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Found 62 with Last Name = 'pokrovsky' and Initial = 'a'
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530468(CHEMBL4436247)
Affinity DataIC50:  90nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530468(CHEMBL4436247)
Affinity DataIC50:  90nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530462(CHEMBL4435210)
Affinity DataIC50:  100nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530462(CHEMBL4435210)
Affinity DataIC50:  100nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530469(CHEMBL4442276)
Affinity DataIC50:  110nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530469(CHEMBL4442276)
Affinity DataIC50:  110nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530467(CHEMBL4467521)
Affinity DataIC50:  190nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530467(CHEMBL4467521)
Affinity DataIC50:  190nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50110796((4-(6-amino-9H-purin-9-yl)cyclopent-2-enyloxy)meth...)
Affinity DataIC50:  200nMAssay Description:Inhibition of DNA synthesis by HIV reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530466(CHEMBL4447343)
Affinity DataIC50:  280nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530466(CHEMBL4447343)
Affinity DataIC50:  280nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50110797(9-[4-(Diphosphoryloxyphosphonylmethoxy)-cyclopent-...)
Affinity DataIC50:  300nMAssay Description:Inhibition of DNA synthesis by HIV reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530465(CHEMBL4460313)
Affinity DataIC50:  500nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530465(CHEMBL4460313)
Affinity DataIC50:  500nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530463(CHEMBL4577295)
Affinity DataIC50:  570nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530463(CHEMBL4577295)
Affinity DataIC50:  570nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50110801(CHEMBL23361 | P,P'-Bis {[4-(guanine-9-yl)cyclopent...)
Affinity DataIC50:  700nMAssay Description:Inhibition of DNA synthesis by HIV reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530472(CHEMBL4560013)
Affinity DataIC50:  710nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530472(CHEMBL4560013)
Affinity DataIC50:  710nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530464(CHEMBL4440022)
Affinity DataIC50:  950nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530464(CHEMBL4440022)
Affinity DataIC50:  950nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530461(CHEMBL4576273)
Affinity DataIC50:  1.49E+3nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530461(CHEMBL4576273)
Affinity DataIC50:  1.49E+3nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50110804(CHEMBL23358 | P,P'-Bis {[4-(adenine-9-yl)cyclopent...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of DNA synthesis by HIV reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530471(CHEMBL4592125)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530471(CHEMBL4592125)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530470(CHEMBL4539724)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530470(CHEMBL4539724)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for 8 mins by fl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530469(CHEMBL4442276)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of recombinant TDP1 H493R mutant (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530468(CHEMBL4436247)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of recombinant TDP1 H493R mutant (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530469(CHEMBL4442276)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of recombinant TDP1 H493R mutant (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530468(CHEMBL4436247)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of recombinant TDP1 H493R mutant (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50110800(CHEMBL23886 | P,P'-Bis {[4-(guanine-9-yl)cyclopent...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of DNA synthesis by HIV reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530467(CHEMBL4467521)
Affinity DataIC50:  9.30E+3nMAssay Description:Inhibition of recombinant TDP1 H493R mutant (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530467(CHEMBL4467521)
Affinity DataIC50:  9.30E+3nMAssay Description:Inhibition of recombinant TDP1 H493R mutant (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50110798(CHEMBL277903 | P,P'-Bis {[4-(adenine-9-yl)cyclopen...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of DNA synthesis by HIV reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50110799(CHEMBL280273 | P,P'-Bis {[4-(guanine-9-yl)cyclopen...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of DNA synthesis by HIV reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530462(CHEMBL4435210)
Affinity DataIC50:  1.93E+4nMAssay Description:Inhibition of recombinant TDP1 H493R mutant (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530462(CHEMBL4435210)
Affinity DataIC50:  1.93E+4nMAssay Description:Inhibition of recombinant TDP1 H493R mutant (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530472(CHEMBL4560013)
Affinity DataIC50:  1.99E+4nMAssay Description:Inhibition of recombinant TDP1 H493R mutant (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530472(CHEMBL4560013)
Affinity DataIC50:  1.99E+4nMAssay Description:Inhibition of recombinant TDP1 H493R mutant (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50110795(CHEMBL23428 | NA1 | P,P'-Bis {[4-(adenine-9-yl)cyc...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of DNA synthesis by HIV reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530464(CHEMBL4440022)
Affinity DataIC50:  2.41E+4nMAssay Description:Inhibition of recombinant TDP1 H493R mutant (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530464(CHEMBL4440022)
Affinity DataIC50:  2.41E+4nMAssay Description:Inhibition of recombinant TDP1 H493R mutant (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50110793(9-[4-(Difluoromethyldiphosphonyl)oxyphosphonylmeth...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of DNA synthesis by HIV reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50110802(9-[4-(Difluoromethyldiphosphonyl)oxyphosphonylmeth...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of DNA synthesis by HIV reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530466(CHEMBL4447343)
Affinity DataIC50:  3.41E+4nMAssay Description:Inhibition of recombinant TDP1 H493R mutant (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530466(CHEMBL4447343)
Affinity DataIC50:  3.41E+4nMAssay Description:Inhibition of recombinant TDP1 H493R mutant (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530465(CHEMBL4460313)
Affinity DataIC50:  3.92E+4nMAssay Description:Inhibition of recombinant TDP1 H493R mutant (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Siberian Branch of The Russian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50530465(CHEMBL4460313)
Affinity DataIC50:  3.92E+4nMAssay Description:Inhibition of recombinant TDP1 H493R mutant (unknown origin) using 5'-(5,6 FAM-aac gtc agg gtc ttc c-BHQ1)-3' as substrate measured every 55 secs for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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