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Found 273 with Last Name = 'fruzinski' and Initial = 'a'
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)
Affinity DataKi:  5.01nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187587(CHEMBL3827598)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187585(CHEMBL3827074)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187591(CHEMBL3827331)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187591(CHEMBL3827331)
Affinity DataKi:  109nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187588(CHEMBL3827201)
Affinity DataKi:  127nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187660(CHEMBL3828002)
Affinity DataKi:  131nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187584(CHEMBL3827187)
Affinity DataKi:  137nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187664(CHEMBL3828555)
Affinity DataKi:  172nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187592(CHEMBL3827301)
Affinity DataKi:  174nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187586(CHEMBL3827623)
Affinity DataKi:  175nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187662(CHEMBL3827267)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187660(CHEMBL3828002)
Affinity DataKi:  184nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221683(9-(4-hydroxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrah...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187605(CHEMBL3827298)
Affinity DataKi:  254nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187593(CHEMBL3827922)
Affinity DataKi:  268nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187590(CHEMBL3827583)
Affinity DataKi:  271nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187659(CHEMBL3827716)
Affinity DataKi:  297nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187591(CHEMBL3827331)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A3 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221697(1,3-dimethyl-9-phenethyl-6,7,8,9-tetrahydropyrimid...)
Affinity DataKi:  320nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221691(9-(2-(1H-indol-3-yl)ethyl)-1,3-dimethyl-6,7,8,9-te...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187664(CHEMBL3828555)
Affinity DataKi:  337nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187676(CHEMBL3828401)
Affinity DataKi:  338nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187589(CHEMBL3827859)
Affinity DataKi:  339nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187676(CHEMBL3828401)
Affinity DataKi:  347nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221703(9-(4-methoxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrah...)
Affinity DataKi:  370nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187674(CHEMBL3828658)
Affinity DataKi:  370nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187674(CHEMBL3828658)
Affinity DataKi:  464nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221681(9-(4-chlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahy...)
Affinity DataKi:  480nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187590(CHEMBL3827583)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187661(CHEMBL3828044)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187655(CHEMBL3827920)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187660(CHEMBL3828002)
Affinity DataKi:  518nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187587(CHEMBL3827598)
Affinity DataKi:  539nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine receptor A1 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187591(CHEMBL3827331)
Affinity DataKi:  546nMAssay Description:Displacement of [3H]MSX2 from recombinant human adenosine receptor A2a expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187589(CHEMBL3827859)
Affinity DataKi:  559nMAssay Description:Displacement of [3H]MSX2 from recombinant human adenosine receptor A2a expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187591(CHEMBL3827331)
Affinity DataKi:  566nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187666(CHEMBL3827653)
Affinity DataKi:  567nMAssay Description:Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187596(CHEMBL3827016)
Affinity DataKi:  585nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221694(9-phenethyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimid...)
Affinity DataKi:  590nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187660(CHEMBL3828002)
Affinity DataKi:  619nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A3 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221694(9-phenethyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimid...)
Affinity DataKi:  620nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221683(9-(4-hydroxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrah...)
Affinity DataKi:  630nMAssay Description:Displacement of [3H]MSX2 from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187676(CHEMBL3828401)
Affinity DataKi:  633nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A3 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187595(CHEMBL3828343)
Affinity DataKi:  645nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187599(CHEMBL3828237)
Affinity DataKi:  653nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187676(CHEMBL3828401)
Affinity DataKi:  658nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187585(CHEMBL3827074)
Affinity DataKi:  658nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine receptor A1 expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187674(CHEMBL3828658)
Affinity DataKi:  663nMAssay Description:Displacement of [3H]PSB-603 from recombinant human adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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