Affinity DataKi: 1nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: <1nM ΔG°: <-50.9kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 1.70nM ΔG°: -49.6kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 1.90nM ΔG°: -49.3kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 4nM ΔG°: -47.5kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 4.80nM ΔG°: -47.0kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 5.80nM ΔG°: -46.5kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 6.60nM ΔG°: -46.2kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 9.80nM ΔG°: -45.3kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 20nM ΔG°: -43.5kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 35.2nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 48nM ΔG°: -41.4kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 62nM ΔG°: -40.7kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 84nM ΔG°: -40.0kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 108nM ΔG°: -39.4kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 169nM ΔG°: -38.3kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 169nM ΔG°: -38.3kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 175nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 287nM ΔG°: -37.0kJ/molepH: 8.0 T: 2°CAssay Description:The enzyme assay was performed in a round-bottom 96-well plate. The enzyme was pre-incubated in the assay buffer in the presence of NADPH and inhibit...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of 11-beta-HSD2More data for this Ligand-Target Pair
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of human 11-beta-HSD1 expressed in HEK293 cells co-transfected with GRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of human 11-beta-HSD1 expressed in HEK293 cells co-transfected with GRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of human 11-beta-HSD1 expressed in HEK293 cells co-transfected with GRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of human 11-beta-HSD1 expressed in HEK293 cells co-transfected with GRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of human 11-beta-HSD1 expressed in HEK293 cells co-transfected with GRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair