,;26.79,-39.12,;25.46,-38.36,;25.47,-36.82,;26.81,-36.05,;28.14,-35.28,;29.47,-36.06,;30.81,-35.3,;30.82,-33.76,;32.14,-36.08,;32.12,-37.61,;33.45,-38.39,;34.79,-37.63,;36.12,-38.4,;34.79,-36.08,;33.46,-35.31,;33.46,-33.77,;25.46,-35.27,;25.46,-33.73,;26.23,-32.4,;24.69,-32.4,;28.14,-36.82,;28.13,-38.36,)|
CN1C[C@H]2[C@H](CN(Cc3cccc(Cl)c3)C(=O)c3cn(C)cn3)[C@H]2C1 |r|
Cn1cnc(c1)C(=O)N(Cc1cccc(Cl)c1)[C@@H]1CC[C@H](N)CC1 |r,wU:17.18,20.22,(3.36,-16.16,;4.05,-14.78,;3.34,-13.41,;4.42,-12.32,;5.8,-13.01,;5.57,-14.53,;7.16,-12.3,;7.23,-10.76,;8.46,-13.13,;9.83,-12.42,;11.12,-13.25,;11.05,-14.78,;12.34,-15.61,;13.71,-14.9,;13.78,-13.36,;15.14,-12.64,;12.48,-12.54,;8.39,-14.67,;7.02,-15.37,;6.95,-16.9,;8.24,-17.73,;8.16,-19.27,;9.61,-17.03,;9.69,-15.48,)|
CN(CC[C@@H](Oc1ccc(cc1)C(=O)c1ccc(C)cc1)c1ccccc1)CC(O)=O |r|
Cn1cnc(c1)C(=O)N(C[C@H]1[C@@H]2CNC[C@H]12)Cc1cccc(Cl)c1 |r|
Cn1cnc(c1)C(=O)N(C[C@H]1[C@@H]2CN(CC3CC3)C[C@H]12)Cc1cccc(OC(F)(F)F)c1 |r|
CN1C[C@H]2[C@H](CN(Cc3ccc(F)c(Cl)c3)C(=O)c3cn(C)cn3)[C@H]2C1 |r|
Cn1cnc(c1)C(=O)N(C[C@H]1[C@@H]2CNC[C@H]12)Cc1cccc(OC(F)(F)F)c1 |r|
Cn1cnc(c1)C(=O)N(C[C@H]1[C@@H]2CNC[C@H]12)Cc1ccc(F)c(Cl)c1 |r|
CCN1C[C@H]2[C@H](CN(Cc3cccc(OC(F)(F)F)c3)C(=O)c3cn(C)cn3)[C@H]2C1 |r|
Cn1cnc(c1)C(=O)N(C[C@H]1[C@@H]2CN(CC3CCCC3)C[C@H]12)Cc1cccc(OC(F)(F)F)c1 |r|
CCN1C[C@H]2[C@H](CN(Cc3cccc(Cl)c3)C(=O)c3cn(C)cn3)[C@H]2C1 |r|
CN1C[C@H]2[C@H](CN(Cc3cccc(OC(F)(F)F)c3)C(=O)c3cn(C)cn3)[C@H]2C1 |r|
CC(F)CN1C[C@@H]2C[C@@H](C[C@@H]2C1)N(Cc1cccc(OC(F)(F)F)c1)C(=O)c1cn(C)cn1 |r|
Cn1cnc(c1)C(=O)N(Cc1cccc(OC(F)(F)F)c1)[C@@H]1C[C@@H]2CNC[C@@H]2C1 |r|
Cn1cnc(c1)C(=O)N(Cc1ccc(F)c(c1)C(F)(F)F)[C@@H]1C[C@@H]2CNC[C@@H]2C1 |r|
CCN1C[C@@H]2C[C@@H](C[C@@H]2C1)N(Cc1ccc(F)c(c1)C(F)(F)F)C(=O)c1cn(C)cn1 |r|
CN1C[C@@H]2C[C@@H](C[C@@H]2C1)N(Cc1ccc(F)c(c1)C(F)(F)F)C(=O)c1cn(C)cn1 |r|
Cn1cnc(c1)C(=O)N(Cc1cccc(OC2CCCC2)c1)[C@@H]1C[C@@H]2CNC[C@@H]2C1 |r|
CCN1C[C@@H]2C[C@@H](C[C@@H]2C1)N(Cc1cccc(OC(F)(F)F)c1)C(=O)c1cn(C)cn1 |r|
CC(C)Oc1cccc(CN([C@@H]2C[C@@H]3CNC[C@@H]3C2)C(=O)c2cn(C)cn2)c1 |r|
CN1C[C@@H]2C[C@@H](C[C@@H]2C1)N(Cc1cccc(OC(F)(F)F)c1)C(=O)c1cn(C)cn1 |r|
COc1ccc(CN([C@@H]2C[C@@H]3CNC[C@@H]3C2)C(=O)c2cn(C)cn2)cc1OC1CCCC1 |r|
Cn1cnc(c1)C(=O)N(Cc1ccc(F)c(c1)C(F)(F)F)[C@H]1C[C@@H]2CNC[C@@H]2C1 |r|
CN1C[C@@H]2C[C@@H](C[C@@H]2C1)N(Cc1ccc(F)c(OC2CCCC2)c1)C(=O)c1cn(C)cn1 |r|
Cn1cnc(c1)C(=O)N(Cc1cccc(OC(F)(F)F)c1)[C@H]1C[C@H]2CN(CC(C)(C)O)C[C@H]2C1 |r|
Cn1cnc(c1)C(=O)N(Cc1cccc(OC(F)(F)F)c1)[C@H]1C[C@H]2CN(CC(O)c3ccccc3)C[C@H]2C1 |r|
Cn1cnc(c1)C(=O)N(Cc1cccc(Cl)c1)[C@@H]1CC[C@H](N)CC1
Cn1cnc(c1)C(=O)N(Cc1ccc(F)c(OC2CCCC2)c1)[C@@H]1C[C@@H]2CNC[C@@H]2C1 |r|
Cn1cnc(c1)C(=O)N(Cc1cccc(OC(F)(F)F)c1)[C@H]1C[C@H]2CN(CCC(F)(F)F)C[C@H]2C1 |r|
C[C@H](Oc1ccc(cc1C(=O)N1Cc2ccc(Cl)cc2C1)S(C)(=O)=O)C(F)(F)F |r|
C[C@H](Oc1ccc(cc1C(=O)N1Cc2ccc(cc2C1)N1CCOCC1)S(C)(=O)=O)C(F)(F)F |r|
CC(C)Oc1ccc(cc1C(=O)N1Cc2ccc(cc2C1)C1CCOCC1)S(C)(=O)=O
CC(C)COc1ccc(cc1C(=O)N1Cc2cc(cnc2C1)C(F)(F)F)S(C)(=O)=O
C[C@H](Oc1ccc(cc1C(=O)N1Cc2ccc(cc2C1)C1CCCCO1)S(C)(=O)=O)C(F)(F)F |r|
C[C@H](Oc1ccc(cc1C(=O)N1Cc2ccc(cc2C1)C1CCOCC1)S(C)(=O)=O)C(F)(F)F |r|
CC(C)Oc1ccc(cc1C(=O)N1Cc2cc(cnc2C1)C(F)(F)F)S(C)(=O)=O
C[C@H](Oc1ccc(cc1C(=O)N1Cc2cccc(C)c2C1)S(C)(=O)=O)C(F)(F)F |r|
COc1cccc2CN(Cc12)C(=O)c1cc(ccc1O[C@@H](C)C(F)(F)F)S(C)(=O)=O |r|
C[C@H](Oc1ccc(cc1C(=O)N1Cc2cccc(C#N)c2C1)S(C)(=O)=O)C(F)(F)F |r|
CS(=O)(=O)c1ccc(N2CCOCC2)c(c1)C(=O)N1Cc2cc(cnc2C1)C(F)(F)F
C[C@H](Oc1ccc(cc1C(=O)N1Cc2cc(cnc2C1)C(F)(F)F)S(C)(=O)=O)C(F)(F)F |r|
C[C@H](Oc1ccc(cc1C(=O)N1Cc2ccc(cc2C1)N1CCCC1)S(C)(=O)=O)C(F)(F)F |r|
C[C@H](Oc1ccc(cc1C(=O)N1Cc2ccc(cc2C1)N1CCN(C)CC1)S(C)(=O)=O)C(F)(F)F |r|
C[C@H](Oc1ccc(cc1C(=O)N1Cc2cnc(cc2C1)C(F)(F)F)S(C)(=O)=O)C(F)(F)F |r|
C[C@H](Oc1ccc(cc1C(=O)N1Cc2ccc(nc2C1)C(F)(F)F)S(C)(=O)=O)C(F)(F)F |r|
C[C@H](Oc1ccc(cc1C(=O)N1Cc2ccc(cc2C1)-c1ccccn1)S(C)(=O)=O)C(F)(F)F |r|
C[C@H](Oc1ccc(cc1C(=O)N1Cc2ccc(cc2C1)-c1ccncc1)S(C)(=O)=O)C(F)(F)F |r|
COc1ccc2CN(Cc2c1)C(=O)c1cc(ccc1O[C@@H](C)C(F)(F)F)S(C)(=O)=O |r|
CS(=O)(=O)c1ccc(OCCC(F)(F)F)c(c1)C(=O)N1Cc2ccc(cc2C1)C1CCOCC1
CS(=O)(=O)c1ccc(OCc2ccccc2)c(c1)C(=O)N1Cc2cc(cnc2C1)C(F)(F)F
CS(=O)(=O)c1ccc(OCCC(F)(F)F)c(c1)C(=O)N1Cc2cc(cnc2C1)C(F)(F)F
C[C@H](Oc1ccc(cc1C(=O)N1Cc2ccccc2C1)S(C)(=O)=O)C(F)(F)F |r|
C[C@H](Oc1ccc(cc1C(=O)N1Cc2ccc(cc2C1)C(F)(F)F)S(C)(=O)=O)C(F)(F)F |r|
C[C@H](Oc1ccc(cc1C(=O)N1Cc2ccc(cc2C1)-c1ccccc1)S(C)(=O)=O)C(F)(F)F |r|
CS(=O)(=O)c1ccc(-c2ccc(F)cc2)c(c1)C(=O)N1Cc2ccc(cc2C1)C1CCOCC1
CS(=O)(=O)c1ccc(-c2ccc(F)c(F)c2)c(c1)C(=O)N1Cc2cc(cnc2C1)C(F)(F)F
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1ccnc2ccccc12 |(49.46,-16.1,;48.73,-17.46,;47.2,-17.51,;46.72,-16.05,;45.18,-16.05,;44.7,-17.51,;43.37,-18.27,;42.04,-17.49,;40.71,-18.25,;40.7,-19.79,;42.04,-20.57,;43.37,-19.8,;39.37,-20.55,;38.03,-19.78,;36.7,-20.54,;36.69,-22.08,;38.03,-22.86,;39.36,-22.09,;45.95,-18.42,;45.95,-19.95,;44.62,-20.72,;44.62,-22.26,;45.95,-23.03,;47.3,-22.25,;48.64,-23.01,;49.97,-22.23,;49.95,-20.67,;48.61,-19.92,;47.29,-20.7,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc2cnccc12 |(18.08,-15.77,;17.35,-17.13,;15.81,-17.17,;15.34,-15.71,;13.8,-15.71,;13.32,-17.17,;11.99,-17.94,;10.66,-17.16,;9.32,-17.92,;9.32,-19.46,;10.65,-20.24,;11.99,-19.47,;7.98,-20.22,;6.65,-19.44,;5.32,-20.21,;5.31,-21.75,;6.65,-22.52,;7.98,-21.75,;14.57,-18.08,;14.57,-19.62,;13.23,-20.39,;13.23,-21.92,;14.57,-22.7,;15.91,-21.92,;17.26,-22.68,;18.59,-21.89,;18.57,-20.34,;17.23,-19.59,;15.9,-20.37,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc2ncccc12 |(33.75,-15.3,;33.02,-16.65,;31.48,-16.7,;31,-15.24,;29.46,-15.24,;28.99,-16.7,;27.66,-17.46,;26.32,-16.68,;24.99,-17.44,;24.98,-18.99,;26.32,-19.76,;27.65,-19,;23.65,-19.75,;22.32,-18.97,;20.98,-19.73,;20.97,-21.27,;22.31,-22.05,;23.64,-21.28,;30.23,-17.61,;30.23,-19.14,;28.9,-19.91,;28.9,-21.45,;30.23,-22.22,;31.58,-21.44,;32.92,-22.2,;34.25,-21.42,;34.23,-19.87,;32.89,-19.11,;31.57,-19.9,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc2cccnc12 |(49.41,-6.17,;48.68,-7.53,;47.14,-7.57,;46.66,-6.11,;45.12,-6.11,;44.65,-7.58,;43.32,-8.34,;41.99,-7.56,;40.65,-8.32,;40.64,-9.86,;41.98,-10.64,;43.31,-9.87,;39.31,-10.62,;37.98,-9.84,;36.64,-10.61,;36.64,-12.15,;37.98,-12.92,;39.31,-12.15,;45.89,-8.48,;45.9,-10.02,;44.56,-10.79,;44.56,-12.33,;45.89,-13.1,;47.24,-12.32,;48.58,-13.08,;49.91,-12.29,;49.89,-10.74,;48.55,-9.99,;47.23,-10.77,)|
CC(C)c1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1ccccc1F |(2.67,-3.47,;1.87,-4.79,;2.6,-6.14,;.33,-4.75,;-.15,-3.28,;-1.69,-3.28,;-2.16,-4.74,;-3.49,-5.52,;-3.48,-7.06,;-4.81,-7.84,;-6.15,-7.07,;-6.16,-5.53,;-4.83,-4.76,;-7.47,-7.84,;-8.81,-7.08,;-10.14,-7.85,;-10.14,-9.39,;-8.8,-10.16,;-7.47,-9.39,;-.92,-5.65,;-.92,-7.18,;-2.26,-7.95,;-2.26,-9.49,;-.93,-10.26,;.41,-9.48,;.41,-7.95,;1.74,-7.18,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1C(C)c1ccncc1
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc2ccncc12 |(2.75,-17.23,;2.02,-18.59,;.48,-18.63,;.01,-17.17,;-1.53,-17.17,;-2.01,-18.64,;-3.34,-19.4,;-4.67,-18.62,;-6.01,-19.38,;-6.01,-20.92,;-4.68,-21.7,;-3.34,-20.93,;-7.35,-21.68,;-8.68,-20.9,;-10.01,-21.67,;-10.02,-23.21,;-8.68,-23.98,;-7.35,-23.22,;-.76,-19.54,;-.76,-21.08,;-2.1,-21.85,;-2.1,-23.39,;-.76,-24.16,;.58,-23.38,;1.93,-24.14,;3.26,-23.35,;3.24,-21.8,;1.9,-21.05,;.57,-21.83,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1ccccc1F |(31.78,4.31,;30.63,3.28,;29.17,3.76,;28.69,5.23,;27.15,5.23,;26.68,3.77,;25.35,2.99,;25.36,1.45,;24.03,.67,;22.69,1.44,;22.68,2.97,;24.01,3.75,;21.37,.67,;20.03,1.43,;18.7,.66,;18.7,-.88,;20.04,-1.65,;21.37,-.88,;27.92,2.86,;27.92,1.33,;26.58,.56,;26.58,-.98,;27.91,-1.75,;29.25,-.98,;29.25,.56,;30.58,1.33,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc2[nH]ncc12 |(17.39,-6.43,;16.66,-7.78,;15.12,-7.83,;14.64,-6.37,;13.1,-6.37,;12.62,-7.83,;11.29,-8.59,;9.96,-7.81,;8.62,-8.58,;8.62,-10.12,;9.96,-10.9,;11.29,-10.13,;7.28,-10.88,;5.95,-10.1,;4.61,-10.87,;4.61,-12.41,;5.95,-13.18,;7.28,-12.42,;13.87,-8.74,;13.87,-10.28,;12.54,-11.05,;12.54,-12.59,;13.87,-13.36,;15.22,-12.58,;16.69,-13.04,;17.58,-11.79,;16.67,-10.55,;15.21,-11.04,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc2CNCCc12 |(20.49,-34.45,;19.76,-35.81,;18.22,-35.85,;17.75,-34.39,;16.21,-34.39,;15.73,-35.86,;14.4,-36.62,;13.07,-35.84,;11.73,-36.6,;11.73,-38.14,;13.07,-38.92,;14.4,-38.15,;10.39,-38.9,;9.06,-38.12,;7.73,-38.89,;7.72,-40.43,;9.06,-41.2,;10.39,-40.44,;16.98,-36.76,;16.98,-38.3,;15.65,-39.07,;15.64,-40.61,;16.98,-41.38,;18.33,-40.6,;19.67,-41.36,;21,-40.57,;20.98,-39.02,;19.64,-38.27,;18.31,-39.05,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc2[nH]cnc12 |(32.52,-5.85,;31.79,-7.21,;30.25,-7.26,;29.77,-5.79,;28.23,-5.79,;27.76,-7.26,;26.43,-8.02,;25.1,-7.24,;23.76,-8,;23.75,-9.54,;25.09,-10.32,;26.42,-9.55,;22.42,-10.3,;21.09,-9.53,;19.75,-10.29,;19.75,-11.83,;21.09,-12.61,;22.42,-11.84,;29,-8.16,;29.01,-9.7,;27.67,-10.47,;27.67,-12.01,;29,-12.78,;30.35,-12,;31.82,-12.47,;32.72,-11.21,;31.8,-9.97,;30.34,-10.46,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1Cc1ccncc1
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc2ccn(C)c12 |(51.49,3.11,;50.76,1.75,;49.22,1.71,;48.74,3.17,;47.2,3.17,;46.73,1.7,;45.39,.94,;44.06,1.72,;42.72,.96,;42.72,-.58,;44.06,-1.36,;45.39,-.59,;41.38,-1.34,;40.05,-.57,;38.71,-1.33,;38.71,-2.87,;40.05,-3.65,;41.38,-2.88,;47.97,.8,;47.98,-.74,;46.64,-1.51,;46.64,-3.05,;47.97,-3.82,;49.32,-3.04,;50.79,-3.5,;51.68,-2.25,;50.76,-1.02,;51.23,.45,;49.31,-1.51,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc2c[n+]([O-])ccc12 |(35.1,-25.27,;34.37,-26.62,;32.83,-26.67,;32.35,-25.21,;30.81,-25.21,;30.34,-26.67,;29.01,-27.43,;27.68,-26.65,;26.34,-27.42,;26.33,-28.96,;27.67,-29.73,;29,-28.97,;25,-29.72,;23.67,-28.94,;22.33,-29.7,;22.33,-31.24,;23.67,-32.02,;25,-31.25,;31.58,-27.58,;31.59,-29.11,;30.25,-29.88,;30.25,-31.42,;31.59,-32.19,;32.93,-31.41,;34.27,-32.17,;35.61,-31.39,;36.95,-32.14,;35.59,-29.84,;34.24,-29.08,;32.92,-29.87,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc2cn[nH]c12 |(1.91,-8.22,;1.18,-9.58,;-.37,-9.62,;-.84,-8.16,;-2.38,-8.16,;-2.86,-9.62,;-4.19,-10.39,;-5.52,-9.6,;-6.86,-10.37,;-6.87,-11.91,;-5.53,-12.69,;-4.2,-11.92,;-8.2,-12.67,;-9.54,-11.89,;-10.87,-12.66,;-10.88,-14.2,;-9.54,-14.98,;-8.21,-14.21,;-1.61,-10.53,;-1.61,-12.07,;-2.95,-12.84,;-2.95,-14.38,;-1.61,-15.15,;-.26,-14.37,;1.2,-14.83,;2.09,-13.58,;1.18,-12.34,;-.28,-12.83,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc2c1cc[nH]c2=O |(3.55,-35.44,;2.82,-36.8,;1.28,-36.84,;.81,-35.38,;-.73,-35.38,;-1.21,-36.84,;-2.54,-37.61,;-3.87,-36.83,;-5.21,-37.59,;-5.21,-39.13,;-3.87,-39.91,;-2.54,-39.14,;-6.55,-39.89,;-7.88,-39.11,;-9.21,-39.88,;-9.22,-41.42,;-7.88,-42.19,;-6.55,-41.42,;.04,-37.75,;.04,-39.29,;-1.29,-40.06,;-1.3,-41.59,;.04,-42.37,;1.39,-41.59,;1.37,-40.04,;2.7,-39.26,;4.04,-40.01,;4.06,-41.56,;2.73,-42.35,;2.74,-43.89,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cncc2ccccc12 |(2.85,-26.54,;2.12,-27.9,;.58,-27.94,;.11,-26.48,;-1.43,-26.48,;-1.91,-27.95,;-3.24,-28.71,;-4.57,-27.93,;-5.91,-28.69,;-5.91,-30.23,;-4.57,-31.01,;-3.24,-30.24,;-7.25,-30.99,;-8.58,-30.21,;-9.91,-30.98,;-9.92,-32.52,;-8.58,-33.29,;-7.25,-32.53,;-.66,-28.85,;-.66,-30.39,;-1.99,-31.16,;-2,-32.7,;-.66,-33.47,;.69,-32.69,;2.03,-33.45,;3.36,-32.66,;3.34,-31.11,;2,-30.36,;.67,-31.14,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc2cc[nH]c12 |(34.8,3.29,;34.07,1.93,;32.52,1.88,;32.05,3.35,;30.51,3.35,;30.03,1.88,;28.7,1.12,;27.37,1.9,;26.03,1.14,;26.02,-.41,;27.36,-1.18,;28.69,-.41,;24.69,-1.17,;23.36,-.39,;22.02,-1.15,;22.01,-2.69,;23.35,-3.47,;24.69,-2.7,;31.28,.98,;31.28,-.56,;29.94,-1.33,;29.94,-2.87,;31.28,-3.64,;32.63,-2.86,;34.09,-3.32,;34.98,-2.07,;34.07,-.84,;32.61,-1.33,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1nccc2ccccc12 |(19.56,-25.35,;18.83,-26.71,;17.29,-26.75,;16.81,-25.29,;15.27,-25.29,;14.8,-26.76,;13.47,-27.52,;12.14,-26.74,;10.8,-27.5,;10.79,-29.04,;12.13,-29.82,;13.46,-29.05,;9.46,-29.8,;8.13,-29.02,;6.79,-29.79,;6.79,-31.33,;8.13,-32.1,;9.46,-31.34,;16.04,-27.66,;16.05,-29.2,;14.71,-29.97,;14.71,-31.51,;16.05,-32.28,;17.39,-31.5,;18.73,-32.26,;20.07,-31.47,;20.05,-29.92,;18.7,-29.17,;17.38,-29.95,)|
CN1CCCC[C@H]1[C@@H](NC(=O)c1cccc(c1I)C(F)(F)F)c1ccccc1 |r|
FC(F)(F)c1cccc(C(=O)N[C@H]([C@@H]2CCCCN2)c2ccccc2)c1Cl |r|
CN1CCCC[C@H]1[C@@H](NC(=O)c1cccc(c1Cl)C(F)(F)F)c1ccccc1 |r|
O=C1NCC(c2ccccc2)C11CCN(CC1)C1(CCCCC1)c1ccc(cc1)C#N
CCCC1CNC(=O)C11CCN(CC1)C1(CCCCC1)c1ccccc1
Fc1cccc(c1)C1(CCCCC1)N1CCC2(CC1)C(CNC2=O)c1ccccc1
Cc1ccc(cc1)C1(CCCCC1)N1CCC2(CC1)C(CNC2=O)c1ccccc1
Fc1ccc(cc1)C1CNC(=O)C11CCN(CC1)C1(CCCCC1)c1ccsc1
Fc1ccc(cc1)C1CNC(=O)C11CCN(CC1)C1(CCCCC1)c1ccc(F)cc1
O=C1NCC(c2ccccc2)C11CCN(CC1)C1(CCCCC1)c1ccccc1
FC(F)(F)c1ccc(cc1)C1(CCCCC1)N1CCC2(CC1)C(CNC2=O)c1ccccc1
Clc1ccc(cc1)C1(CCCCC1)N1CCC2(CC1)C(CNC2=O)c1ccccc1
Fc1ccc(cc1)C1CNC(=O)C11CCN(CC1)C1(CCCCC1)c1cccs1
Cc1cccc(c1)C1(CCCCC1)N1CCC2(CC1)C(CNC2=O)c1ccc(F)cc1
COc1cccc(c1)C1(CCCCC1)N1CCC2(CC1)C(CNC2=O)c1ccccc1
Cc1ccc(cc1)C1(CCCCC1)N1CCC2(CC1)C(CNC2=O)c1ccc(F)cc1
Fc1ccc(cc1)C1CNC(=O)C11CCN(CC1)C1(CCCCC1)c1cccc(OC(F)(F)F)c1
O=C1NCC(c2ccccc2)C11CCN(CC1)C1(CCOCC1)c1ccccc1
COc1ccc(Sc2ccccc2N2CCN(CC(O)=O)C(C)(C)C2)cc1
COc1ccc(Sc2ccccc2N2CCN(CC(O)=O)CC2C)cc1
COc1ccc(Sc2ccccc2N2C[C@H](C)N(CC(O)=O)C[C@H]2C)cc1
CN(CC[C@@H](Oc1ccc(cc1)C(F)(F)F)c1ccccc1)CC(O)=O
CC1CN(C(C)CN1CC(O)=O)c1ccccc1Sc1ccc(NC(C)=O)cc1
COc1ccc(Sc2ccccc2N2CCN(CC(O)=O)CC2)cc1
COc1ccc(Sc2ccccc2N2CC(C)N(CC(O)=O)CC2C)cc1
COc1ccc(Sc2ccc(C)cc2N2CCN(CC(O)=O)C(C)C2)cc1
CC1CN(C(C)CN1CC(O)=O)c1ccccc1Sc1ccc(F)cc1
COc1ccc(Sc2ccc(OC)cc2N2CCN(CC(O)=O)C(C)C2)cc1
CC1CN(C(C)CN1CC(O)=O)c1ccccc1Sc1ccc(C)cc1
CC1CN(C(C)CN1CC(O)=O)c1ccccc1Sc1ccc(O)cc1
CC1CN(C(C)CN1CC(O)=O)c1ccccc1Sc1ccc(Cl)cc1
COc1ccc(Sc2ccc(Cl)cc2N2CCN(CC(O)=O)C(C)C2)cc1
COc1ccc(Sc2ccc(OC)cc2N2CC(C)N(CC(O)=O)CC2C)cc1
CN(CC[C@@H](Oc1ccc(cc1)-c1ccccc1)c1ccc(F)cc1)CC(O)=O |r|
COc1ccc(Sc2ccc(Cl)cc2N2CCN(CC(O)=O)[C@@H](C)C2)cc1
COc1ccc(Sc2ccccc2N2C[C@H](C)N(CC(O)=O)C[C@@H]2C)cc1
COc1ccc(Sc2ccccc2N2C[C@@H](C)N(CC(O)=O)C[C@H]2C)cc1
COc1ccc(Sc2ccc(Cl)cc2N2CCN(CC(O)=O)[C@H](C)C2)cc1
CC1CN(C(C)CN1CC(O)=O)c1ccccc1Sc1ccc(cc1)-c1ccccc1
COc1ccc(Sc2ccc(Cl)cc2N2CC(C)N(CC(O)=O)CC2C)cc1
COc1ccc(Sc2ccccc2N2C[C@@H](C)N(CC(O)=O)C[C@@H]2C)cc1
CC1CN(C(C)CN1CC(O)=O)c1ccccc1Sc1ccccc1
COc1ccc(Sc2ccccc2N2CCN(CC(O)=O)C(C)C2)cc1
CCc1nnc(-c2ccc(nc2)-c2ccccc2)n1-c1cccc(C#N)c1C |(17.73,-47.68,;16.46,-48.55,;15.07,-47.89,;14.59,-46.43,;13.05,-46.43,;12.58,-47.9,;11.25,-48.66,;9.92,-47.87,;8.58,-48.63,;8.57,-50.17,;9.91,-50.95,;11.24,-50.19,;7.24,-50.94,;5.91,-50.15,;4.57,-50.92,;4.56,-52.46,;5.9,-53.23,;7.23,-52.47,;13.83,-48.8,;13.83,-50.34,;12.5,-51.11,;12.5,-52.65,;13.84,-53.42,;15.17,-52.65,;16.51,-53.42,;17.84,-54.17,;15.17,-51.1,;16.5,-50.33,)|
FC(F)(F)c1cccc(C(=O)N[C@H]([C@@H]2CCCCN2)c2ccccc2)c1I |r|
CC(C)c1ccc(cc1)C(=C/CC(N)C([O-])=O)\c1ccsc1
CC(C)c1ccc(cc1)C(=C/CC(N)C([O-])=O)\c1ccccc1F
CC(C)c1ccc(cc1)C(=C\CC(N)C([O-])=O)\c1ccc(F)cc1F
NC(C\C=C(\c1ccc(cc1)-c1ccccc1)c1ccc(F)cc1F)C([O-])=O
CCc1ccc(cc1CC)C(=C/CC(N)C([O-])=O)\c1ccc(F)cc1F
NC(C\C=C(/c1cccc(c1)-c1ccccc1)c1ccc(F)cc1F)C([O-])=O
NC(C\C=C(/c1cccnc1)c1ccc(F)cc1F)C([O-])=O
NC(C\C=C(\c1ccc(F)cc1F)c1ccccc1-c1ccccc1)C([O-])=O
CC(C)c1ccc(cc1)C(=C/CC(N)C([O-])=O)\c1cccnc1
CC(C)c1cccc(c1)C(=C/CC(N)C([O-])=O)\c1ccc(F)cc1F
CC(C)c1ccc(cc1)C(=C/CC(N)C([O-])=O)\c1ccc(cc1)C(C)(C)C
NC(C\C=C(/c1ccsc1)c1ccc(F)cc1F)C([O-])=O
COc1ccc(cc1)C(=C\CC(N)C([O-])=O)\c1ccc(cc1)C(C)C
CC(C)c1ccc(cc1)C(=C/CC(N)C([O-])=O)\c1ccc(cc1)C#N
[#6]-[#6](-[#6])-c1ccc(cc1)-[#6](=[#6]/[#6]-[#6](-[#7])-[#6](-[#8-])=O)\c1ccc(cc1)-[#6](-[#6])-[#6]
CCc1ccc(cc1)C(=C/CC(N)C([O-])=O)\c1ccc(F)cc1F
CC(C)c1ccc(cc1)C(=C/CC(N)C([O-])=O)\c1ccc(F)cc1F
COc1ccc(cc1)C(=C/CC(N)C([O-])=O)\c1ccc(F)cc1F
NC(C\C=C(/c1ccc(cc1)C#N)c1ccc(F)cc1F)C([O-])=O
CC(C)c1ccc(cc1)C(=C/CC(N)C([O-])=O)\c1ccccc1
Cc1ccc(cc1)C(=C/CC(N)C([O-])=O)\c1ccc(F)cc1F
NC(C\C=C(/c1ccc(cc1)-c1ccccc1)c1ccc(F)cc1F)C([O-])=O
NC(C\C=C(/c1ccccc1)c1ccc(F)cc1F)C([O-])=O
CC(C)c1ccc(cc1)C(=C/CC(N)C([O-])=O)\c1ccc(cc1)-c1ccccc1
NC(C\C=C(/c1ccc2ccccc2c1)c1ccc(F)cc1F)C([O-])=O
CC(C)(C)c1ccc(cc1)C(=C/CC(N)C([O-])=O)\c1ccc(F)cc1F
O=C1NCC(c2ccccc2)C11CCN(CC1)C1(CCCCC1)C1CCCC1
O=C1NCC(c2ccccc2)C11CCN(CC1)C1(CCCCC1)C1CCCCC1
CC(C)C1(CCCCC1)N1CCC2(CC1)C(CNC2=O)c1ccc(F)cc1
Fc1ccc(cc1)C1CNC(=O)C11CCN(CC1)C1(CCCCC1)c1cccc(c1)C#N
O=C1NCN(c2ccccc2)C11CCN(CC1)C1(CCCCC1)c1ccccc1
[#6]\[#6](-[#6])=[#6]/C1([#6]-[#6]-[#6]-[#6]-[#6]1)[#7]-1-[#6]-[#6]C2([#6]-[#6]-1)[#6](-[#6]-[#7]-[#6]2=O)-c1ccccc1
CCC1(CCCCC1)N1CCC2(CC1)C(CNC2=O)c1ccc(F)cc1
Fc1ccc(cc1)C1CNC(=O)C11CCN(CC1)C1(CCCCC1)C1CC1
O=C1NCC(c2ccccc2)C11CCN(CC1)C1(CCCCC1)C1CC1
CC(C)C1(CCCCC1)N1CCC2(CC1)C(CNC2=O)c1ccccc1
O=C1NCC(c2ccccc2)C11CCN(CC1)C1(CCCCC1)c1ccsc1
CCCC1CNC(=O)C11CCN(CC1)C1(CCCCC1)c1ccc(C)s1
CCCC1CNC(=O)C11CCN(CC1)C1(CCCCC1)c1cccs1
CCCC1CNC(=O)C11CCN(CC1)C1(CCCCC1)c1ccc(F)cc1
Cc1ccccc1C1(CCCCC1)N1CCC2(CC1)C(CNC2=O)c1ccc(F)cc1
Fc1ccc(cc1)C1CNC(=O)C11CCN(CC1)C1(CCCCC1)c1cccc(F)c1
O=C1NCC(c2ccccc2)C11CCN(CC1)C1(CCCOC1)c1ccccc1
FC(F)(F)Oc1ccc(cc1)C1(CCCCC1)N1CCC2(CC1)C(CNC2=O)c1ccccc1
Cc1ccc(cc1)C1CNC(=O)C11CCN(CC1)C1(CCCCC1)c1ccccc1
Cc1ccc(cc1)C1CNC(=O)C11CCN(CC1)C1(CCCCC1)c1ccc(F)cc1
Fc1ccc(cc1)C1(CCCCC1)N1CCC2(CC1)C(CNC2=O)c1ccc(cc1)C(F)(F)F
O=C1NCC(c2ccccc2)C11CCN(CC1)C1(CCCCC1)c1cccs1
Fc1ccc(cc1)C1CNC(=O)C11CCN(CC1)C1(CCC1)c1ccc(F)cc1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)C(=O)N(C)C
CCCS(=O)(=O)N1CCC(CNC(=O)c2c(F)ccc(Cl)c2F)(CC1)C(=O)N1CCOCC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(F)cc2C(F)(F)F)(CC1)C(=O)N1CCOCC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)C(=O)N1CCOCC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(cc2F)C(F)(F)F)(CC1)C(=O)N1CCOCC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(F)cc2Cl)(CC1)C(=O)N1CCOCC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2Cl)(CC1)C(=O)N1CCOCC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)C(=O)N1CCN(C)CC1
CCCS(=O)(=O)N1CCC(CC1)([C@H](C)NC(=O)c1ccc(Cl)cc1Cl)C(=O)N1CCOCC1
CCCS(=O)(=O)N1CCC(CNC(=O)CC)(CC1)C(=O)N1CCOCC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)C(=O)NCC
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)C(=O)NCC1(C)COC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2c(F)cccc2Cl)(CC1)C(=O)N1CCOCC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2cc(F)c(Cl)cc2Cl)(CC1)C(=O)N1CCOCC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2c(F)cccc2F)(CC1)C(=O)N1CCOCC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)C(=O)C1CC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)C(=O)N1CC(N)C1
CCCS(=O)(=O)N1CCC(CC1)([C@@H](C)NC(=O)c1ccc(Cl)cc1Cl)C(=O)N1CCOCC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC1)C(=O)N1CCC(C1)N(C)C
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2)(CC1)C(=O)N1CCOCC1
CCCS(=O)(=O)N1CCC(CNC(=O)c2ccccc2OC(F)(F)F)(CC1)C(=O)N1CCOCC1
CCCS(=O)(=O)N1CCC(CNC(=O)C2CC2)(CC1)C(=O)N1CCOCC1
CS(=O)(=O)c1ccc(O)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1F)C#N
COc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1F)C#N)S(C)(=O)=O
CCOc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1F)C#N)S(C)(=O)=O
CCCOc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1F)C#N)S(C)(=O)=O
CC(C)COc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1F)C#N)S(C)(=O)=O
CC(C)Oc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1F)C#N)S(C)(=O)=O
CS(=O)(=O)c1ccc(OC2CCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1F)C#N
CS(=O)(=O)c1ccc(OC2CCCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1F)C#N
CS(=O)(=O)c1ccc(OC2CCCCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1F)C#N
CS(=O)(=O)c1ccc(OCC(F)(F)F)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1F)C#N
CC(Oc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1F)C#N)S(C)(=O)=O)C(F)(F)F
CS(=O)(=O)c1ccc(OCC2CCCCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1F)C#N
CS(=O)(=O)c1ccc(OCc2ccccc2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1F)C#N
CS(=O)(=O)c1ccc(OC2CCOCC2)c(c1)C(=O)N1CCN(CC1)c1ccc(cc1F)C#N
CN(C)CCOc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1F)C#N)S(C)(=O)=O
CC(Oc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(C)cc1)S(C)(=O)=O)C(F)(F)F
COc1ccc(cc1)N1CCN(CC1)C(=O)c1cc(ccc1OC(C)C(F)(F)F)S(C)(=O)=O
CC(Oc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1)C#N)S(C)(=O)=O)C(F)(F)F
CC(Oc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1)C(F)(F)F)S(C)(=O)=O)C(F)(F)F
CC(Oc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1)S(C)(=O)=O)S(C)(=O)=O)C(F)(F)F
CC(Oc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1)C(C)=O)S(C)(=O)=O)C(F)(F)F
CC(Oc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1F)C(F)(F)F)S(C)(=O)=O)C(F)(F)F
CC(Oc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cc1Cl)C(F)(F)F)S(C)(=O)=O)C(F)(F)F
CC(Oc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(cn1)C(F)(F)F)S(C)(=O)=O)C(F)(F)F
CC(Oc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(nc1)C(F)(F)F)S(C)(=O)=O)C(F)(F)F
CC(Oc1ccc(cc1C(=O)N1CCN(CC1)c1cnc(cn1)C(F)(F)F)S(C)(=O)=O)C(F)(F)F
CC(Oc1ccc(cc1C(=O)N1CCN(CC1)c1ncc(cn1)C(F)(F)F)S(C)(=O)=O)C(F)(F)F
CC(Oc1ccc(cc1C(=O)N1CCN(CC1)c1cnc(nc1)C(F)(F)F)S(C)(=O)=O)C(F)(F)F
CC(Oc1ccc(cc1C(=O)N1CCN(CC1)c1ccc(nn1)C(F)(F)F)S(C)(=O)=O)C(F)(F)F
C[C@H](Oc1ccc(cc1C(=O)N1CCN(CC1)c1ncc(cc1F)C(F)(F)F)S(C)(=O)=O)C(F)(F)F |r|
CC(Oc1ccc(cc1C(=O)N1CCN(CC1)c1ncc(cc1C)C(F)(F)F)S(C)(=O)=O)C(F)(F)F
CC(Oc1ccc(cc1C(=O)N1CCN(CC1)c1ncc(cc1Cl)C(F)(F)F)S(C)(=O)=O)C(F)(F)F
Cc1nnc(Cc2ccc(cc2)-c2ccccc2)n1-c1ccccc1F |(4.87,-24.99,;3.41,-24.51,;2.93,-23.04,;1.39,-23.04,;.92,-24.51,;-.41,-25.28,;-1.75,-24.53,;-1.75,-22.99,;-3.09,-22.23,;-4.42,-23.01,;-4.4,-24.56,;-3.06,-25.31,;-5.76,-22.26,;-5.77,-20.71,;-7.11,-19.96,;-8.44,-20.74,;-8.42,-22.29,;-7.08,-23.04,;2.16,-25.41,;2.16,-26.95,;.82,-27.71,;.82,-29.25,;2.15,-30.02,;3.49,-29.25,;3.49,-27.71,;4.82,-26.94,)|
Fc1ccccc1-n1cnnc1-c1ccc(cc1)-c1ccccc1
CNc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1ccccc1F |(17.26,-39.7,;16.11,-40.73,;14.65,-40.25,;14.17,-38.79,;12.63,-38.79,;12.16,-40.25,;10.83,-41.03,;10.84,-42.57,;9.51,-43.34,;8.17,-42.57,;8.16,-41.04,;9.49,-40.26,;6.85,-43.35,;5.51,-42.58,;4.18,-43.35,;4.18,-44.9,;5.51,-45.67,;6.85,-44.9,;13.4,-41.16,;13.4,-42.69,;12.06,-43.45,;12.06,-44.99,;13.39,-45.77,;14.73,-44.99,;14.73,-43.45,;16.06,-42.68,)|
COc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1ccccc1F |(31.47,-39.01,;30.32,-40.04,;28.86,-39.56,;28.38,-38.09,;26.84,-38.09,;26.37,-39.56,;25.04,-40.33,;25.05,-41.88,;23.72,-42.65,;22.38,-41.88,;22.37,-40.35,;23.7,-39.57,;21.06,-42.65,;19.72,-41.89,;18.39,-42.66,;18.39,-44.21,;19.72,-44.98,;21.06,-44.2,;27.61,-40.46,;27.61,-42,;26.27,-42.76,;26.27,-44.3,;27.6,-45.07,;28.94,-44.3,;28.94,-42.76,;30.27,-41.99,)|
CSc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1ccccc1F |(45.91,-38.95,;44.76,-39.98,;43.3,-39.51,;42.83,-38.04,;41.29,-38.04,;40.81,-39.5,;39.49,-40.28,;39.49,-41.82,;38.16,-42.6,;36.82,-41.83,;36.82,-40.29,;38.14,-39.52,;35.5,-42.6,;34.16,-41.84,;32.84,-42.61,;32.83,-44.15,;34.17,-44.92,;35.5,-44.15,;42.05,-40.41,;42.05,-41.94,;40.72,-42.71,;40.71,-44.25,;42.05,-45.02,;43.39,-44.24,;43.38,-42.71,;44.71,-41.94,)|
CS(=O)(=O)c1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1ccccc1F |(2.75,5.1,;1.61,4.07,;.82,2.75,;2.69,2.88,;.14,4.55,;-.33,6.01,;-1.87,6.01,;-2.35,4.55,;-3.67,3.77,;-3.67,2.23,;-5,1.46,;-6.33,2.23,;-6.34,3.76,;-5.02,4.54,;-7.66,1.45,;-8.99,2.22,;-10.32,1.45,;-10.33,-.1,;-8.99,-.87,;-7.65,-.1,;-1.11,3.64,;-1.11,2.11,;-2.44,1.35,;-2.45,-.19,;-1.11,-.97,;.23,-.19,;.22,1.35,;1.56,2.12,)|
Fc1ccccc1-n1c(nnc1C(F)(F)F)-c1ccc(cc1)-c1ccccc1 |(15.61,2.56,;14.28,1.79,;14.28,.25,;12.94,-.52,;11.61,.25,;11.61,1.79,;12.95,2.56,;12.95,4.09,;11.7,4.99,;12.18,6.46,;13.72,6.46,;14.2,4.99,;15.73,4.99,;16.51,3.66,;16.5,6.33,;17.27,4.99,;10.38,4.22,;10.39,2.67,;9.06,1.9,;7.72,2.67,;7.71,4.2,;9.04,4.98,;6.39,1.9,;5.06,2.66,;3.73,1.89,;3.73,.35,;5.06,-.43,;6.4,.35,)|
CC(C)(C)c1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1ccccc1F |(16.84,-2.84,;16.03,-4.15,;16.77,-5.5,;17.57,-4.15,;14.49,-4.11,;14.02,-2.64,;12.48,-2.64,;12,-4.11,;10.68,-4.88,;10.68,-6.43,;9.35,-7.2,;8.02,-6.43,;8.01,-4.9,;9.33,-4.12,;6.69,-7.2,;5.36,-6.44,;4.03,-7.21,;4.02,-8.75,;5.36,-9.53,;6.7,-8.75,;13.24,-5.01,;13.24,-6.54,;11.91,-7.31,;11.9,-8.85,;13.24,-9.62,;14.58,-8.85,;14.57,-7.31,;15.91,-6.54,)|
COc1ccccc1-n1c(C)nnc1-c1ccc(cc1)-c1ccccc1 |(18.22,-5.11,;16.73,-4.71,;15.64,-5.81,;16.04,-7.28,;14.95,-8.38,;13.47,-7.98,;13.07,-6.5,;14.17,-5.41,;13.77,-3.93,;14.8,-2.77,;16.34,-2.77,;14.01,-1.43,;12.51,-1.76,;12.35,-3.3,;11.02,-4.08,;9.68,-3.32,;8.36,-4.1,;8.37,-5.63,;9.7,-6.41,;11.04,-5.63,;7.04,-6.41,;7.04,-7.96,;5.69,-8.73,;4.36,-7.96,;4.36,-6.41,;5.69,-5.64,)|
Cc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1ccccc1
Cc1nnc(-c2ccc(cc2)-c2ccccc2)n1C1CCCCC1
CC(C)n1c(C)nnc1-c1ccc(cc1)-c1ccccc1
Cc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1ccccc1F |(14.8,-4.75,;13.34,-4.27,;12.87,-2.81,;11.33,-2.81,;10.85,-4.27,;9.53,-5.05,;9.53,-6.59,;8.2,-7.36,;6.86,-6.59,;6.86,-5.06,;8.18,-4.28,;5.54,-7.37,;4.2,-6.6,;2.88,-7.37,;2.87,-8.92,;4.21,-9.69,;5.54,-8.92,;12.09,-5.18,;12.09,-6.71,;10.76,-7.47,;10.75,-9.01,;12.09,-9.79,;13.43,-9.01,;13.42,-7.47,;14.75,-6.7,)|
Cc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc(F)c1
Cc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1ccc(F)cc1
Cc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1ccccc1Cl |(15.78,-13.83,;14.32,-13.35,;13.85,-11.89,;12.3,-11.89,;11.83,-13.35,;10.5,-14.13,;10.51,-15.67,;9.18,-16.45,;7.84,-15.68,;7.83,-14.14,;9.16,-13.36,;6.51,-16.45,;5.18,-15.69,;3.85,-16.46,;3.85,-18,;5.18,-18.77,;6.52,-18,;13.07,-14.26,;13.07,-15.79,;11.73,-16.56,;11.73,-18.1,;13.06,-18.87,;14.4,-18.09,;14.4,-16.56,;15.73,-15.79,)|
Cc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1ccccc1C(F)(F)F |(29.74,-13.3,;28.27,-13.31,;27.8,-11.84,;26.26,-11.84,;25.78,-13.31,;24.46,-14.08,;24.46,-15.63,;23.13,-16.4,;21.8,-15.63,;21.79,-14.1,;23.11,-13.32,;20.47,-16.4,;19.14,-15.64,;17.81,-16.41,;17.81,-17.96,;19.14,-18.73,;20.48,-17.95,;27.03,-14.21,;27.03,-15.75,;25.69,-16.51,;25.69,-18.05,;27.02,-18.82,;28.36,-18.05,;28.35,-16.51,;29.69,-15.74,;31.02,-16.51,;29.69,-14.2,;31.01,-14.96,)|
Cc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1ccccc1C#N |(2.17,-22.75,;.7,-22.27,;.23,-20.8,;-1.31,-20.8,;-1.79,-22.27,;-3.11,-23.04,;-3.11,-24.59,;-4.44,-25.36,;-5.77,-24.59,;-5.78,-23.06,;-4.46,-22.28,;-7.1,-25.36,;-8.43,-24.6,;-9.76,-25.37,;-9.77,-26.92,;-8.43,-27.69,;-7.09,-26.91,;-.55,-23.17,;-.55,-24.71,;-1.88,-25.47,;-1.89,-27.01,;-.55,-27.78,;.79,-27.01,;.78,-25.47,;2.11,-24.7,;3.44,-23.93,)|
Cc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1ccccc1O |(17.62,-21.86,;16.16,-21.38,;15.68,-19.91,;14.14,-19.91,;13.67,-21.37,;12.34,-22.15,;12.35,-23.69,;11.02,-24.47,;9.68,-23.7,;9.67,-22.17,;11,-21.39,;8.36,-24.47,;7.02,-23.71,;5.69,-24.48,;5.69,-26.02,;7.02,-26.79,;8.36,-26.02,;14.91,-22.28,;14.91,-23.81,;13.57,-24.58,;13.57,-26.12,;14.9,-26.89,;16.24,-26.12,;16.24,-24.58,;17.57,-23.81,)|
Cc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1ccccc1C |(32.05,-21.71,;30.58,-21.23,;30.11,-19.76,;28.57,-19.76,;28.09,-21.22,;26.77,-22,;26.77,-23.54,;25.44,-24.32,;24.11,-23.55,;24.1,-22.02,;25.42,-21.24,;22.78,-24.32,;21.45,-23.56,;20.12,-24.33,;20.12,-25.87,;21.45,-26.64,;22.79,-25.87,;29.34,-22.13,;29.34,-23.66,;28,-24.43,;28,-25.97,;29.33,-26.74,;30.67,-25.97,;30.66,-24.43,;32,-23.66,)|
CCc1ccccc1-n1c(C)nnc1-c1ccc(cc1)-c1ccccc1 |(46.21,-23.09,;44.88,-22.32,;43.54,-23.09,;43.55,-24.63,;42.21,-25.4,;40.88,-24.63,;40.88,-23.09,;42.22,-22.33,;42.22,-20.79,;43.46,-19.89,;44.93,-20.37,;42.99,-18.42,;41.45,-18.42,;40.97,-19.89,;39.65,-20.66,;39.65,-22.21,;38.32,-22.98,;36.99,-22.21,;36.98,-20.68,;38.3,-19.9,;35.66,-22.98,;34.33,-22.22,;33,-22.99,;33,-24.54,;34.33,-25.31,;35.67,-24.53,)|
CCCc1ccccc1-n1c(C)nnc1-c1ccc(cc1)-c1ccccc1 |(4.16,-33.08,;2.83,-33.85,;1.49,-33.08,;.16,-33.86,;.16,-35.39,;-1.18,-36.17,;-2.51,-35.4,;-2.51,-33.86,;-1.17,-33.09,;-1.17,-31.56,;.08,-30.65,;1.54,-31.13,;-.39,-29.19,;-1.93,-29.19,;-2.41,-30.65,;-3.73,-31.43,;-3.73,-32.97,;-5.06,-33.74,;-6.4,-32.98,;-6.41,-31.44,;-5.08,-30.66,;-7.72,-33.75,;-9.06,-32.98,;-10.39,-33.76,;-10.39,-35.3,;-9.05,-36.07,;-7.72,-35.3,)|
CC(C)c1ccccc1-n1c(C)nnc1-c1ccc(cc1)-c1ccccc1 |(17.79,-33.51,;16.46,-32.74,;16.46,-31.2,;15.12,-33.51,;15.13,-35.05,;13.79,-35.83,;12.46,-35.05,;12.46,-33.51,;13.8,-32.75,;13.8,-31.22,;15.04,-30.31,;16.51,-29.92,;14.57,-28.85,;13.03,-28.85,;12.55,-30.31,;11.23,-31.09,;11.23,-32.63,;9.9,-33.4,;8.57,-32.63,;8.56,-31.1,;9.88,-30.32,;7.24,-33.41,;5.91,-32.64,;4.58,-33.41,;4.58,-34.96,;5.91,-35.73,;7.25,-34.96,)|
Cc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1ccccc1-c1ccccc1 |(4.25,2.26,;2.72,2.42,;1.95,3.76,;.44,3.44,;.28,1.91,;-1.05,1.14,;-1.06,-.4,;-2.39,-1.17,;-3.73,-.39,;-3.72,1.14,;-2.39,1.91,;-5.06,-1.16,;-6.39,-.38,;-7.72,-1.15,;-7.74,-2.69,;-6.41,-3.47,;-5.07,-2.71,;1.69,1.28,;2.1,-.68,;.79,-1.49,;.84,-3.03,;2.2,-3.76,;3.51,-2.93,;3.46,-1.4,;4.88,-.82,;6.1,-1.77,;7.52,-1.19,;7.74,.33,;6.51,1.28,;5.09,.7,)|
Cc1nnc(-c2ccccc2)n1-c1ccccc1F |(29.99,-5.57,;28.52,-5.1,;28.05,-3.63,;26.51,-3.63,;26.03,-5.09,;24.71,-5.87,;24.71,-7.41,;23.38,-8.19,;22.05,-7.42,;22.04,-5.88,;23.36,-5.11,;27.28,-6,;27.28,-7.53,;25.94,-8.3,;25.94,-9.84,;27.27,-10.61,;28.61,-9.84,;28.6,-8.3,;29.94,-7.53,)|
Cc1nnc(-c2ccc(cc2)C2CCCCC2)n1-c1ccccc1F |(1.61,-13.73,;.14,-13.26,;-.33,-11.79,;-1.87,-11.79,;-2.35,-13.25,;-3.67,-14.03,;-3.67,-15.57,;-5,-16.35,;-6.33,-15.58,;-6.34,-14.04,;-5.02,-13.27,;-7.66,-16.36,;-9,-15.59,;-10.31,-16.36,;-10.33,-17.9,;-8.99,-18.67,;-7.66,-17.9,;-1.11,-14.16,;-1.11,-15.69,;-2.44,-16.46,;-2.45,-18,;-1.11,-18.77,;.23,-17.99,;.22,-16.46,;1.56,-15.69,)|
Cc1nnc(-c2ccccc2-c2ccccc2)n1-c1ccccc1F |(13.67,-15.2,;12.21,-14.72,;11.73,-13.25,;10.19,-13.25,;9.71,-14.72,;8.39,-15.49,;8.4,-17.04,;7.07,-17.81,;5.73,-17.04,;5.72,-15.51,;7.05,-14.73,;7.03,-13.2,;8.36,-12.42,;8.35,-10.88,;7.01,-10.12,;5.68,-10.9,;5.7,-12.44,;10.96,-15.62,;10.96,-17.15,;9.62,-17.92,;9.62,-19.46,;10.95,-20.23,;12.29,-19.46,;12.29,-17.92,;13.62,-17.15,)|
Cc1nnc(-c2cccc(c2)-c2ccccc2)n1-c1ccccc1F |(25.33,-14.03,;23.87,-13.55,;23.39,-12.09,;21.85,-12.09,;21.37,-13.55,;20.05,-14.33,;20.06,-15.87,;18.73,-16.64,;17.39,-15.87,;17.38,-14.34,;18.71,-13.56,;16.05,-13.59,;16.04,-12.04,;14.7,-11.28,;13.37,-12.06,;13.39,-13.61,;14.73,-14.36,;22.62,-14.46,;22.62,-15.99,;21.28,-16.76,;21.28,-18.29,;22.61,-19.07,;23.95,-18.29,;23.95,-16.76,;25.28,-15.98,)|
CCS(=O)(=O)N1CCC(CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1
Clc1ccc(C(=O)NC[C@]2(CC3CC3)CC[C@@H](CC2)S(=O)(=O)c2cnn[nH]2)c(Cl)c1 |r,wU:9.8,16.20,wD:9.9,(23.01,-13.12,;21.69,-12.33,;20.34,-13.08,;19.02,-12.29,;19.05,-10.76,;17.73,-9.97,;17.75,-8.43,;16.38,-10.72,;15.01,-10.03,;13.72,-10.87,;12.65,-9.74,;11.15,-10.09,;9.68,-9.65,;10.03,-11.15,;12.39,-11.64,;12.39,-13.18,;13.72,-13.95,;15.05,-13.18,;15.05,-11.64,;13.72,-15.49,;12.17,-15.48,;12.93,-16.82,;14.89,-16.47,;16.34,-15.96,;17.28,-17.18,;16.4,-18.45,;14.93,-18.01,;20.38,-10,;20.39,-8.46,;21.71,-10.78,)|
Clc1ccc(C(=O)NC[C@@]2(CC3CC3)CC[C@@H](CC2)S(=O)(=O)c2cnn[nH]2)c(Cl)c1 |r,wU:9.9,16.20,wD:9.8,(38.69,-13.12,;37.37,-12.33,;36.02,-13.08,;34.7,-12.29,;34.73,-10.76,;33.41,-9.97,;33.43,-8.43,;32.06,-10.72,;30.69,-10.03,;29.4,-10.87,;28.33,-9.74,;26.83,-10.09,;25.36,-9.65,;25.71,-11.15,;28.07,-11.64,;28.07,-13.18,;29.4,-13.95,;30.73,-13.18,;30.73,-11.64,;29.4,-15.49,;27.85,-15.48,;28.61,-16.82,;30.57,-16.47,;32.02,-15.96,;32.96,-17.18,;32.08,-18.45,;30.61,-18.01,;36.06,-10,;36.07,-8.46,;37.39,-10.78,)|
Cc1cc(no1)S(=O)(=O)[C@H]1CC[C@](CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1 |r,wU:9.9,12.13,wD:12.26,(-1.11,-33.46,;-1.63,-32.01,;-3.1,-31.57,;-3.13,-30.04,;-1.69,-29.53,;-.75,-30.75,;-4.31,-29.05,;-5.86,-29.04,;-5.09,-30.38,;-4.31,-27.51,;-5.64,-26.75,;-5.64,-25.21,;-4.31,-24.43,;-3.02,-23.59,;-1.65,-24.29,;-.3,-23.54,;-.28,-22,;1.02,-24.32,;.99,-25.86,;2.31,-26.65,;3.66,-25.89,;4.98,-26.68,;3.68,-24.35,;2.35,-23.57,;2.37,-22.03,;-5.38,-23.3,;-6.88,-23.66,;-8.35,-23.21,;-8,-24.71,;-2.98,-25.21,;-2.98,-26.75,)|
Cc1cc(no1)S(=O)(=O)[C@H]1CC[C@@](CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1 |r,wU:12.26,9.9,wD:12.13,(16.36,-33.1,;15.85,-31.65,;14.38,-31.21,;14.34,-29.67,;15.79,-29.16,;16.73,-30.38,;13.17,-28.69,;11.62,-28.68,;12.38,-30.02,;13.17,-27.15,;11.84,-26.38,;11.84,-24.84,;13.17,-24.07,;14.46,-23.23,;15.83,-23.93,;17.18,-23.17,;17.2,-21.63,;18.5,-23.96,;18.47,-25.5,;19.79,-26.28,;21.14,-25.53,;22.46,-26.32,;21.16,-23.98,;19.83,-23.2,;19.84,-21.66,;12.1,-22.94,;10.6,-23.29,;9.12,-22.85,;9.48,-24.35,;14.5,-24.84,;14.5,-26.38,)|
Cc1nnc(s1)S(=O)(=O)[C@H]1CC[C@@](CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1 |r,wU:12.26,9.9,wD:12.13,(-.13,-47.31,;-.64,-45.86,;.24,-44.59,;-.7,-43.37,;-2.15,-43.88,;-2.11,-45.42,;-3.32,-42.9,;-4.87,-42.89,;-4.11,-44.23,;-3.32,-41.36,;-4.65,-40.6,;-4.65,-39.06,;-3.32,-38.28,;-2.03,-37.44,;-.66,-38.14,;.69,-37.38,;.71,-35.84,;2.01,-38.17,;1.98,-39.71,;3.3,-40.49,;4.65,-39.74,;5.97,-40.53,;4.66,-38.19,;3.34,-37.41,;3.35,-35.87,;-4.39,-37.15,;-5.89,-37.5,;-7.37,-37.06,;-7.01,-38.56,;-1.99,-39.06,;-1.99,-40.6,)|
Cc1ccc(nn1)S(=O)(=O)[C@H]1CC[C@@](CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1 |r,wU:13.27,10.10,wD:13.14,(19.25,-45.27,;17.95,-44.45,;16.59,-45.15,;15.3,-44.33,;15.37,-42.79,;16.72,-42.09,;18.02,-42.9,;14.08,-41.97,;12.53,-41.96,;13.29,-43.3,;14.08,-40.43,;12.75,-39.66,;12.75,-38.12,;14.08,-37.34,;15.37,-36.51,;16.74,-37.2,;18.09,-36.45,;18.11,-34.91,;19.41,-37.24,;19.38,-38.77,;20.7,-39.56,;22.05,-38.81,;23.37,-39.6,;22.07,-37.26,;20.74,-36.48,;20.75,-34.94,;13.01,-36.21,;11.51,-36.57,;10.03,-36.13,;10.39,-37.63,;15.41,-38.12,;15.41,-39.66,)|
CCCS(=O)(=O)[C@H]1CC[C@](CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1 |r,wU:9.9,6.5,wD:9.22,(.37,-2.47,;-.93,-1.64,;-2.29,-2.35,;-3.59,-1.53,;-5.13,-1.52,;-4.37,-2.85,;-3.59,.02,;-4.92,.78,;-4.92,2.32,;-3.59,3.1,;-2.3,3.93,;-.92,3.24,;.42,3.99,;.44,5.53,;1.74,3.2,;1.72,1.67,;3.04,.88,;4.38,1.63,;5.71,.85,;4.4,3.18,;3.08,3.96,;3.09,5.5,;-4.66,4.23,;-6.15,3.87,;-7.63,4.31,;-7.27,2.81,;-2.26,2.32,;-2.26,.78,)|
CCS(=O)(=O)[C@H]1CC[C@](CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1 |r,wU:8.8,5.4,wD:8.21,(19.78,-2.92,;18.41,-3.63,;17.12,-2.8,;15.57,-2.79,;16.33,-4.13,;17.12,-1.26,;15.79,-.5,;15.79,1.04,;17.12,1.82,;18.41,2.66,;19.78,1.96,;21.13,2.71,;21.15,4.25,;22.45,1.93,;22.42,.39,;23.74,-.4,;25.09,.36,;26.41,-.43,;25.1,1.9,;23.78,2.68,;23.79,4.22,;16.05,2.95,;14.55,2.59,;13.07,3.04,;13.43,1.54,;18.45,1.04,;18.45,-.5,)|
CS(=O)(=O)[C@H]1CC[C@](CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1 |r,wU:7.7,4.3,wD:7.20,(-1.38,-15.19,;-2.67,-14.37,;-4.22,-14.36,;-3.45,-15.7,;-2.67,-12.83,;-4,-12.06,;-4,-10.52,;-2.67,-9.75,;-1.38,-8.91,;-.01,-9.6,;1.34,-8.85,;1.36,-7.31,;2.66,-9.64,;2.63,-11.17,;3.96,-11.96,;5.3,-11.21,;6.63,-12,;5.32,-9.66,;3.99,-8.88,;4.01,-7.34,;-3.74,-8.62,;-5.24,-8.97,;-6.71,-8.53,;-6.36,-10.03,;-1.34,-10.52,;-1.34,-12.06,)|
CCCS(=O)(=O)[C@H]1CC[C@@](CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1 |r,wU:9.22,6.5,wD:9.9,(19.26,-16.28,;17.96,-15.45,;16.59,-16.16,;15.3,-15.34,;13.75,-15.33,;14.51,-16.67,;15.3,-13.8,;13.97,-13.04,;13.97,-11.5,;15.3,-10.72,;16.59,-9.88,;17.96,-10.58,;19.31,-9.83,;19.33,-8.29,;20.63,-10.61,;20.6,-12.15,;21.92,-12.94,;23.27,-12.18,;24.59,-12.97,;23.29,-10.63,;21.96,-9.85,;21.97,-8.31,;14.23,-9.59,;12.73,-9.95,;11.26,-9.5,;11.61,-11,;16.63,-11.5,;16.63,-13.04,)|
CCS(=O)(=O)[C@H]1CC[C@@](CNC(=O)c2ccc(Cl)cc2Cl)(CC2CC2)CC1 |r,wU:8.21,5.4,wD:8.8,(35.66,-14.4,;34.29,-15.11,;33,-14.28,;31.45,-14.27,;32.22,-15.61,;33,-12.74,;31.67,-11.98,;31.67,-10.44,;33,-9.66,;34.29,-8.82,;35.66,-9.52,;37.01,-8.77,;37.03,-7.23,;38.33,-9.55,;38.3,-11.09,;39.62,-11.88,;40.97,-11.12,;42.29,-11.91,;40.99,-9.58,;39.66,-8.8,;39.68,-7.26,;31.93,-8.53,;30.43,-8.89,;28.96,-8.44,;29.31,-9.94,;34.33,-10.44,;34.33,-11.98,)|
Clc1ccc(C(=O)NC[C@]2(CC3CC3)CC[C@@H](CC2)S(=O)(=O)CC2CCC2)c(Cl)c1 |r,wU:9.8,16.20,wD:9.9,(5.66,-27.32,;4.34,-26.53,;2.99,-27.28,;1.67,-26.5,;1.7,-24.96,;.37,-24.17,;.39,-22.63,;-.97,-24.93,;-2.34,-24.23,;-3.63,-25.07,;-4.7,-23.94,;-6.2,-24.29,;-7.68,-23.85,;-7.32,-25.35,;-4.96,-25.85,;-4.96,-27.39,;-3.63,-28.15,;-2.3,-27.39,;-2.3,-25.85,;-3.63,-29.69,;-5.18,-29.68,;-4.42,-31.02,;-2.34,-30.51,;-1.01,-29.74,;.47,-30.14,;.87,-28.65,;-.62,-28.25,;3.03,-24.2,;3.04,-22.66,;4.35,-24.98,)|
Clc1ccc(C(=O)NC[C@]2(CC3CC3)CC[C@@H](CC2)S(=O)(=O)CC2CC2)c(Cl)c1 |r,wU:9.8,16.20,wD:9.9,(24.58,-27.06,;23.25,-26.28,;21.91,-27.03,;20.59,-26.24,;20.61,-24.71,;19.29,-23.92,;19.31,-22.38,;17.95,-24.67,;16.57,-23.97,;15.28,-24.81,;14.21,-23.68,;12.72,-24.04,;11.24,-23.6,;11.6,-25.09,;13.95,-25.59,;13.95,-27.13,;15.28,-27.89,;16.61,-27.13,;16.61,-25.59,;15.28,-29.43,;13.74,-29.42,;14.5,-30.76,;16.58,-30.26,;17.94,-29.55,;19.47,-29.61,;18.76,-28.24,;21.95,-23.95,;21.96,-22.41,;23.27,-24.73,)|
CN(CCCC([O-])=O)CCC(Oc1ccc(cc1)C(F)(F)F)c1ccccc1
CN(CCC(Oc1ccc(cc1)S(C)(=O)=O)c1ccccc1)CC([O-])=O
C[C@H](Oc1ccc(cc1C(=O)N1CCN(CC1)c1ncc(cc1F)C(F)(F)F)S(C)(=O)=O)C(C)(C)C |r|
C[C@@H](Oc1ccc(cc1C(=O)N1CCN(CC1)c1ncc(cc1F)C(F)(F)F)S(C)(=O)=O)C(C)(C)C |r|
CC(C)CN(CC(=O)Nc1cc(F)cc(F)c1)C(=O)c1ccc(cc1)-c1ccccn1
Fc1cc(F)cc(NC(=O)CN(CC2CC2)C(=O)c2ccc(cc2)-c2ccccn2)c1
Fc1cc(F)cc(NC(=O)CN(C2CCCC2)C(=O)c2ccc(cc2)-c2ccccn2)c1
CC(C)N(CC(=O)Nc1cc(F)cc(F)c1)C(=O)c1ccc(cc1)-c1ccccn1
Fc1cc(F)cc(NC(=O)CN(C2CCOCC2)C(=O)c2ccc(cc2)-c2ccccn2)c1
Fc1cc(F)cc(NC(=O)CN(C2CCOC2)C(=O)c2ccc(cc2)-c2ccccn2)c1
CCC(COC)N(CC(=O)Nc1cc(F)cc(F)c1)C(=O)c1ccc(cc1)-c1ccccn1
COCCN(CC(=O)Nc1cc(F)cc(F)c1)C(=O)c1ccc(cc1)-c1ccccn1
COCC(C)N(CC(=O)Nc1cc(F)cc(F)c1)C(=O)c1ccc(cc1)-c1ccccn1
CCC(C)N(CC(=O)Nc1cc(F)cc(F)c1)C(=O)c1ccc(cc1)-c1ccccn1
COc1ccc(cc1)C(=O)N(Cc1[nH]ncc1-c1ccccc1)C1CCCCC1
Cn1ccc(n1)C(=O)N(CC(=O)Nc1cc(F)cc(F)c1)C1CCCCC1
Fc1cc(F)cc(NC(=O)CN(C2CCCCC2)C(=O)c2cccnc2)c1
CN1CCC(CC1)C(=O)N(CC(=O)Nc1cc(F)cc(F)c1)C1CCCCC1
Fc1cc(F)cc(NC(=O)CN(C2CCCCC2)C(=O)c2ccc(cc2)-c2ccccn2)c1
Fc1cc(F)cc(NC(=O)CN(C2CCCCC2)C(=O)c2ccc(nc2)N2CCCC2)c1
COc1ccc(cc1)C(=O)N(Cc1cc(on1)-c1ccccc1)C1CCCCC1
COc1ccc(cc1)C(=O)N(CC(=O)Nc1cc(F)cc(F)c1)C1CCCCC1
Fc1cc(F)cc(NC(=O)CN(C2CCCCC2)C(=O)c2ccc(cc2)-n2ccnc2)c1
Fc1cc(F)cc(NC(=O)CN(C2CCCCC2)C(=O)c2cccc(Cl)c2)c1
COc1ccc(cc1)C(=O)N(Cc1cn(nn1)-c1ccccc1)C1CCCCC1
Fc1cc(F)cc(NC(=O)CN(C2CCCCC2)C(=O)C2CCOCC2)c1
COc1ccc(cc1)C(=O)N(Cc1c(C)noc1-c1ccccc1)C1CCCCC1
CN(C)CCOc1ccc(cc1)C(=O)N(CC(=O)Nc1cc(F)cc(F)c1)C1CCCCC1
Fc1cc(F)cc(NC(=O)CN(C2CCCCC2)C(=O)c2ccccc2Cl)c1
Fc1cc(F)cc(NC(=O)CN(C2CCCCC2)C(=O)Nc2ccc(Cl)cc2)c1
Fc1cc(F)cc(NC(=O)CN(Cc2ccc(Cl)cc2)C2CCCCC2)c1
CC(N(C1CCCCC1)C(=O)c1ccc(Cl)cc1)C(=O)Nc1cc(F)cc(F)c1
COc1ccc(cc1)C(=O)N(Cc1csc(n1)-c1ccccc1)C1CCCCC1
CC(C)CN(CC(=O)Nc1cc(F)cc(F)c1)C(=O)c1ccc(Cl)cc1
Fc1cc(F)cc(NC(=O)CCN(C2CCCCC2)C(=O)c2ccc(Cl)cc2)c1
Fc1cc(F)cc(NC(=O)CN(C2CCCCC2)C(=O)c2ccc(Cl)cc2)c1
Fc1cc(F)cc(NC(=O)CN(C2CCCOC2)C(=O)c2ccc(cc2)-c2ccccn2)c1
Fc1cc(F)cc(NC(=O)CN(CC2CCC2)C(=O)c2ccc(cc2)-c2ccccn2)c1
Fc1cc(F)cc(NC(=O)CN(C2CCCCC2)C(=O)c2ccc(cc2)N2CCCC2)c1
COc1ccc(cc1)C(=O)N(Cc1ccc(o1)-c1ccc(Cl)cc1)C1CCCCC1
Fc1cc(F)cc(NC(=O)CN(C2CCCCC2)C(=O)C2CCCCC2)c1
COc1ccc(cc1)C(=O)N(Cc1cnc([nH]1)-c1ccccc1)C1CCCCC1
Fc1cc(F)cc(NC(=O)CN(C2CCCCC2)S(=O)(=O)c2ccc(Cl)cc2)c1
CN(CCC(Oc1ccc(cc1)C(F)(F)F)c1ccccc1)CC([O-])=O
CN(CCC(Cc1ccc(cc1)C(F)(F)F)c1ccccc1)CC([O-])=O
CN(CCC(Oc1ccc(Cl)c(Cl)c1)c1ccccc1)CC([O-])=O
CN(CC[C@H](Oc1ccc(cc1)C(F)(F)F)c1ccccc1)CC([O-])=O
COc1ccccc1OC(CCN(C)CC([O-])=O)c1ccccc1
CN(CCC(Oc1ccccc1Cl)c1ccccc1)CC([O-])=O
COc1ccc(cc1)C(CCN(C)CC([O-])=O)Oc1ccc(cc1)C(F)(F)F
CCN(CCC(Oc1ccc(cc1)C(F)(F)F)c1ccccc1)CC([O-])=O
CN(CCC(Oc1ccc(Cl)c(c1)C(F)(F)F)c1ccccc1)CC([O-])=O
CN(CCC(Oc1ccc(cc1)C(F)(F)F)c1ccc(Cl)cc1)CC([O-])=O
CN(CCC(Oc1ccc(cc1)C(F)(F)F)c1ccc(F)cc1)CC([O-])=O
CN(CC[C@H](Oc1ccc(cc1)-c1ccccc1)c1ccccc1)CC([O-])=O
CN(CCC(Oc1ccc(C)cc1)c1ccccc1)CC([O-])=O
CN(CC[C@@H](Oc1ccc(cc1)C(C)(C)C)c1ccccc1)CC([O-])=O
CN(CCC(Oc1ccc(Cl)cc1)c1ccccc1)CC([O-])=O
CN(CCC(Oc1cccc(c1)C(F)(F)F)c1ccccc1)CC([O-])=O
COc1ccc(OC(CCN(C)CC([O-])=O)c2ccccc2)cc1
CN(CC[C@@H](Oc1ccc(cc1)C(F)(F)F)c1ccccc1)CC([O-])=O
CN(CCC(Oc1ccc(cc1)C(F)(F)F)c1ccccc1)CCC([O-])=O
CN(CC[C@H](Oc1ccc(cc1)C(C)(C)C)c1ccccc1)CC([O-])=O
CN(CC[C@@H](Oc1ccc(cc1)-c1ccccc1)c1ccccc1)CC([O-])=O
CCC1CCCCN1C[C@@H](O)CNS(=O)(=O)c1cccc2ccccc12
CC1CCCN1C[C@@H](O)CNS(=O)(=O)c1cccc2ccccc12
CCCN(C[C@@H](O)CNS(=O)(=O)c1cccc2ccccc12)C(C)CC
CC1CCCN1C[C@H](O)CNS(=O)(=O)c1cccc2ccccc12
CC1CCCN(C[C@@H](O)CNS(=O)(=O)c2cccc3ccccc23)C1
CC1CCCCN1C[C@@H](O)CNS(=O)(=O)c1cccc2ccccc12
CCC1CCC(C)N(C[C@@H](O)CNS(=O)(=O)c2cccc3ccccc23)C1
CC1CCC(C)N1C[C@H](O)CNS(=O)(=O)c1cccc2ccccc12
CC1CC(C)N(C[C@@H](O)CNS(=O)(=O)c2cc(Cl)sc2Cl)C1
O[C@@H](CNS(=O)(=O)c1cccc2ccccc12)CN1CCCC1
CC1CCC(C)N1C[C@@H](O)CNS(=O)(=O)c1cccc2ccccc12
CC[C@H]1CCCCN1C[C@@H](O)CNS(=O)(=O)c1cccc2ccccc12
CC1CC(C)N(C[C@@H](O)CNS(=O)(=O)c2cccc(Cl)c2Cl)C1
CCCN(C[C@@H](O)CNS(=O)(=O)c1cccc2ccccc12)C(C)(C)C
CC1CC(C)N(C[C@@H](O)CNS(=O)(=O)c2cc(C)c(Cl)cc2C)C1
O[C@@H](CNS(=O)(=O)c1cccc2ccccc12)CN1CCCCC1
CC1CC(C)N(C[C@@H](O)CNS(=O)(=O)c2ccc3ccccc3c2)C1
CCc1cc(Br)ccc1S(=O)(=O)NC[C@H](O)CN1CC(C)CC1C
CCS(=O)(=O)c1ccc(O[C@@H](C)C(F)(F)F)c(c1)C(=O)N1Cc2cn(nc2C1)-c1ccccc1F |r|
C[C@H](Oc1ccc(cc1C(=O)N1Cc2cn(nc2C1)-c1ccccc1F)S(C)(=O)=O)C(F)(F)F |r|
CS(=O)(=O)c1ccc(N2CCC(F)(F)CC2)c(c1)C(=O)N1Cc2cn(nc2C1)-c1ccccc1F
Cc1cc(ccn1)-n1cc2CN(Cc2n1)C(=O)c1cc(ccc1OCC1CC1)C#N
CC(C)Oc1ccc(cc1C(=O)N1Cc2cn(nc2C1)-c1ccnc(C)c1)C#N
CC(C)S(=O)(=O)c1ccc(O[C@@H](C)C(F)(F)F)c(c1)C(=O)N1Cc2cn(nc2C1)-c1ccccc1 |r|
CCS(=O)(=O)c1ccc(O[C@@H](C)C(F)(F)F)c(c1)C(=O)N1Cc2cn(nc2C1)-c1ccnc(C)c1 |r|
CS(=O)(=O)c1ccc(-c2cccc(F)c2)c(c1)C(=O)N1Cc2cn(nc2C1)-c1cncc(F)c1
CS(=O)(=O)c1ccc(-c2cccc(F)c2)c(c1)C(=O)N1Cc2cn(nc2C1)-c1ccccc1F
CS(=O)(=O)c1ccc(N2CCC(F)(F)CC2)c(c1)C(=O)N1Cc2cn(nc2C1)-c1cncc(F)c1
CS(=O)(=O)c1ccc(OCC2CC2)c(c1)C(=O)N1Cc2cn(nc2C1)-c1ccccc1F
CC(C)(C)Oc1ccc(cc1C(=O)N1Cc2cn(nc2C1)-c1ccccc1F)S(C)(=O)=O
C[C@H](Oc1ccc(cc1C(=O)N1Cc2cn(nc2C1)-c1ccnc(C)c1)S(C)(=O)=O)C(F)(F)F |r|
C[C@H](Oc1ccc(cc1C(=O)N1Cc2cn(nc2C1)-c1cncc(F)c1)S(C)(=O)=O)C(F)(F)F |r|
C[C@H](Oc1ccc(cc1C(=O)N1Cc2cn(nc2C1)-c1cccc(C)c1)S(C)(=O)=O)C(F)(F)F |r|
CC(C)Oc1ccc(cc1C(=O)N1Cc2cn(nc2C1)-c1ccccc1F)S(C)(=O)=O
CCS(=O)(=O)c1ccc(O[C@@H](C)C(F)(F)F)c(c1)C(=O)N1Cc2cn(nc2C1)-c1cncc(F)c1 |r|
C[C@H](Oc1ccc(cc1C(=O)N1Cc2cn(nc2C1)-c1ccccc1)S(C)(=O)=O)C(F)(F)F |r|
Cc1cc(ccn1)-n1cc2CN(Cc2n1)C(=O)c1cc(ccc1-c1cccc(F)c1)C#N
Cc1cc(ccn1)-n1cc2CN(Cc2n1)C(=O)c1cc(ccc1N1CCC(F)(F)CC1)C#N
CC(C)Oc1ccc(cc1C(=O)N1Cc2cn(nc2C1)-c1cncc(F)c1)C#N
C[C@H](Oc1ccc(cc1C(=O)N1Cc2cn(nc2C1)-c1ccnc(C)c1)C#N)C(F)(F)F |r|
C[C@H](Oc1ccc(cc1C(=O)N1Cc2cn(nc2C1)-c1cncc(F)c1)C#N)C(F)(F)F |r|
Fc1cccc(c1)-c1ccc(cc1C(=O)N1Cc2cn(nc2C1)-c1cncc(F)c1)C#N
C[C@H](Oc1ccc(cc1C(=O)N1Cc2cn(nc2C1)C1CCCC1)C#N)C(F)(F)F |r|
Cc1cc(ccn1)-n1cc2CN(Cc2n1)C(=O)c1cc(ccc1-c1cccc(F)c1)S(C)(=O)=O
Cc1cc(ccn1)-n1cc2CN(Cc2n1)C(=O)c1cc(ccc1N1CCC(F)(F)CC1)S(C)(=O)=O
C[C@H](Oc1ccc(cc1C(=O)N1Cc2cn(nc2C1)C1CCCC1)S(C)(=O)=O)C(F)(F)F |r|
C[C@H](Oc1ccc(cc1C(=O)N1Cc2cn(nc2C1)-c1ccccc1F)C#N)C(F)(F)F |r|
CC(C)Oc1ccc(cc1C(=O)N1Cc2cn(nc2C1)-c1ccccc1)C#N
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(F)cccc2F)CCC(F)(F)CC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(F)cccc2F)CCCOCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(N)cccc2Cl)CCN(C)CC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(Cl)cc2Cl)CCOCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(F)cccc2F)CCC2(CC2)CC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(F)cccc2F)C[C@@H]2C[C@@H]2C1 |r|
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(Cl)cc2Cl)CCc2ccccc12
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(N)cccc2Cl)Cc2ccccc2C1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(N)cccc2Cl)CCCCCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(N)cccc2Cl)CCCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(OC)cc(F)cc2SC)CCCCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(OC)cc(cc2C(F)(F)F)C(F)(F)F)CCCCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(Cl)cccc2Cl)CCCCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(F)cccc2F)CCCCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(Cl)c(Cl)c2)CCCCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(F)cc2C)CCCCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(Cl)cc2Cl)CCCCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(OC)cc2F)CCCCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2cccc(c2Cl)C(F)(F)F)CCCCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2cccc(OC(F)(F)F)c2)CCCCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(OC(F)(F)F)cc2)CCCCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(Cl)cc2)CCCCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccccc2OC(F)(F)F)CCCCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccccc2C(F)(F)F)CCCCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccccc2)CCCCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(N)cccc2Cl)CCCCC1
CCCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(N)cccc2Cl)CCC1
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc(C#N)c1C |(17.02,-34.76,;15.75,-35.63,;14.36,-34.96,;13.88,-33.5,;12.34,-33.5,;11.87,-34.97,;10.54,-35.73,;9.21,-34.95,;7.88,-35.71,;7.86,-37.25,;9.2,-38.03,;10.53,-37.26,;6.53,-38.01,;5.2,-37.23,;3.86,-37.99,;3.85,-39.53,;5.19,-40.31,;6.52,-39.54,;13.12,-35.87,;13.12,-37.41,;11.8,-38.18,;11.79,-39.73,;13.13,-40.5,;14.47,-39.72,;15.8,-40.49,;17.13,-41.26,;14.46,-38.17,;15.79,-37.4,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc(c1C)C(F)(F)F |(39.06,-21.58,;37.79,-22.45,;36.4,-21.78,;35.92,-20.32,;34.38,-20.32,;33.91,-21.79,;32.58,-22.55,;31.25,-21.76,;29.91,-22.52,;29.9,-24.07,;31.24,-24.84,;32.57,-24.08,;28.57,-24.83,;27.24,-24.05,;25.9,-24.81,;25.89,-26.35,;27.23,-27.13,;28.56,-26.36,;35.16,-22.69,;35.16,-24.23,;33.83,-25,;33.83,-26.54,;35.16,-27.31,;36.5,-26.54,;36.5,-24.99,;37.83,-24.22,;37.84,-27.31,;37.84,-28.85,;39.17,-26.54,;39.16,-28.08,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc(C(N)=O)c1C |(17.34,-20.97,;16.07,-21.84,;14.68,-21.17,;14.2,-19.71,;12.66,-19.71,;12.19,-21.18,;10.86,-21.94,;9.53,-21.16,;8.19,-21.92,;8.18,-23.46,;9.52,-24.24,;10.85,-23.47,;6.85,-24.22,;5.52,-23.44,;4.18,-24.2,;4.17,-25.74,;5.51,-26.52,;6.84,-25.75,;13.44,-22.08,;13.44,-23.62,;12.12,-24.39,;12.11,-25.94,;13.45,-26.71,;14.78,-25.93,;16.12,-26.7,;16.12,-28.24,;17.45,-25.93,;14.78,-24.38,;16.11,-23.61,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc(C(=O)OC)c1C |(42.08,-6.94,;40.81,-7.81,;39.43,-7.14,;38.94,-5.68,;37.41,-5.68,;36.93,-7.15,;35.6,-7.91,;34.27,-7.13,;32.94,-7.89,;32.93,-9.43,;34.26,-10.21,;35.6,-9.44,;31.59,-10.19,;30.26,-9.41,;28.92,-10.17,;28.91,-11.71,;30.25,-12.49,;31.58,-11.72,;38.18,-8.05,;38.19,-9.59,;36.86,-10.36,;36.85,-11.9,;38.19,-12.68,;39.53,-11.9,;40.86,-12.67,;40.86,-14.21,;42.19,-11.9,;43.53,-12.67,;39.52,-10.35,;40.85,-9.58,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc(Br)c1C |(20.35,-7.11,;19.08,-7.98,;17.69,-7.31,;17.21,-5.85,;15.67,-5.85,;15.2,-7.32,;13.87,-8.08,;12.54,-7.3,;11.2,-8.06,;11.19,-9.6,;12.53,-10.38,;13.86,-9.61,;9.86,-10.36,;8.53,-9.58,;7.19,-10.34,;7.18,-11.88,;8.52,-12.66,;9.85,-11.89,;16.45,-8.22,;16.45,-9.76,;15.13,-10.53,;15.12,-12.08,;16.46,-12.85,;17.79,-12.07,;19.13,-12.84,;17.79,-10.52,;19.12,-9.75,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc(Cl)c1C |(49.15,-50.86,;47.88,-51.73,;46.49,-51.06,;46.01,-49.6,;44.47,-49.6,;43.99,-51.07,;42.66,-51.83,;41.34,-51.05,;40,-51.81,;39.99,-53.35,;41.32,-54.13,;42.66,-53.36,;38.65,-54.11,;37.32,-53.33,;35.98,-54.09,;35.98,-55.63,;37.31,-56.41,;38.65,-55.64,;45.24,-51.97,;45.25,-53.51,;43.92,-54.28,;43.92,-55.83,;45.25,-56.6,;46.59,-55.82,;47.92,-56.59,;46.58,-54.27,;47.91,-53.5,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc(F)c1C |(33.17,-50.76,;31.9,-51.63,;30.52,-50.96,;30.04,-49.5,;28.5,-49.51,;28.02,-50.97,;26.69,-51.73,;25.37,-50.95,;24.03,-51.71,;24.02,-53.25,;25.35,-54.03,;26.69,-53.26,;22.68,-54.01,;21.35,-53.23,;20.02,-53.99,;20.01,-55.53,;21.34,-56.31,;22.68,-55.54,;29.27,-51.87,;29.28,-53.41,;27.95,-54.18,;27.95,-55.73,;29.28,-56.5,;30.62,-55.73,;31.95,-56.49,;30.61,-54.18,;31.94,-53.4,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc(CN(C)C)c1C |(14.7,-48.85,;13.43,-49.72,;12.04,-49.06,;11.56,-47.59,;10.02,-47.6,;9.55,-49.06,;8.22,-49.82,;6.89,-49.04,;5.55,-49.8,;5.54,-51.34,;6.88,-52.12,;8.21,-51.36,;4.2,-52.1,;2.87,-51.32,;1.54,-52.08,;1.53,-53.62,;2.87,-54.4,;4.2,-53.63,;10.8,-49.96,;10.8,-51.5,;9.47,-52.27,;9.47,-53.82,;10.8,-54.59,;12.14,-53.82,;13.47,-54.59,;13.48,-56.13,;14.81,-56.89,;12.14,-56.9,;12.13,-52.27,;13.47,-51.49,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc(COC)c1C |(33.47,-40.28,;32.2,-41.15,;30.81,-40.48,;30.33,-39.02,;28.79,-39.02,;28.32,-40.49,;26.99,-41.25,;25.66,-40.47,;24.32,-41.23,;24.31,-42.77,;25.65,-43.55,;26.98,-42.78,;22.98,-43.53,;21.65,-42.75,;20.31,-43.51,;20.3,-45.05,;21.64,-45.83,;22.97,-45.06,;29.57,-41.39,;29.57,-42.93,;28.24,-43.7,;28.24,-45.24,;29.58,-46.02,;30.91,-45.24,;32.25,-46.01,;32.25,-47.55,;33.59,-48.32,;30.91,-43.69,;32.24,-42.92,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc(CO)c1C |(14.92,-39.34,;13.65,-40.21,;12.26,-39.55,;11.78,-38.08,;10.24,-38.09,;9.77,-39.55,;8.44,-40.31,;7.11,-39.53,;5.78,-40.29,;5.76,-41.83,;7.1,-42.61,;8.44,-41.85,;4.43,-42.59,;3.1,-41.81,;1.76,-42.57,;1.75,-44.11,;3.09,-44.89,;4.42,-44.13,;11.02,-40.45,;11.03,-41.99,;9.7,-42.76,;9.69,-44.31,;11.03,-45.08,;12.37,-44.31,;13.7,-45.08,;13.7,-46.62,;12.36,-42.76,;13.69,-41.98,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc(O)c1C |(34.05,-28.9,;32.78,-29.77,;31.39,-29.11,;30.91,-27.64,;29.37,-27.65,;28.9,-29.11,;27.57,-29.87,;26.24,-29.09,;24.9,-29.85,;24.89,-31.39,;26.23,-32.17,;27.56,-31.41,;23.56,-32.15,;22.23,-31.37,;20.89,-32.13,;20.88,-33.67,;22.22,-34.45,;23.55,-33.69,;30.15,-30.01,;30.15,-31.55,;28.82,-32.32,;28.82,-33.87,;30.15,-34.64,;31.49,-33.87,;32.83,-34.64,;31.49,-32.32,;32.82,-31.54,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc(N(C)C)c1C |(16.04,-28.67,;14.77,-29.54,;13.38,-28.87,;12.9,-27.41,;11.36,-27.41,;10.88,-28.88,;9.55,-29.64,;8.23,-28.86,;6.89,-29.62,;6.88,-31.16,;8.21,-31.94,;9.55,-31.17,;5.54,-31.92,;4.21,-31.14,;2.88,-31.9,;2.87,-33.44,;4.2,-34.22,;5.54,-33.45,;12.13,-29.78,;12.14,-31.32,;10.81,-32.09,;10.81,-33.64,;12.14,-34.41,;13.48,-33.63,;14.81,-34.4,;14.82,-35.94,;16.15,-33.63,;13.47,-32.08,;14.8,-31.31,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc(N)c1C |(37.67,-16.43,;36.4,-17.3,;35.01,-16.63,;34.53,-15.17,;32.99,-15.17,;32.52,-16.64,;31.19,-17.4,;29.86,-16.61,;28.53,-17.37,;28.51,-18.92,;29.85,-19.69,;31.18,-18.93,;27.18,-19.68,;25.85,-18.9,;24.51,-19.66,;24.5,-21.2,;25.84,-21.98,;27.17,-21.21,;33.77,-17.54,;33.77,-19.08,;32.45,-19.85,;32.44,-21.39,;33.78,-22.16,;35.12,-21.39,;36.45,-22.16,;35.11,-19.84,;36.44,-19.07,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc(C)c1C |(17.93,-17.5,;16.66,-18.37,;15.27,-17.7,;14.79,-16.24,;13.25,-16.24,;12.77,-17.71,;11.44,-18.47,;10.12,-17.69,;8.78,-18.45,;8.77,-19.99,;10.1,-20.77,;11.44,-20,;7.43,-20.75,;6.1,-19.97,;4.77,-20.73,;4.76,-22.27,;6.09,-23.05,;7.43,-22.28,;14.02,-18.61,;14.03,-20.15,;12.7,-20.92,;12.7,-22.47,;14.03,-23.24,;15.37,-22.47,;16.7,-23.23,;15.36,-20.92,;16.69,-20.14,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1ccccc1C |(36.18,-5.89,;34.91,-6.76,;33.52,-6.09,;33.04,-4.63,;31.5,-4.63,;31.03,-6.1,;29.7,-6.86,;28.37,-6.08,;27.03,-6.84,;27.02,-8.38,;28.36,-9.16,;29.69,-8.39,;25.69,-9.14,;24.36,-8.36,;23.02,-9.12,;23.01,-10.66,;24.35,-11.44,;25.68,-10.67,;32.28,-7,;32.28,-8.54,;30.95,-9.31,;30.95,-10.85,;32.29,-11.63,;33.62,-10.85,;33.62,-9.3,;34.95,-8.53,)|
CCc1nnc(N2CCN(CC2)c2ccccc2)n1-c1ccccc1F |(36.3,-46.33,;35.01,-47.16,;33.64,-46.45,;33.16,-44.99,;31.62,-44.99,;31.15,-46.46,;29.82,-47.22,;28.49,-46.43,;27.15,-47.19,;27.14,-48.74,;28.48,-49.51,;29.81,-48.75,;25.8,-49.5,;24.47,-48.72,;23.14,-49.48,;23.13,-51.02,;24.47,-51.8,;25.8,-51.03,;32.39,-47.36,;32.4,-48.9,;31.07,-49.67,;31.07,-51.21,;32.4,-51.98,;33.74,-51.21,;33.73,-49.66,;35.06,-48.89,)|
CCc1nnc(N2CCC(CC2)c2ccccc2)n1-c1ccccc1F |(16.82,-45.79,;15.55,-46.66,;14.16,-45.99,;13.68,-44.53,;12.14,-44.53,;11.67,-46,;10.34,-46.76,;9.01,-45.98,;7.67,-46.73,;7.66,-48.28,;9,-49.06,;10.33,-48.29,;6.33,-49.04,;5,-48.26,;3.66,-49.02,;3.65,-50.56,;4.99,-51.34,;6.32,-50.57,;12.92,-46.9,;12.92,-48.44,;11.59,-49.21,;11.59,-50.75,;12.93,-51.52,;14.26,-50.75,;14.26,-49.2,;15.59,-48.43,)|
CCc1nnc(C2CCN(CC2)c2ccccc2)n1-c1ccccc1F |(35.43,-36.51,;34.09,-37.27,;32.76,-36.49,;32.28,-35.03,;30.74,-35.03,;30.27,-36.5,;28.94,-37.26,;27.61,-36.47,;26.27,-37.23,;26.26,-38.78,;27.6,-39.55,;28.93,-38.79,;24.93,-39.54,;23.6,-38.76,;22.26,-39.52,;22.25,-41.06,;23.59,-41.84,;24.92,-41.07,;31.52,-37.4,;31.52,-38.94,;30.19,-39.71,;30.19,-41.25,;31.53,-42.02,;32.86,-41.25,;32.86,-39.7,;34.19,-38.93,)|
CCc1nnc(-c2ccc(cn2)-c2ccccc2)n1-c1ccccc1F |(17.93,-34.77,;16.62,-35.57,;15.27,-34.84,;14.79,-33.37,;13.25,-33.38,;12.77,-34.84,;11.44,-35.6,;10.12,-34.82,;8.78,-35.58,;8.77,-37.12,;10.1,-37.9,;11.44,-37.14,;7.43,-37.88,;6.1,-37.1,;4.76,-37.86,;4.76,-39.41,;6.09,-40.18,;7.43,-39.42,;14.02,-35.75,;14.03,-37.29,;12.7,-38.06,;12.7,-39.6,;14.03,-40.37,;15.37,-39.6,;15.36,-38.05,;16.69,-37.27,)|
CCc1nnc(-c2ccc(nc2)-c2ccccc2)n1-c1ccccc1F |(35.66,-25.77,;34.52,-26.8,;33.06,-26.33,;32.58,-24.87,;31.04,-24.87,;30.56,-26.34,;29.23,-27.1,;27.9,-26.32,;26.57,-27.08,;26.56,-28.62,;27.89,-29.4,;29.23,-28.63,;25.22,-29.38,;23.89,-28.6,;22.55,-29.36,;22.55,-30.9,;23.88,-31.68,;25.22,-30.91,;31.81,-27.24,;31.82,-28.78,;30.49,-29.55,;30.49,-31.09,;31.82,-31.86,;33.16,-31.09,;33.15,-29.54,;34.48,-28.77,)|
Cc1nnc(-c2ccc(cc2)-c2ccccn2)n1-c1ccccc1F |(16.51,-26.63,;15.04,-26.16,;14.56,-24.69,;13.02,-24.7,;12.55,-26.16,;11.22,-26.92,;9.89,-26.14,;8.55,-26.9,;8.54,-28.44,;9.88,-29.22,;11.21,-28.46,;7.21,-29.2,;5.88,-28.42,;4.54,-29.18,;4.53,-30.73,;5.87,-31.5,;7.2,-30.74,;13.8,-27.07,;13.8,-28.6,;12.47,-29.38,;12.47,-30.92,;13.8,-31.69,;15.14,-30.92,;15.14,-29.37,;16.47,-28.59,)|
Cc1nnc(-c2ccc(cc2)-c2cccnc2)n1-c1ccccc1F |(36.24,-15.74,;34.77,-15.27,;34.29,-13.8,;32.75,-13.81,;32.28,-15.27,;30.95,-16.03,;29.62,-15.25,;28.28,-16.01,;28.27,-17.55,;29.61,-18.33,;30.94,-17.57,;26.94,-18.31,;25.61,-17.53,;24.27,-18.3,;24.26,-19.84,;25.6,-20.61,;26.93,-19.85,;33.53,-16.18,;33.53,-17.72,;32.2,-18.49,;32.2,-20.03,;33.54,-20.8,;34.87,-20.03,;34.87,-18.48,;36.2,-17.7,)|
Cc1nnc(-c2ccc(cc2)-c2ccncc2)n1-c1ccccc1F |(16.83,-15.73,;15.36,-15.25,;14.88,-13.79,;13.34,-13.8,;12.87,-15.26,;11.54,-16.02,;10.21,-15.24,;8.87,-16,;8.86,-17.54,;10.2,-18.32,;11.53,-17.55,;7.53,-18.3,;6.2,-17.52,;4.86,-18.28,;4.85,-19.82,;6.19,-20.6,;7.52,-19.83,;14.12,-16.16,;14.12,-17.7,;12.79,-18.47,;12.79,-20.02,;14.12,-20.79,;15.46,-20.02,;15.46,-18.47,;16.79,-17.69,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc(CC#N)c1C |(17.37,-45.76,;16.1,-46.63,;14.71,-45.97,;14.23,-44.5,;12.69,-44.51,;12.22,-45.97,;10.89,-46.73,;9.56,-45.95,;8.23,-46.71,;8.21,-48.25,;9.55,-49.03,;10.88,-48.27,;6.88,-49.01,;5.55,-48.23,;4.21,-48.99,;4.2,-50.54,;5.54,-51.31,;6.87,-50.55,;13.47,-46.88,;13.47,-48.42,;12.15,-49.19,;12.14,-50.73,;13.48,-51.5,;14.82,-50.73,;16.15,-51.49,;16.15,-53.03,;16.16,-54.57,;14.81,-49.18,;16.14,-48.4,)|
CCc1nnc(-c2ccc(cc2)-c2ccccc2)n1-c1cccc(c1C)[N+]([O-])=O |(33.7,-35.11,;32.43,-35.98,;31.05,-35.32,;30.57,-33.85,;29.03,-33.86,;28.55,-35.32,;27.22,-36.08,;25.89,-35.3,;24.56,-36.06,;24.55,-37.6,;25.88,-38.38,;27.22,-37.62,;23.21,-38.36,;21.88,-37.58,;20.54,-38.35,;20.54,-39.89,;21.87,-40.66,;23.21,-39.9,;29.8,-36.23,;29.81,-37.77,;28.48,-38.54,;28.48,-40.08,;29.81,-40.85,;31.15,-40.08,;31.14,-38.53,;32.47,-37.75,;32.48,-40.84,;32.49,-42.38,;33.81,-40.08,)|
O=C1OC[C@H](Cc2ccc3OCOc3c2)[C@H]1Cc1ccc2OCOc2c1 |r|
C(C(=O)O)N
Cn1cnc(c1)S(=O)(=O)N1C[C@H]2[C@@H](C1)[C@]2(CNC(=O)c1ccc(Cl)cc1)CC1CC1 |r|
Cn1cnc(c1)S(=O)(=O)N1C[C@H]2[C@@H](C1)[C@]2(CNC(=O)c1cc(Cl)cc(Cl)c1)CC1CC1 |r|
Cn1cnc(c1)S(=O)(=O)N1C[C@H]2[C@@H](C1)[C@]2(CNC(=O)c1ccc(Cl)c(Cl)c1)CC1CC1 |r|
Cn1cnc(c1)S(=O)(=O)N1C[C@H]2[C@@H](C1)[C@]2(CNC(=O)c1ccccc1Cl)CC1CC1 |r|
Cn1cnc(c1)S(=O)(=O)N1C[C@H]2[C@@H](C1)[C@]2(CNC(=O)c1cccc(c1)C(F)(F)F)CC1CC1 |r|
Cn1cnc(c1)S(=O)(=O)N1C[C@H]2[C@@H](C1)[C@]2(CNC(=O)c1ccccc1C(F)(F)F)CC1CC1 |r|
Cn1cnc(c1)S(=O)(=O)N1C[C@H]2[C@@H](C1)[C@]2(CNC(=O)c1c(Cl)cccc1Cl)CC1CC1 |r|
Cn1cnc(c1)S(=O)(=O)N1C[C@H]2[C@@H](C1)[C@]2(CNC(=O)c1ccc(Cl)cc1Cl)CC1CC1 |r|
Cn1cnc(c1)S(=O)(=O)N1C[C@H]2[C@@H](C1)[C@]2(CNC(=O)c1ccccc1C(F)(F)F)c1ccccn1 |r|
Cn1cnc(c1)S(=O)(=O)N1C[C@H]2[C@@H](C1)[C@]2(CNC(=O)c1ccc(Cl)cc1Cl)c1ccccn1 |r|
Fc1ccccc1S(=O)(=O)N1C[C@H]2[C@@H](C1)[C@]2(CNC(=O)c1ccc(Cl)cc1Cl)CC1CC1 |r|
Clc1ccc(C(=O)NC[C@@]2(CC3CC3)[C@H]3CN(C[C@@H]23)S(=O)(=O)c2ccccc2)c(Cl)c1 |r|
Clc1ccc(C(=O)NC[C@@]2(CC3CC3)[C@H]3CN(C[C@@H]23)S(=O)(=O)c2cccnc2)c(Cl)c1 |r|
Clc1ccc(C(=O)NC[C@@]2(CC3CC3)[C@H]3CN(C[C@@H]23)S(=O)(=O)c2ccccn2)c(Cl)c1 |r|
CC(C)CS(=O)(=O)N1C[C@H]2[C@@H](C1)[C@]2(CNC(=O)c1ccc(Cl)cc1Cl)CC1CC1 |r|
CCCCS(=O)(=O)N1C[C@H]2[C@@H](C1)[C@]2(CNC(=O)c1ccc(Cl)cc1Cl)CC1CC1 |r|
Clc1ccc(C(=O)NC[C@@]2(CC3CC3)[C@H]3CN(C[C@@H]23)S(=O)(=O)CC2CC2)c(Cl)c1 |r|
CC(C)S(=O)(=O)N1C[C@H]2[C@@H](C1)[C@]2(CNC(=O)c1ccc(Cl)cc1Cl)CC1CC1 |r|
CCCS(=O)(=O)N1C[C@H]2[C@@H](C1)[C@]2(CNC(=O)c1ccc(Cl)cc1Cl)CC1CC1 |r|
CCS(=O)(=O)N1C[C@H]2[C@@H](C1)[C@]2(CNC(=O)c1ccc(Cl)cc1Cl)CC1CC1 |r|
CCCS(=O)(=O)N1CCC(CC1)([C@H](C)NC(=O)c1ccc(Cl)cc1Cl)c1ccccc1 |r|
Cn1cnc(c1)S(=O)(=O)N1CC(C1)[C@@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccccn1 |r|
Cn1cnc(c1)S(=O)(=O)N1CC(C1)[C@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccccn1 |r|
Cn1cnc(c1)S(=O)(=O)N1CC2CCC(NC(=O)c3ccccc3Cl)C2C1
Cn1cnc(c1)S(=O)(=O)N1CC2CCC(NC(=O)c3ccccc3C(F)(F)F)C2C1
Cn1cnc(c1)S(=O)(=O)N1CC2CCC(NC(=O)c3cccc(F)c3)C2C1
Clc1ccc(C(=O)NC2CCC3CN(CC23)S(=O)(=O)c2cccs2)c(Cl)c1
Clc1ccc(C(=O)NC2CCC3CN(CC23)S(=O)(=O)c2ccccn2)c(Cl)c1
Clc1ccc(C(=O)NC2CCC3CN(CC23)S(=O)(=O)c2ccccc2)c(Cl)c1
CCCCS(=O)(=O)N1CC2CCC(NC(=O)c3ccc(Cl)cc3Cl)C2C1
CCCS(=O)(=O)N1CC2CCC(NC(=O)c3ccc(Cl)cc3Cl)C2C1
CCS(=O)(=O)N1CC2CCC(NC(=O)c3ccc(Cl)cc3Cl)C2C1
Cn1cnc(c1)S(=O)(=O)N1CC2CCC(NC(=O)c3ccc(F)cc3)C2C1
Cn1cnc(c1)S(=O)(=O)N1CC2CCC(NC(=O)c3ccccc3F)C2C1
Cn1cnc(c1)S(=O)(=O)N1CC2CCC(NC(=O)c3ccc(F)c(F)c3)C2C1
CCCS(=O)(=O)N1CCC(CC1)C(NC(=O)c1ccc(Cl)cc1Cl)c1ccccc1
Cn1cnc(c1)S(=O)(=O)N1CC2CCC(NC(=O)c3ccc(Cl)cc3)C2C1
Cn1cnc(c1)S(=O)(=O)N1CC2CCC(NC(=O)c3ccc(F)cc3F)C2C1
Cn1cnc(c1)S(=O)(=O)N1CC2CCC(NC(=O)c3ccc(Cl)c(Cl)c3)C2C1
Cn1cnc(c1)S(=O)(=O)N1CC2CCC(NC(=O)c3c(F)cccc3F)C2C1
CCCS(=O)(=O)N1CC(C1)C(NC(=O)c1ccc(Cl)cc1Cl)c1ccccc1
Cn1cnc(c1)S(=O)(=O)N1CC2CCC(NC(=O)C3CCCCC3)C2C1
Cn1cnc(c1)S(=O)(=O)N1C[C@H]2CC[C@@H](NC(=O)c3ccc(Cl)cc3Cl)[C@H]2C1 |r|
Cn1cnc(c1)S(=O)(=O)N1CCC(CC1)C(NC(=O)c1ccc(Cl)cc1Cl)c1cccs1
Cn1cnc(c1)S(=O)(=O)N1CCC(CC1)C(NC(=O)c1ccc(Cl)cc1Cl)c1ccccc1
Cn1cnc(c1)S(=O)(=O)N1CC(C1)C(NC(=O)c1ccc(Cl)cc1Cl)c1ccccn1
Cn1cnc(c1)S(=O)(=O)N1CCC(CC1)C(NC(=O)c1ccc(Cl)cc1Cl)c1ccccn1
Cn1cnc(c1)S(=O)(=O)N1CC(C1)C(NC(=O)c1ccc(Cl)cc1Cl)c1cccs1
Cn1cnc(c1)S(=O)(=O)N1CC(C1)C(NC(=O)c1ccc(Cl)cc1Cl)c1ccccc1
Cn1cnc(c1)S(=O)(=O)N1C[C@@H]2CC[C@H](NC(=O)c3ccc(Cl)cc3Cl)[C@@H]2C1 |r|
Cn1cnc(c1)S(=O)(=O)N1CC2CCC(NC(=O)c3ccc(Cl)cc3Cl)C2C1
Cn1cc(nn1)S(=O)(=O)N1CC2CCC(NC(=O)c3ccc(Cl)cc3Cl)C2C1
Cn1cnc(c1)S(=O)(=O)N1C[C@H](Oc2cc(ncn2)C(F)(F)F)[C@H](C1)c1ccc(F)cc1 |r|
Cc1cccc(NC2CN(CC2c2ccccc2)S(=O)(=O)c2cn(C)cn2)c1
Cn1cnc(c1)S(=O)(=O)N1CC(Nc2cccc(Cl)c2)C(C1)c1ccccc1F
Cn1cnc(c1)S(=O)(=O)N1C[C@H](Nc2cccc(OC(F)(F)F)c2)[C@H](C1)C1OCCCCO1 |r|
Cn1cnc(c1)S(=O)(=O)N1CC(Nc2cccc(c2)C(F)(F)F)C(C1)c1ccc(F)cc1
Cn1cc(nn1)S(=O)(=O)N1C[C@H](Nc2ccc(F)c(c2)C(F)(F)F)[C@H](C1)c1ccc(F)cc1
Cn1cnc(c1)S(=O)(=O)N1C[C@H](Cc2ccccc2)[C@H](C1)c1ccccc1 |r|
Cn1cnc(c1)S(=O)(=O)N1CC(NC(=O)c2cccc(c2Cl)C(F)(F)F)C(C1)c1ccccc1
Cn1cnc(c1)S(=O)(=O)N1CC(Nc2cccc(c2)C(F)(F)F)C(C1)c1ccccc1
Cn1cnc(c1)S(=O)(=O)N1CC(Nc2cccc(c2)C(F)(F)F)C(C1)c1cccnc1
Cn1cnc(c1)S(=O)(=O)N1C[C@H](Nc2cc(ccn2)C(F)(F)F)[C@H](C1)c1ccc(F)cc1
Cn1cnc(c1)S(=O)(=O)N1C[C@H](COc2cccc(OC(F)(F)F)c2)[C@H](C1)c1ccc(F)cc1 |r|
[H][C@@]1(CN(C[C@@H]1Nc1cccc(OC(F)(F)F)c1)S(=O)(=O)c1cn(C)cn1)[C@@]1([H])CCCCO1 |r|
Cn1cnc(c1)S(=O)(=O)N1C[C@@H]([C@H](C1)c1ccc(F)cc1)C(=O)Nc1cccc(OC(F)(F)F)c1 |r|
Cn1cnc(c1)S(=O)(=O)N1C[C@@H]([C@H](C1)c1ccc(F)cc1)C(=O)c1cccc(OC(F)(F)F)c1 |r|
Cn1cnc(c1)S(=O)(=O)N1C[C@H](CNc2cccc(OC(F)(F)F)c2)[C@H](C1)c1ccc(F)cc1 |r|
Cn1cnc(c1)S(=O)(=O)N1C[C@H](Nc2cccc(c2)C#N)[C@H](C1)c1ccccc1 |r|
Cn1cnc(c1)S(=O)(=O)N1CC(Nc2ccccc2)C(C1)c1ccccc1
Cc1ccccc1NC1CN(CC1c1ccccc1)S(=O)(=O)c1cn(C)cn1
Cn1cnc(c1)S(=O)(=O)N1CC(Nc2ccc(F)c(c2)C(F)(F)F)C(C1)c1ccc(F)cc1
Cn1cnc(c1)S(=O)(=O)N1CC(Nc2cncc(c2)C(F)(F)F)C(C1)c1ccc(F)cc1
Cn1cnc(c1)S(=O)(=O)N1CC(Nc2cccc(Cl)c2)C(C1)c1cccc(F)c1
Cn1cnc(c1)S(=O)(=O)N1C[C@H](Nc2cccc(c2)C(F)(F)F)[C@H](C1)c1ccc(F)cc1
Cn1cnc(c1)S(=O)(=O)N1C[C@H](Nc2cccc(OC(F)(F)F)c2)[C@H](C1)c1ccc(F)cc1
Cn1cnc(c1)S(=O)(=O)N1C[C@H](Nc2ccc(F)c(OC(F)(F)F)c2)[C@H](C1)c1ccc(F)cc1
[H][C@]1(CCc2ccccc12)N[C@H]1CN(C[C@@H]1c1ccc(F)cc1)S(=O)(=O)c1cn(C)cn1 |r|
Cc1ccc(NC2CN(CC2c2ccccc2)S(=O)(=O)c2cn(C)cn2)cc1
Cn1cnc(c1)S(=O)(=O)N1CC(Nc2ccnc(c2)C(F)(F)F)C(C1)c1ccc(F)cc1
Cn1cnc(c1)S(=O)(=O)N1CC(Nc2cccc(Cl)c2)C(C1)c1ccc(F)cc1
Cn1cnc(c1)S(=O)(=O)N1C[C@H](Nc2cc(ncn2)C(F)(F)F)[C@H](C1)c1ccc(F)cc1
Cn1cnc(c1)S(=O)(=O)N1C[C@H](Nc2cccc(OC(F)(F)F)c2)[C@H](C1)C1OCCCO1 |r|
[H][C@]1(CCCO1)[C@@]1([H])CN(C[C@@H]1Nc1cccc(OC(F)(F)F)c1)S(=O)(=O)c1cn(C)cn1 |r|
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CC[C@@H]([C@H](Cc3ccccc3)c2c1)N1CCCC1 |r|
O=S(=O)(CC1CC1)NC1CN(C1)c1ccc2CC[C@@H]([C@H](Cc3ccccc3)c2c1)N1CCC1 |r|
N[C@H]1CCc2ccc(OCCNS(=O)(=O)C3CCC3)cc2[C@H]1Cc1ccc(Cl)c(Cl)c1 |r|
CCCS(=O)(=O)NCc1ccc2CC[C@H](NC)[C@H](Cc3ccccc3)c2c1 |r|
CCCS(=O)(=O)N[C@@H]1CCN(C1=O)c1ccc2CC[C@@H]([C@H](Cc3ccccc3)c2c1)N1CCC1 |r|
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CC[C@H](N)[C@H](Cc3ccccc3)c2c1 |r|
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CC[C@H](N)[C@H](Cc3cccc(c3)C(F)(F)F)c2c1 |r|
Cn1cnc(c1)S(=O)(=O)NCc1ccc2CC[C@@H]([C@H](Cc3ccccc3)c2c1)N1CCC1 |r|
O=S(=O)(CC1CC1)NCCOc1ccc2OC[C@@H]([C@H](Cc3ccccc3)c2c1)N1CCC1 |r|
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CC[C@H](N)[C@H](Cc3ccc(Cl)cc3)c2c1 |r|
Cn1cc(cn1)S(=O)(=O)NCCOc1ccc2CC[C@H](N)[C@H](Cc3ccc(Cl)c(Cl)c3)c2c1 |r|
CS(=O)(=O)NCCOc1ccc2CC[C@H](N)[C@H](Cc3ccc(Cl)c(Cl)c3)c2c1 |r|
CCCS(=O)(=O)NC1CN(C1)c1ccc2OC[C@@H]([C@H](Cc3ccccc3)c2c1)N1CCC1 |r|
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CC[C@H](N)[C@H](Cc3ccccc3Cl)c2c1 |r|
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CC[C@H](N)[C@H](Cc3cc(F)cc(Cl)c3)c2c1 |r|
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CC[C@@H]([C@H](Cc3ccccc3)c2c1)N1CCC1 |r|
O=S(=O)(CC1CC1)NCCOc1ccc2CC[C@@H]([C@H](Cc3ccccc3)c2c1)N1CCC1 |r|
CN[C@H]1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2[C@H]1Cc1ccccc1 |r|
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2OC[C@@H]([C@H](Cc3ccccc3)c2c1)N1CCC1 |r|
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CC[C@H](NCC(F)(F)F)[C@H](Cc3ccccc3)c2c1 |r|
CCCS(=O)(=O)NCc1ccc2CC[C@@H]([C@H](Cc3ccccc3)c2c1)N1CCC1 |r|
O=S(=O)(CC1CC1)NC1CN(C1)c1ccc2OC[C@@H]([C@H](Cc3ccccc3)c2c1)N1CCC1 |r|
CCCS(=O)(=O)NC1CN(C1)c1ccc2CC[C@@H]([C@H](Cc3ccccc3)c2c1)N1CCC1
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CC[C@H](N)[C@H](Cc3cccc(Cl)c3)c2c1 |r|
N[C@H]1CCc2ccc(OCCNS(=O)(=O)c3ccccc3)cc2[C@H]1Cc1ccc(Cl)c(Cl)c1 |r|
Cn1cnc(c1)S(=O)(=O)NCCOc1ccc2CC[C@H](N)[C@H](Cc3ccc(Cl)c(Cl)c3)c2c1 |r|
N[C@H]1CCc2ccc(OCCNS(=O)(=O)CC3CC3)cc2[C@H]1Cc1ccc(Cl)c(Cl)c1 |r|
CCCCS(=O)(=O)NCCOc1ccc2CC[C@H](N)[C@H](Cc3ccc(Cl)c(Cl)c3)c2c1 |r|
Oc1ccc2CCNC(c2c1)C1(CCC1)c1ccc(Cl)cc1
CCCS(=O)(=O)NCCOc1ccc2CC[C@H](N)[C@H](Cc3ccc(Cl)c(Cl)c3)c2c1 |r|
N[C@H]1CCc2ccc(OCCNS(=O)(=O)c3cccs3)cc2[C@H]1Cc1ccc(Cl)c(Cl)c1 |r|
CNCC(=O)O
COc1ccc2[C@H]([C@@H](CN(C)CC(O)=O)CCc2c1)c1ccccc1 |r|
N[C@@H](COC(c1cccc(F)c1)c1ccccc1OCc1ccccc1)C(O)=O |r|
Cc1cccc(C)c1C(=O)NC(c1ccncc1)C12CCC(CC1)N2
CN1CC2CCC1(CC2)C(NC(=O)c1cccc(c1Cl)C(F)(F)F)c1ccco1 |(20.39,-7.64,;20.39,-6.1,;19.04,-5.33,;19.04,-3.78,;20.39,-2.99,;21.73,-3.78,;21.73,-5.33,;21.12,-4,;20.03,-5.11,;23.07,-6.1,;23.07,-7.63,;24.39,-8.4,;25.7,-7.63,;24.39,-9.92,;23.06,-10.67,;23.06,-12.19,;24.38,-12.96,;25.7,-12.19,;25.7,-10.67,;27.02,-9.91,;27.02,-12.95,;28.34,-13.7,;28.34,-12.18,;27.03,-14.48,;24.4,-5.33,;24.57,-3.8,;26.08,-3.47,;26.85,-4.81,;25.82,-5.96,)|
CN1CC2CCC1(CC2)[C@H](NC(=O)c1ccncc1Br)c1ccccc1 |r,wU:9.11,(29.66,-17.93,;29.66,-16.4,;28.33,-15.65,;28.33,-14.11,;29.66,-13.33,;30.99,-14.11,;30.99,-15.65,;30.39,-14.33,;29.31,-15.42,;32.31,-16.41,;32.31,-17.96,;33.64,-18.73,;34.98,-17.96,;33.64,-20.27,;32.3,-21.04,;32.3,-22.58,;33.64,-23.36,;34.98,-22.58,;34.98,-21.04,;36.3,-20.27,;33.65,-15.64,;34.98,-16.42,;36.32,-15.65,;36.32,-14.1,;34.98,-13.33,;33.64,-14.1,)|
CN1CC2CCC1(CC2)C(NC(=O)c1c(C)cccc1C)c1cccc(c1)-c1cnn(C)c1 |(27.48,-27.58,;27.48,-26.03,;26.13,-25.26,;26.13,-23.69,;27.48,-22.9,;28.83,-23.69,;28.83,-25.26,;28.22,-23.92,;27.12,-25.03,;30.18,-26.03,;30.18,-27.57,;31.51,-28.34,;32.83,-27.57,;31.51,-29.87,;30.17,-30.63,;28.83,-29.84,;30.17,-32.16,;31.5,-32.93,;32.83,-32.16,;32.82,-30.63,;34.17,-29.84,;31.5,-25.26,;31.5,-23.74,;32.82,-22.97,;34.16,-23.74,;34.16,-25.27,;32.83,-26.04,;35.51,-26.04,;35.67,-27.59,;37.19,-27.92,;37.97,-26.57,;39.52,-26.41,;36.93,-25.41,)|
CCN1C2CCC1(CC2)C(NC(=O)c1c(C)cccc1C)c1ccccc1 |TLB:1:2:4.5:7.8|
CN1CC2CCC1(CC2)C(NC(=O)c1cccc(c1Cl)C(F)(F)F)c1cccc(C)c1 |(18.64,-24,;18.64,-22.44,;17.28,-21.67,;17.28,-20.1,;18.64,-19.31,;19.99,-20.1,;19.99,-21.67,;19.38,-20.33,;18.28,-21.44,;21.34,-22.45,;21.34,-23.99,;22.68,-24.76,;24,-23.99,;22.67,-26.3,;21.34,-27.06,;21.33,-28.59,;22.67,-29.37,;24,-28.59,;24,-27.06,;25.33,-26.29,;25.33,-29.35,;26.66,-30.12,;26.67,-28.58,;25.34,-30.9,;22.67,-21.68,;24,-22.46,;25.34,-21.69,;25.34,-20.15,;24,-19.38,;23.99,-17.82,;22.67,-20.15,)|
CN1CC2CCC1(CC2)[C@H](NC(=O)c1c(Cl)cccc1Cl)c1ccccc1 |r,wU:9.11,(15.28,-15.58,;15.28,-14.06,;13.95,-13.3,;13.95,-11.76,;15.28,-10.98,;16.61,-11.76,;16.61,-13.3,;16.01,-11.99,;14.93,-13.08,;17.93,-14.07,;17.93,-15.61,;19.26,-16.38,;20.6,-15.61,;19.26,-17.93,;17.92,-18.69,;16.6,-17.92,;17.92,-20.24,;19.26,-21.01,;20.6,-20.23,;20.6,-18.69,;21.92,-17.92,;19.27,-13.3,;20.6,-14.07,;21.94,-13.3,;21.94,-11.76,;20.6,-10.98,;19.26,-11.76,)|
CN1CC2CCC1(CC2)[C@H](NC(=O)c1ccnc(Cl)c1Cl)c1ccccc1 |r,wU:9.11,(28.99,-44.75,;28.99,-43.22,;27.66,-42.46,;27.66,-40.92,;28.99,-40.15,;30.31,-40.92,;30.31,-42.46,;29.71,-41.15,;28.63,-42.24,;31.63,-43.23,;31.63,-44.77,;32.97,-45.54,;34.31,-44.77,;32.97,-47.09,;31.63,-47.85,;31.63,-49.4,;32.96,-50.17,;34.3,-49.39,;35.64,-50.16,;34.3,-47.85,;35.64,-47.08,;32.97,-42.46,;34.31,-43.23,;35.64,-42.46,;35.65,-40.92,;34.3,-40.14,;32.97,-40.92,)|
Cn1cnc(c1)-c1cscn1
CN1CC2CC1(C2)C(NC(=O)c1c(C)cccc1C)c1ccccc1 |(27.16,-27.5,;27.49,-25.97,;26.44,-24.81,;27.22,-23.46,;28.75,-23.78,;28.91,-25.33,;27.62,-24.96,;30.27,-26.11,;30.27,-27.64,;31.6,-28.42,;32.92,-27.65,;31.6,-29.96,;30.26,-30.71,;28.91,-29.93,;30.26,-32.25,;31.59,-33.03,;32.92,-32.25,;32.92,-30.71,;34.27,-29.93,;31.59,-25.34,;31.59,-23.8,;32.92,-23.04,;34.26,-23.81,;34.26,-25.34,;32.92,-26.11,)|
Cc1cccc(C)c1C(=O)NC(c1ccccc1)C12CCC(CC1)N2
Cc1cccc(C)c1C(=O)NC(c1ccccc1)C12CCC(CC1)N2C1CC1 |TLB:25:24:20.19:23.22|
CN1C2CCC1(CC2)C(NC(=O)c1c(C)cccc1C)c1ccccc1 |TLB:0:1:3.4:6.7|
Cc1cccc(C)c1C(=O)NC(c1ccccc1)C12CCC(CC1)CN2
CN1CC2CCC1(CC2)C(NC(=O)c1c(C)cccc1C)c1ccncc1 |(37.75,-10.82,;37.75,-9.26,;36.4,-8.49,;36.4,-6.92,;37.75,-6.13,;39.1,-6.92,;39.1,-8.49,;38.49,-7.15,;37.39,-8.26,;40.45,-9.27,;40.45,-10.8,;41.78,-11.58,;43.11,-10.81,;41.78,-13.11,;40.45,-13.87,;39.1,-13.08,;40.44,-15.4,;41.78,-16.18,;43.11,-15.4,;43.1,-13.87,;44.45,-13.09,;41.78,-8.5,;41.78,-6.97,;43.1,-6.2,;44.44,-6.97,;44.44,-8.51,;43.11,-9.27,)|
CN1CC2CCC1(CC2)C(NC(=O)c1c(C)cccc1C)c1ccc(C)o1 |(24.77,-10.28,;24.77,-8.72,;23.42,-7.95,;23.42,-6.39,;24.77,-5.59,;26.13,-6.39,;26.13,-7.95,;25.51,-6.61,;24.41,-7.72,;27.48,-8.73,;27.47,-10.26,;28.8,-11.04,;30.13,-10.27,;28.8,-12.57,;27.47,-13.33,;26.12,-12.54,;27.47,-14.86,;28.8,-15.63,;30.13,-14.86,;30.12,-13.33,;31.47,-12.54,;28.8,-7.96,;28.95,-6.44,;30.45,-6.11,;31.22,-7.44,;32.77,-7.6,;30.2,-8.58,)|
CN1CC2CCC1(CC2)C(NC(=O)c1cccc(c1Cl)C(F)(F)F)c1ccccn1 |(31.87,-24.02,;31.87,-22.46,;30.52,-21.68,;30.52,-20.11,;31.87,-19.32,;33.23,-20.11,;33.23,-21.68,;32.62,-20.34,;31.51,-21.46,;34.58,-22.46,;34.58,-24,;35.92,-24.78,;37.24,-24.01,;35.91,-26.32,;34.58,-27.07,;34.57,-28.61,;35.91,-29.39,;37.24,-28.61,;37.24,-27.07,;38.57,-26.3,;38.58,-29.37,;39.91,-30.14,;39.91,-28.59,;38.58,-30.92,;35.91,-21.69,;35.91,-20.16,;37.24,-19.39,;38.58,-20.16,;38.58,-21.7,;37.24,-22.47,)|
COc1ccc(cc1)C(NC(=O)c1cccc(c1Cl)C(F)(F)F)C12CCC(CC1)CN2C
CN1CC2CCC1(CC2)C(NC(=O)c1cccc(c1Cl)C(F)(F)F)c1ccc(C)cc1 |(7.2,-37.44,;7.2,-35.88,;5.85,-35.11,;5.85,-33.54,;7.2,-32.74,;8.56,-33.54,;8.56,-35.11,;7.94,-33.77,;6.84,-34.88,;9.91,-35.89,;9.91,-37.42,;11.24,-38.2,;12.57,-37.43,;11.24,-39.73,;9.9,-40.49,;9.9,-42.03,;11.23,-42.8,;12.56,-42.03,;12.56,-40.49,;13.89,-39.72,;13.9,-42.79,;15.23,-43.55,;15.23,-42.01,;13.9,-44.33,;11.24,-35.11,;11.23,-33.58,;12.56,-32.82,;13.9,-33.58,;15.25,-32.8,;13.9,-35.12,;12.57,-35.89,)|
COc1cccc(c1)C(NC(=O)c1cccc(c1Cl)C(F)(F)F)C12CCC(CC1)CN2C
CN1CC2CCC1(CC2)C(NC(=O)c1cccc(c1Cl)C(F)(F)F)c1ccccc1C |(20.57,-7.71,;20.57,-6.15,;19.22,-5.38,;19.22,-3.81,;20.57,-3.02,;21.93,-3.81,;21.93,-5.38,;21.31,-4.04,;20.21,-5.15,;23.28,-6.16,;23.28,-7.7,;24.61,-8.47,;25.94,-7.7,;24.61,-10.01,;23.27,-10.77,;23.27,-12.3,;24.6,-13.08,;25.93,-12.3,;25.93,-10.77,;27.26,-10,;27.27,-13.06,;28.6,-13.83,;28.6,-12.29,;27.27,-14.61,;24.61,-5.39,;25.94,-6.17,;27.27,-5.4,;27.27,-3.86,;25.93,-3.09,;24.6,-3.86,;23.25,-3.08,)|
COc1ccccc1C(NC(=O)c1cccc(c1Cl)C(F)(F)F)C12CCC(CC1)CN2C
COc1cccc(OC)c1C(=O)N[C@H](c1ccccc1)C12CCC(CC1)CN2C |r|
CN1CC2CCC1(CC2)[C@H](NC(=O)c1c(Cl)cncc1Cl)c1ccccc1 |r,wU:9.11,(15.28,-15.58,;15.28,-14.06,;13.95,-13.3,;13.95,-11.76,;15.28,-10.98,;16.61,-11.76,;16.61,-13.3,;16.01,-11.99,;14.93,-13.08,;17.93,-14.07,;17.93,-15.61,;19.26,-16.38,;20.6,-15.61,;19.26,-17.93,;17.92,-18.69,;16.6,-17.92,;17.92,-20.24,;19.26,-21.01,;20.6,-20.23,;20.6,-18.69,;21.92,-17.92,;19.27,-13.3,;20.6,-14.07,;21.94,-13.3,;21.94,-11.76,;20.6,-10.98,;19.26,-11.76,)|
CN1CC2CCC1(CC2)[C@H](NC(=O)c1c(Cl)ccnc1Cl)c1ccccc1 |r,wU:9.11,(15.28,-15.58,;15.28,-14.06,;13.95,-13.3,;13.95,-11.76,;15.28,-10.98,;16.61,-11.76,;16.61,-13.3,;16.01,-11.99,;14.93,-13.08,;17.93,-14.07,;17.93,-15.61,;19.26,-16.38,;20.6,-15.61,;19.26,-17.93,;17.92,-18.69,;16.6,-17.92,;17.92,-20.24,;19.26,-21.01,;20.6,-20.23,;20.6,-18.69,;21.92,-17.92,;19.27,-13.3,;20.6,-14.07,;21.94,-13.3,;21.94,-11.76,;20.6,-10.98,;19.26,-11.76,)|
CN1CC2CCC1(CC2)[C@H](NC(=O)c1c(C)ccnc1C)c1ccccc1 |r,wU:9.11,(15.28,-15.58,;15.28,-14.06,;13.95,-13.3,;13.95,-11.76,;15.28,-10.98,;16.61,-11.76,;16.61,-13.3,;16.01,-11.99,;14.93,-13.08,;17.93,-14.07,;17.93,-15.61,;19.26,-16.38,;20.6,-15.61,;19.26,-17.93,;17.92,-18.69,;16.6,-17.92,;17.92,-20.24,;19.26,-21.01,;20.6,-20.23,;20.6,-18.69,;21.92,-17.92,;19.27,-13.3,;20.6,-14.07,;21.94,-13.3,;21.94,-11.76,;20.6,-10.98,;19.26,-11.76,)|
CN1CC2CCC1(CC2)[C@H](NC(=O)c1c(C)cccc1C)c1ccccc1 |r,wU:9.11,(15.28,-15.58,;15.28,-14.06,;13.95,-13.3,;13.95,-11.76,;15.28,-10.98,;16.61,-11.76,;16.61,-13.3,;16.01,-11.99,;14.93,-13.08,;17.93,-14.07,;17.93,-15.61,;19.26,-16.38,;20.6,-15.61,;19.26,-17.93,;17.92,-18.69,;16.6,-17.92,;17.92,-20.24,;19.26,-21.01,;20.6,-20.23,;20.6,-18.69,;21.92,-17.92,;19.27,-13.3,;20.6,-14.07,;21.94,-13.3,;21.94,-11.76,;20.6,-10.98,;19.26,-11.76,)|
CN1CC2CCC1(CC2)[C@H](NC(=O)c1cccc(Cl)c1Cl)c1ccccc1 |r,wU:9.11,(28.97,-44.71,;28.97,-43.19,;27.64,-42.43,;27.64,-40.9,;28.97,-40.12,;30.29,-40.9,;30.29,-42.43,;29.69,-41.12,;28.61,-42.21,;31.61,-43.2,;31.61,-44.74,;32.95,-45.51,;34.28,-44.74,;32.94,-47.06,;31.61,-47.82,;31.6,-49.36,;32.94,-50.14,;34.28,-49.36,;35.62,-50.12,;34.28,-47.82,;35.61,-47.04,;32.95,-42.43,;34.28,-43.2,;35.62,-42.43,;35.62,-40.89,;34.28,-40.12,;32.95,-40.89,)|
CN1CC2CCC1(CC2)[C@H](NC(=O)c1cccc(c1Cl)C(F)(F)F)c1ccccc1 |r,wU:9.11,(38.41,-40.07,;38.41,-38.51,;37.06,-37.73,;37.06,-36.17,;38.41,-35.37,;39.77,-36.17,;39.77,-37.73,;39.16,-36.39,;38.05,-37.51,;41.12,-38.51,;41.12,-40.05,;42.45,-40.83,;43.78,-40.06,;42.45,-42.36,;41.11,-43.12,;41.11,-44.66,;42.45,-45.43,;43.78,-44.65,;43.77,-43.12,;45.11,-42.35,;45.11,-45.42,;46.44,-46.18,;46.44,-44.64,;45.12,-46.96,;42.45,-37.74,;42.44,-36.21,;43.77,-35.44,;45.12,-36.21,;45.11,-37.75,;43.78,-38.52,)|
CN1CC2CCC1(CC2)[C@@H](NC(=O)c1cccc(c1Cl)C(F)(F)F)c1ccccc1 |r,wD:9.11,(38.41,-40.07,;38.41,-38.51,;37.06,-37.73,;37.06,-36.17,;38.41,-35.37,;39.77,-36.17,;39.77,-37.73,;39.16,-36.39,;38.05,-37.51,;41.12,-38.51,;41.12,-40.05,;42.45,-40.83,;43.78,-40.06,;42.45,-42.36,;41.11,-43.12,;41.11,-44.66,;42.45,-45.43,;43.78,-44.65,;43.77,-43.12,;45.11,-42.35,;45.11,-45.42,;46.44,-46.18,;46.44,-44.64,;45.12,-46.96,;42.45,-37.74,;42.44,-36.21,;43.77,-35.44,;45.12,-36.21,;45.11,-37.75,;43.78,-38.52,)|
CC(C)N1C2CCC1(CC2)C(NC(=O)c1c(C)cccc1C)c1ccccc1 |TLB:1:3:5.6:8.9|
CN1CC2CCC1(CC2)[C@H](NC(=O)c1c(N)cccc1Cl)c1ccccc1 |r,wU:9.11,(15.37,-15.67,;15.37,-14.14,;14.05,-13.38,;14.05,-11.85,;15.37,-11.06,;16.7,-11.85,;16.7,-13.38,;16.1,-12.07,;15.02,-13.16,;18.02,-14.15,;18.02,-15.69,;19.36,-16.47,;20.69,-15.69,;19.35,-18.01,;18.01,-18.77,;16.69,-18.01,;18.01,-20.32,;19.35,-21.1,;20.69,-20.31,;20.69,-18.77,;22.01,-18.01,;19.36,-13.38,;20.69,-14.15,;22.03,-13.39,;22.03,-11.84,;20.69,-11.06,;19.36,-11.84,)|
CN1CC2CCC1(CC2)[C@H](NC(=O)c1ccnc(c1F)C(F)(F)F)c1ccccc1 |r,wU:9.11,(7.01,-35.16,;7.01,-33.63,;5.68,-32.88,;5.68,-31.34,;7.01,-30.56,;8.34,-31.34,;8.34,-32.88,;7.74,-31.57,;6.66,-32.65,;9.66,-33.64,;9.66,-35.19,;10.99,-35.96,;12.33,-35.19,;10.99,-37.5,;9.65,-38.27,;9.65,-39.81,;10.99,-40.59,;12.33,-39.81,;12.33,-38.27,;13.66,-37.49,;13.67,-40.57,;13.67,-42.12,;15,-39.79,;15,-41.34,;11,-32.87,;12.33,-33.65,;13.67,-32.88,;13.67,-31.33,;12.33,-30.56,;10.99,-31.33,)|
CN1CC2CCC1(CC2)C(NC(=O)c1cccc(c1Cl)C(F)(F)F)c1cccnc1 |(18.64,-24.01,;18.64,-22.45,;17.29,-21.68,;17.29,-20.11,;18.64,-19.31,;20,-20.11,;20,-21.68,;19.39,-20.34,;18.28,-21.45,;21.35,-22.46,;21.35,-24,;22.68,-24.77,;24.01,-24,;22.68,-26.31,;21.35,-27.07,;21.34,-28.6,;22.68,-29.38,;24.01,-28.6,;24,-27.07,;25.34,-26.3,;25.34,-29.36,;26.67,-30.13,;26.67,-28.59,;25.35,-30.91,;22.68,-21.69,;22.68,-20.15,;24,-19.39,;25.35,-20.15,;25.34,-21.69,;24.01,-22.46,)|
CCN1CC2CC1(C2)C(NC(=O)c1c(C)cccc1C)c1ccccc1 |(25.68,-27.98,;27.16,-27.5,;27.49,-25.97,;26.44,-24.81,;27.22,-23.46,;28.75,-23.78,;28.91,-25.33,;27.62,-24.96,;30.27,-26.11,;30.27,-27.64,;31.6,-28.42,;32.92,-27.65,;31.6,-29.96,;30.26,-30.71,;28.91,-29.93,;30.26,-32.25,;31.59,-33.03,;32.92,-32.25,;32.92,-30.71,;34.27,-29.93,;31.59,-25.34,;31.59,-23.8,;32.92,-23.04,;34.26,-23.81,;34.26,-25.34,;32.92,-26.11,)|
CC(C)N1C2CCC1(CC2)C(NC(=O)c1c(C)cccc1C)c1ccncc1 |TLB:1:3:5.6:8.9|
CN1CC2CCC1(CC2)C(NC(=O)c1c(C)cccc1C)c1ccc(cc1)S(=O)(=O)CC1CC1 |(8.01,-25.32,;8.01,-23.77,;6.66,-23,;6.66,-21.44,;8.01,-20.64,;9.36,-21.44,;9.36,-23,;8.75,-21.66,;7.65,-22.77,;10.7,-23.77,;10.7,-25.31,;12.03,-26.08,;13.35,-25.31,;12.03,-27.61,;10.7,-28.36,;9.35,-27.58,;10.69,-29.89,;12.02,-30.67,;13.35,-29.89,;13.35,-28.36,;14.69,-27.58,;12.03,-23.01,;12.02,-21.48,;13.35,-20.72,;14.68,-21.48,;14.68,-23.01,;13.35,-23.78,;16.03,-20.7,;15.24,-19.35,;16.81,-19.35,;17.38,-21.48,;18.72,-20.7,;20.28,-20.69,;19.5,-19.34,)|
CN1CC2CCC1(CC2)C(NC(=O)c1cccc(c1Cl)C(F)(F)F)c1ccncc1 |(5.54,-23.59,;5.54,-22.03,;4.18,-21.26,;4.18,-19.69,;5.54,-18.89,;6.89,-19.69,;6.89,-21.26,;6.28,-19.92,;5.18,-21.03,;8.25,-22.04,;8.25,-23.58,;9.58,-24.35,;10.91,-23.58,;9.58,-25.89,;8.24,-26.65,;8.24,-28.18,;9.57,-28.96,;10.9,-28.18,;10.9,-26.65,;12.23,-25.88,;12.24,-28.94,;13.57,-29.71,;13.57,-28.17,;12.24,-30.49,;9.58,-21.27,;9.57,-19.74,;10.9,-18.97,;12.24,-19.74,;12.24,-21.27,;10.91,-22.04,)|
CN1CC2CCC1(CC2)C(NC(=O)c1cccc(c1Cl)C(F)(F)F)c1cccc(Br)c1 |(5.54,-23.59,;5.54,-22.03,;4.18,-21.26,;4.18,-19.69,;5.54,-18.89,;6.89,-19.69,;6.89,-21.26,;6.28,-19.92,;5.18,-21.03,;8.25,-22.04,;8.25,-23.58,;9.58,-24.35,;10.91,-23.58,;9.58,-25.89,;8.24,-26.65,;8.24,-28.18,;9.57,-28.96,;10.9,-28.18,;10.9,-26.65,;12.23,-25.88,;12.24,-28.94,;13.57,-29.71,;13.57,-28.17,;12.24,-30.49,;9.58,-21.27,;10.91,-22.04,;12.24,-21.27,;12.24,-19.74,;10.9,-18.97,;10.9,-17.41,;9.57,-19.74,)|
CN1CC2CCC1(CC2)C(NC(=O)c1cccc(c1Cl)C(F)(F)F)c1ccccc1 |(8.69,-30.27,;8.69,-28.71,;7.34,-27.94,;7.34,-26.37,;8.69,-25.57,;10.05,-26.37,;10.05,-27.94,;9.44,-26.6,;8.33,-27.71,;11.4,-28.72,;11.4,-30.26,;12.73,-31.03,;14.06,-30.26,;12.73,-32.57,;11.39,-33.33,;11.39,-34.86,;12.73,-35.64,;14.06,-34.86,;14.05,-33.33,;15.39,-32.56,;15.39,-35.62,;16.72,-36.39,;16.72,-34.85,;15.4,-37.17,;12.73,-27.95,;12.73,-26.41,;14.05,-25.65,;15.4,-26.42,;15.39,-27.95,;14.06,-28.72,)|
COc1cncc(Cl)c1C(=O)N[C@H](c1ccccc1)C12CCC(CC1)CN2C |r|
CSc1ncccc1C(=O)N[C@H](c1ccccc1)C12CCC(CC1)CN2C |r|
CCCCC(NC(=O)c1cccc(c1Cl)C(F)(F)F)C12CCC(CC1)CN2C
Cc1cccc(C)c1C(=O)NC(c1ccccc1)C12CC(C1)CN2 |(28.91,-29.93,;30.26,-30.71,;30.26,-32.25,;31.59,-33.03,;32.92,-32.25,;32.92,-30.71,;34.27,-29.93,;31.6,-29.96,;31.6,-28.42,;32.92,-27.65,;30.27,-27.64,;30.27,-26.11,;31.59,-25.34,;31.59,-23.8,;32.92,-23.04,;34.26,-23.81,;34.26,-25.34,;32.92,-26.11,;28.91,-25.33,;28.75,-23.78,;27.22,-23.46,;27.62,-24.96,;26.44,-24.81,;27.49,-25.97,)|
COC(C)c1ccc(N2CCN(CC2)C(=O)c2cc(ccc2-c2ccc(F)cc2)S(C)(=O)=O)c(F)c1
CS(=O)(=O)c1ccc(-c2ccc(F)cc2)c(c1)C(=O)N1CCN(CC1)c1ccc(N)cc1F
Fc1ccc(cc1)C(CCCN1CCC(Cc2nc3cccnc3n2Cc2cccs2)CC1)c1ccc(F)cc1
CCOCCn1c(CN2CCN(CCCC(c3ccc(F)cc3)c3ccc(F)cc3)CC2)nc2cccnc12
Cn1cc(nn1)S(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(Cl)cc2Cl)CCCCC1
CS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(N)cccc2Cl)CCCCC1
Cn1cc(nn1)S(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(Cl)cc2Cl)CCC(F)(F)CC1
CCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(Cl)cccc2OC(F)(F)F)CCC(F)(F)CC1
CC(NC(=O)c1ccc(cc1Cl)C(F)(F)F)C1(CCC(F)(F)CC1)N1CCN(CC1)S(=O)(=O)c1cn(C)nn1
Cn1cc(nn1)S(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(F)cc2Cl)CCC(F)(F)CC1
Cn1cc(nn1)S(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(Cl)cccc2OC(F)(F)F)CCC(F)(F)CC1
Cn1cnc(c1)S(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(cc2Cl)C(F)(F)F)CCC(F)(F)CC1
Cn1cnc(c1)S(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(Cl)cc2Cl)CCC(F)(F)CC1
Cn1cnc(c1)S(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(Cl)cccc2OC(F)(F)F)CCC(F)(F)CC1
Cn1cnc(c1)S(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(F)cccc2F)CCC(F)(F)CC1
Cn1cnc(c1)S(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(Cl)cc2Cl)CCCCC1
Clc1ccc(C(=O)NCC2(CCCCC2)N2CCN(CC2)S(=O)(=O)C2CCC2)c(Cl)c1
Nc1cccc(Cl)c1C(=O)NCC1(CCCCC1)N1CCN(CC1)S(=O)(=O)Cc1ccccc1
CCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(C)cc(F)cc2OC)CCC(F)(F)CC1
CCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(cc2C(F)(F)F)C(F)(F)F)CCC(F)(F)CC1
CCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(cc2Cl)C(F)(F)F)CCC(F)(F)CC1
CCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(Cl)cc2Cl)CCC(F)(F)CC1
CCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(Cl)cccc2Cl)CCC(F)(F)CC1
Cn1cc(nn1)S(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(cc2C(F)(F)F)C(F)(F)F)CCC(F)(F)CC1
Cn1cc(nn1)S(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(Cl)cccc2Cl)CCC(F)(F)CC1
Cn1cnc(c1)S(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(Cl)cccc2Cl)CCC(F)(F)CC1
Clc1ccc(C(=O)NCC2(CCCCC2)N2CCN(CC2)S(=O)(=O)CC2CC2)c(Cl)c1
CC(C)CS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(N)cccc2Cl)CCCCC1
CCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(F)cc2Cl)CCC(F)(F)CC1
Cn1cc(nn1)S(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(cc2Cl)C(F)(F)F)CCC(F)(F)CC1
Cn1cc(cn1)S(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(Cl)cc2Cl)CCCCC1
CCS(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(N)cccc2Cl)CCCCC1
Nc1cccc(Cl)c1C(=O)NCC1(CCCCC1)N1CCN(CC1)S(=O)(=O)c1ccccc1
Cn1cc(nn1)S(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2c(F)cccc2F)CCC(F)(F)CC1
Cn1cnc(c1)S(=O)(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(F)cc2Cl)CCC(F)(F)CC1
O=c1[nH]c2CN(Cc3ccccc3)CCc2c(=O)[nH]1
OC(=O)CCSc1[nH]c(=O)nc2[nH]c(=O)[nH]c12
OC(=O)CCCCSc1ncnc2[nH]c(=O)[nH]c12
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@@H](CC(C)C)C(O)=O |r|
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@H](Cc1ccccc1)C(O)=O |r|
CCCCCCCCC=C/CCCCCCCC(=O)N[C@@H](CCCCN)C(O)=O
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@@H](CC(O)=O)C(O)=O |r|
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@@H](CCC(O)=O)C(O)=O |r|
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@H](CCC(O)=O)C(O)=O |r|
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@@H](CCc1ccccc1)C(O)=O |r|
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@H](CCc1ccccc1)C(O)=O |r|
CCCCCCCCC=C/CCCCCCCC(=O)N[C@@H](Cc1cnc[nH]1)C(O)=O
CCCCCCCCC=C/CCCCCCCC(=O)N[C@H](Cc1cnc[nH]1)C(O)=O
CCCCCCCCC=C/CCCCCCCC(=O)N[C@H](CCCNC(N)=N)C(O)=O
CCCCCCCCC=C/CCCCCCCC(=O)N[C@H](CCCCN)C(O)=O
CCCCCCCCC=C/CCCCCCCC(=O)N[C@@H](CCCN)C(O)=O
CCCCCCCCC=C/CCCCCCCC(=O)N[C@@H](CN)C(O)=O
CCCCCCCCC=C/CCCCCCCC(=O)NCCCCCN
CCCCCCCC\C=C/CCCCCCCC(=O)NCC(O)=O
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@H](C)C(O)=O |r|
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@@H](C(C)C)C(O)=O |r|
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@H](C(C)C)C(O)=O |r|
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@H](CCSC)C(O)=O |r|
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@@H](CCCC)C(O)=O |r|
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@H](CO)C(O)=O |r|
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@H](CC(O)=O)C(O)=O |r|
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@@H](CC(N)=O)C(O)=O |r|
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(O)=O |r|
CCCCCCCCC=C/CCCCCCCC(=O)N[C@@H](CCCNC(N)=N)C(O)=O
CCCCCCCCC=C/CCCCCCCC(=O)N[C@@H](CCN)C(O)=O
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@@H](C)C(O)=O
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@H](CC(C)C)C(O)=O |r|
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@@H](CO)C(O)=O |r|
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(O)=O |r|
CCCCCCCCC=C/CCCCCCCC(=O)N[C@@H](CCCCN)C(=O)OC
CCCCCCCC\C=C/CCCCCCCC(=O)N[C@@H](CCSC)C(O)=O |r|
C[C@H](Oc1ccc(C#N)c(Cl)c1C(=O)N1Cc2cn(nc2C1)-c1ccc(F)cn1)C(F)(F)F |r|
COc1c(ccc(O[C@@H](C)C(F)(F)F)c1C(=O)N1Cc2cn(nc2C1)-c1ccc(F)cn1)C#N |r|
COc1c(ccc(O[C@@H](C)C(F)(F)F)c1C(=O)N1Cc2cn(nc2C1)-c1ccc(F)cn1)S(C)(=O)=O |r|
COc1c(ccc(O[C@@H](C)C(F)(F)F)c1C(=O)N1CC(C1)c1ccc(cc1)C(F)(F)F)S(C)(=O)=O |r|
COc1c(ccc(O[C@@H](C)C(F)(F)F)c1C(=O)N1CC(C1)c1ccccc1)S(C)(=O)=O |r|
COc1c(ccc(O[C@@H](C)C(F)(F)F)c1C(=O)N1CC(C1)c1ccc(cn1)C(F)(F)F)S(C)(=O)=O |r|
COc1c(ccc(O[C@@H](C)C(F)(F)F)c1C(=O)N1CC(C1)c1ncc(cc1F)C(F)(F)F)S(C)(=O)=O |r|
COc1c(ccc(O[C@@H](C)C(F)(F)F)c1C(=O)N1CC(C1)c1ncc(cc1Cl)C(F)(F)F)S(C)(=O)=O |r|
C[C@H](Oc1ccc(cc1C(=O)N1CC(C1)c1ccc(cc1)C(F)(F)F)S(C)(=O)=O)C(F)(F)F |r|