Affinity DataKi: 0.150nMAssay Description:Inhibition of cathepsin G (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Inhibition of human PR3 using ABZ-VADnVADYQ-EDDnp as substrate by FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Inhibition of human PR3 using ABZ-VADnVADYQ-EDDnp as substrate by FRET assayMore data for this Ligand-Target Pair
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
Faculty Of Chemistry Gdansk University
Curated by ChEMBL
Faculty Of Chemistry Gdansk University
Curated by ChEMBL
Affinity DataKi: 54.3nMAssay Description:Inhibition of human HAT by FRET assayMore data for this Ligand-Target Pair
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
Faculty Of Chemistry Gdansk University
Curated by ChEMBL
Faculty Of Chemistry Gdansk University
Curated by ChEMBL
Affinity DataKi: 112nMAssay Description:Inhibition of human HAT by FRET assayMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Centre D'Etude Des Pathologies Respiratoires And Universit£
Curated by ChEMBL
Centre D'Etude Des Pathologies Respiratoires And Universit£
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Faculty Of Chemistry Gdansk University
Curated by ChEMBL
Faculty Of Chemistry Gdansk University
Curated by ChEMBL
Affinity DataKi: 973nMAssay Description:Inhibition of human matriptase by FRET assayMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Faculty Of Chemistry Gdansk University
Curated by ChEMBL
Faculty Of Chemistry Gdansk University
Curated by ChEMBL
Affinity DataKi: 1.71E+3nMAssay Description:Inhibition of human matriptase by FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.60E+3nMAssay Description:Inhibition of human PR3 using ABZ-VADnVADYQ-EDDnp as substrate by FRET assayMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
Centre D'Etude Des Pathologies Respiratoires And Universit£
Curated by ChEMBL
Centre D'Etude Des Pathologies Respiratoires And Universit£
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of human cathepsin CMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Centre D'Etude Des Pathologies Respiratoires And Universit£
Curated by ChEMBL
Centre D'Etude Des Pathologies Respiratoires And Universit£
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair