Affinity DataIC50: 6nMAssay Description:Inhibition of human DYRK1A at 3 uM in presence of ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of human wild type DYRK1A (M1 to S629) expressed in bacterial system by Ambit Kinomescan binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of DYRK1A (unknown origin) in presence of ATP at 15 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of DYRK1A (unknown origin) at 10 uM by ADP hunter plus assayMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 84nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 89nMAssay Description:Inhibition of human DYRK1A by Eu kinase activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 97nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 98nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of human wild type DYRK1A (M1 to S629) expressed in bacterial system by Ambit Kinomescan binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 112nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 139nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 152nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 168nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 168nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 215nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 950nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: >8.30E+3nMAssay Description:Inhibition of GSK3beta (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 9.41E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) at 1 uM by kinomescan methodMore data for this Ligand-Target Pair
Affinity DataKd: 185nMAssay Description:Binding affinity to DYRK1A (unknown origin) assessed as dissociation constant at 3 uMMore data for this Ligand-Target Pair
Affinity DataKd: 71nMAssay Description:Binding affinity to DYRK1A (unknown origin) assessed as dissociation constant at 3 uMMore data for this Ligand-Target Pair
Affinity DataKd: 7.30E+3nMAssay Description:Binding affinity to DYRK1A (unknown origin) assessed as dissociation constant by ADP hunter plus assayMore data for this Ligand-Target Pair
Affinity DataKd: 7.30E+3nMAssay Description:Binding affinity to DYRK1A (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair