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Found 11 with Last Name = 'lesner' and Initial = 'a'
TargetCathepsin G(Homo sapiens (Human))
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM21737(2-[(1R,4S,7S,13S,19S,22S,25S,28S,31R,34S,40S,43S,4...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of cathepsin G (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50263166(CHEMBL4071346)
Affinity DataKi:  5.40nMAssay Description:Inhibition of human PR3 using ABZ-VADnVADYQ-EDDnp as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50263172(CHEMBL4085013)
Affinity DataKi:  21nMAssay Description:Inhibition of human PR3 using ABZ-VADnVADYQ-EDDnp as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
Faculty Of Chemistry Gdansk University

Curated by ChEMBL
LigandPNGBDBM50323871((6S,9S,12S,15S)-1,20-diamino-12-(3-amino-3-oxoprop...)
Affinity DataKi:  54.3nMAssay Description:Inhibition of human HAT by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
Faculty Of Chemistry Gdansk University

Curated by ChEMBL
LigandPNGBDBM50323872((6S,9S,12S,15S)-1,19-diamino-9-(3-amino-3-oxopropy...)
Affinity DataKi:  112nMAssay Description:Inhibition of human HAT by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Centre D'Etude Des Pathologies Respiratoires And Universit£

Curated by ChEMBL
LigandPNGBDBM50084637(2,2-Dimethyl-propionic acid 4-[2-(carboxymethyl-ca...)
Affinity DataKi:  200nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Faculty Of Chemistry Gdansk University

Curated by ChEMBL
LigandPNGBDBM50323871((6S,9S,12S,15S)-1,20-diamino-12-(3-amino-3-oxoprop...)
Affinity DataKi:  973nMAssay Description:Inhibition of human matriptase by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Faculty Of Chemistry Gdansk University

Curated by ChEMBL
LigandPNGBDBM50323872((6S,9S,12S,15S)-1,19-diamino-9-(3-amino-3-oxopropy...)
Affinity DataKi:  1.71E+3nMAssay Description:Inhibition of human matriptase by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50263165(CHEMBL4102959)
Affinity DataKi:  3.60E+3nMAssay Description:Inhibition of human PR3 using ABZ-VADnVADYQ-EDDnp as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
Centre D'Etude Des Pathologies Respiratoires And Universit£

Curated by ChEMBL
LigandPNGBDBM50546373(CHEMBL4764657)
Affinity DataIC50:  15nMAssay Description:Inhibition of human cathepsin CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Centre D'Etude Des Pathologies Respiratoires And Universit£

Curated by ChEMBL
LigandPNGBDBM50084637(2,2-Dimethyl-propionic acid 4-[2-(carboxymethyl-ca...)
Affinity DataIC50:  44nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed