Compile Data Set for Download or QSAR
maximum 50k data
Found 38 with Last Name = 'garcia-ocana' and Initial = 'a'
LigandPNGBDBM50597836(CHEMBL5186778)
Affinity DataIC50:  6nMAssay Description:Inhibition of human DYRK1A at 3 uM in presence of ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50597836(CHEMBL5186778)
Affinity DataIC50:  6nMAssay Description:Inhibition of human wild type DYRK1A (M1 to S629) expressed in bacterial system by Ambit Kinomescan binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50538083(CHEMBL4638292)
Affinity DataIC50:  6nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50511159(CHEMBL4550946)
Affinity DataIC50:  13nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
Affinity DataIC50:  13nMAssay Description:Inhibition of DYRK1A (unknown origin) in presence of ATP at 15 uMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50511162(CHEMBL4575812)
Affinity DataIC50:  14nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))TBA
LigandPNGBDBM50538083(CHEMBL4638292)
Affinity DataIC50:  16nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50511154(CHEMBL4442374)
Affinity DataIC50:  19nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50511152(CHEMBL4474836)
Affinity DataIC50:  25nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)
Affinity DataIC50:  27nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)
Affinity DataIC50:  27nMAssay Description:Inhibition of DYRK1A (unknown origin) at 10 uM by ADP hunter plus assayMore data for this Ligand-Target Pair
LigandPNGBDBM50511155(CHEMBL4456985)
Affinity DataIC50:  27nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50511150(CHEMBL4440790)
Affinity DataIC50:  39nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))TBA
LigandPNGBDBM50597836(CHEMBL5186778)
Affinity DataIC50:  40nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50538085(CHEMBL4634969)
Affinity DataIC50:  43nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50511164(CHEMBL4514653)
Affinity DataIC50:  56nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50511156(CHEMBL4521356)
Affinity DataIC50:  64nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50511161(CHEMBL4579529)
Affinity DataIC50:  74nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50511165(CHEMBL4563765)
Affinity DataIC50:  84nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50571728(CHEMBL4855547)
Affinity DataIC50:  89nMAssay Description:Inhibition of human DYRK1A by Eu kinase activity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50511158(CHEMBL4437998)
Affinity DataIC50:  97nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50511157(CHEMBL4552025)
Affinity DataIC50:  98nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50538083(CHEMBL4638292)
Affinity DataIC50:  100nMAssay Description:Inhibition of human wild type DYRK1A (M1 to S629) expressed in bacterial system by Ambit Kinomescan binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)
Affinity DataIC50: <100nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
LigandPNGBDBM50511160(CHEMBL4513287)
Affinity DataIC50:  112nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50511153(CHEMBL4564623)
Affinity DataIC50:  139nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50379523(CHEMBL2012558)
Affinity DataIC50:  152nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50511147(CHEMBL4476003)
Affinity DataIC50:  168nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50511151(CHEMBL4483653)
Affinity DataIC50:  168nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50511149(CHEMBL4438785)
Affinity DataIC50:  215nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50511148(CHEMBL4539999)
Affinity DataIC50:  950nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50511163(CHEMBL4528315)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))TBA
LigandPNGBDBM50367664(CHEMBL4066450)
Affinity DataIC50: >8.30E+3nMAssay Description:Inhibition of GSK3beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50466133(CHEMBL4292847 | US11547712, Compound 3-1)
Affinity DataIC50:  9.41E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) at 1 uM by kinomescan methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50466136(CHEMBL4292463 | US11547712, Compound 3-12)
Affinity DataKd:  185nMAssay Description:Binding affinity to DYRK1A (unknown origin) assessed as dissociation constant at 3 uMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50466137(CHEMBL4280328 | US11547712, Compound 3-15)
Affinity DataKd:  71nMAssay Description:Binding affinity to DYRK1A (unknown origin) assessed as dissociation constant at 3 uMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50466133(CHEMBL4292847 | US11547712, Compound 3-1)
Affinity DataKd:  7.30E+3nMAssay Description:Binding affinity to DYRK1A (unknown origin) assessed as dissociation constant by ADP hunter plus assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50466133(CHEMBL4292847 | US11547712, Compound 3-1)
Affinity DataKd:  7.30E+3nMAssay Description:Binding affinity to DYRK1A (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed